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中文名称 英文名称 CAS号 化学式 结构式图片
—— Furan-2-carboxylic acid [5-[(6-dimethylamino-methylpyridin-2-ylmethyl)-carbamoyl]-2-(4-o-tolyl-piperazin-1-yl)-phenyl]-amide 1419870-23-7 C32H36N6O3
Furan-2-carboxylic acid [5-[(6-dimethylamino-methylpyridin-2-ylmethyl)-carbamoyl]-2-(4-o-tolyl-piperazin-1-yl)-phenyl]-amide
—— (S)-tert-butyl 2-(8-bromo-4,5-dihydrobenzo[2,3]oxepino[4,5-d]oxazol-2-yl)pyrrolidine-1-carboxylate 1422428-77-0 C20H23BrN2O4
(S)-tert-butyl 2-(8-bromo-4,5-dihydrobenzo[2,3]oxepino[4,5-d]oxazol-2-yl)pyrrolidine-1-carboxylate
—— 6-(5-isopropyl-2-methylphenyl)-4-((2R,4R)-4-methoxy-2-methylpiperidin-1-yl)-2-(3-methyl-1H-indol-4-yl)-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidine 1421249-23-1 C33H41N5O
6-(5-isopropyl-2-methylphenyl)-4-((2R,4R)-4-methoxy-2-methylpiperidin-1-yl)-2-(3-methyl-1H-indol-4-yl)-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidine
—— (S)-3-{3-[3-(2-fluoro-phenyl)-[1,2,4]oxadiazol-5-yl]-propionylamino}-3-(2-trifluoromethyl-phenyl)-propionic acid 1420834-18-9 C21H17F4N3O4
(S)-3-{3-[3-(2-fluoro-phenyl)-[1,2,4]oxadiazol-5-yl]-propionylamino}-3-(2-trifluoromethyl-phenyl)-propionic acid
—— 2-(5-chloro-2-methylphenyl)-4-(3,3-dimethylpiperidin-1-yl)-6-(5-isopropyl-2-methylphenyl)-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidine 1421249-86-6 C31H39ClN4
2-(5-chloro-2-methylphenyl)-4-(3,3-dimethylpiperidin-1-yl)-6-(5-isopropyl-2-methylphenyl)-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidine
—— N-(5-hydroxyadamantane-2-yl)-2-(2-methyl-N-methylphenylsulfonamido)-2-methylpropanamide 1422026-48-9 C22H32N2O4S
N-(5-hydroxyadamantane-2-yl)-2-(2-methyl-N-methylphenylsulfonamido)-2-methylpropanamide
—— (E)-N-[2-(pyridin-4-yl)phenyl]-5,5-bis[4-(trifluoromethyl)phenyl]-2,4-pentadienamide 1002124-17-5 C30H20F6N2O
(E)-N-[2-(pyridin-4-yl)phenyl]-5,5-bis[4-(trifluoromethyl)phenyl]-2,4-pentadienamide
—— 1-((1-(3-fluorophenyl)-3-(trifluoromethyl)-1H-pyrazol-5-yl)methyl)-3-(6-(2-hydroxyethylamino)pyridin-3-yl)urea 1419599-28-2 C19H18F4N6O2
1-((1-(3-fluorophenyl)-3-(trifluoromethyl)-1H-pyrazol-5-yl)methyl)-3-(6-(2-hydroxyethylamino)pyridin-3-yl)urea
—— (R)-4-((R)-1-(7-(4-(morpholinomethyl)phenyl)quinolin-5-yloxy)ethyl)pyrrolidin-2-one 1421340-12-6 C26H29N3O3
(R)-4-((R)-1-(7-(4-(morpholinomethyl)phenyl)quinolin-5-yloxy)ethyl)pyrrolidin-2-one
—— 8-(4-(3,4-difluorophenoxy)phenethoxy)-1-methyl-3,4-dihydro-1H-pyrimido[1,6-a]pyrimidin-6(2H)-one 1420369-72-7 C22H21F2N3O3
8-(4-(3,4-difluorophenoxy)phenethoxy)-1-methyl-3,4-dihydro-1H-pyrimido[1,6-a]pyrimidin-6(2H)-one
—— (2E,4Z)-5-[6-([1,4]oxazepan-4-yl)pyridin-3-yl]-5-[4-(trifluoromethyl)phenyl]-2,4-pentadienoic acid 1002128-51-9 C22H21F3N2O3
(2E,4Z)-5-[6-([1,4]oxazepan-4-yl)pyridin-3-yl]-5-[4-(trifluoromethyl)phenyl]-2,4-pentadienoic acid
—— (Z)-(3,4-difluorophenyl)[2-methyl-4-(1H,1'H-spiro[furo[3,4-c]pyridine-3,4'-piperidin]-1'-ylmethyl)phenyl]methanone O-methyloxime 1017599-55-1 C27H27F2N3O2
(Z)-(3,4-difluorophenyl)[2-methyl-4-(1H,1'H-spiro[furo[3,4-c]pyridine-3,4'-piperidin]-1'-ylmethyl)phenyl]methanone O-methyloxime
—— 2-{[(2,5-dichlorophenyl)oxy]acetyl}hydrazinecarbothioamide 1052694-58-2 C9H9Cl2N3O2S
2-{[(2,5-dichlorophenyl)oxy]acetyl}hydrazinecarbothioamide
—— (E)-N-(isoquinolin-5-yl)-5,5-bis(2-methylphenyl)-2,4-pentadienamide 1002123-56-9 C28H24N2O
(E)-N-(isoquinolin-5-yl)-5,5-bis(2-methylphenyl)-2,4-pentadienamide
—— 4-(3-fluoro-4-methylbenzyloxy)benzaldehyde 1187212-33-4 C15H13FO2
4-(3-fluoro-4-methylbenzyloxy)benzaldehyde
—— 2-(4-(benzyloxy)phenyl)-3-(2-chloropyrimidin-4-yl)-6-fluoropyrazolo[1,5-a]pyridine 1257078-93-5 C24H16ClFN4O
2-(4-(benzyloxy)phenyl)-3-(2-chloropyrimidin-4-yl)-6-fluoropyrazolo[1,5-a]pyridine
—— (2E,4E)-5-(4-chlorophenyl)-5-(4-ethoxyphenyl)-N-(3-hydroxy-1,2,3,4-tetrahydroquinolin-5-yl)-2,4-pentadienamide monohydrochloride 1002125-00-9 C28H27ClN2O3*ClH
(2E,4E)-5-(4-chlorophenyl)-5-(4-ethoxyphenyl)-N-(3-hydroxy-1,2,3,4-tetrahydroquinolin-5-yl)-2,4-pentadienamide monohydrochloride
—— tert-butyl 4-(2-(diphenylmethyleneaminooxy)ethoxy)piperidine-1-carboxylate 1190365-40-2 C25H32N2O4
tert-butyl 4-(2-(diphenylmethyleneaminooxy)ethoxy)piperidine-1-carboxylate
—— N-(adamantane-2-yl)-2-methyl-2-(3-nitrophenylsulfonamido)propanamide 1422025-08-8 C20H27N3O5S
N-(adamantane-2-yl)-2-methyl-2-(3-nitrophenylsulfonamido)propanamide
—— methyl (2E)-2-[2-[[1-[3-(2,2-difluoroethenyl)phenyl]ethylideneamino]oxymethyl]phenyl]-2-methoxyiminoacetate 1159342-17-2 C21H20F2N2O4
methyl (2E)-2-[2-[[1-[3-(2,2-difluoroethenyl)phenyl]ethylideneamino]oxymethyl]phenyl]-2-methoxyiminoacetate
—— 2-(3,5-dimethylisoxazol-4-yl)-4'-hydroxy-5-propyl-[1,1'-biphenyl]-3-carboxamide 1422018-31-2 C21H22N2O3
2-(3,5-dimethylisoxazol-4-yl)-4'-hydroxy-5-propyl-[1,1'-biphenyl]-3-carboxamide
—— (R)-2-(3,5-dimethyl-1H-indazol-4-yl)-4-(4-methoxy-3,3-dimethylpiperidin-1-yl)-6-(2-methyl-5-(trifluoromethyl)phenyl)-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidine 1421250-41-0 C32H37F3N6O
(R)-2-(3,5-dimethyl-1H-indazol-4-yl)-4-(4-methoxy-3,3-dimethylpiperidin-1-yl)-6-(2-methyl-5-(trifluoromethyl)phenyl)-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidine
—— (4-methyl-1,4-diazepan-1-yl)-[5-[(4-pyridin-2-ylpyrimidin-2-yl)amino]-1H-indol-2-yl]methanone 1391600-02-4 C24H25N7O
(4-methyl-1,4-diazepan-1-yl)-[5-[(4-pyridin-2-ylpyrimidin-2-yl)amino]-1H-indol-2-yl]methanone
—— N-(3-bromo-5-fluoro-2-methyl-phenyl)-4-dimethylamino-benzamide 1418128-82-1 C16H16BrFN2O
N-(3-bromo-5-fluoro-2-methyl-phenyl)-4-dimethylamino-benzamide
—— N-((2,4-dimethylphenyl)(phenyl)methyl)-2-(2-(pyridin-4-yl)benzo[d]oxazol-5-yl)acetamide 1422168-48-6 C29H25N3O2
N-((2,4-dimethylphenyl)(phenyl)methyl)-2-(2-(pyridin-4-yl)benzo[d]oxazol-5-yl)acetamide
—— (R)-1-(2-(3,5-dimethyl-1H-indazol-4-yl)-6-(5-methoxy-2-methylphenyl)-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-yl)-N,N-dimethylpyrrolidin-3-amine 1421250-62-5 C30H37N7O
(R)-1-(2-(3,5-dimethyl-1H-indazol-4-yl)-6-(5-methoxy-2-methylphenyl)-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-yl)-N,N-dimethylpyrrolidin-3-amine
—— (S)-3-(2,3-dichloro-phenyl)-3-{[2-(2-fluoro-phenyl)-5-methyl-oxazole-4-carbonyl]-amino}-propionic acid 1420834-02-1 C20H15Cl2FN2O4
(S)-3-(2,3-dichloro-phenyl)-3-{[2-(2-fluoro-phenyl)-5-methyl-oxazole-4-carbonyl]-amino}-propionic acid
—— 1-((2-(3-fluorophenyl)-6-(trifluoromethyl)pyridin-3-yl)methyl)-3-(oxazolo[5,4-b]pyridin-6-yl)urea 1421428-57-0 C20H13F4N5O2
1-((2-(3-fluorophenyl)-6-(trifluoromethyl)pyridin-3-yl)methyl)-3-(oxazolo[5,4-b]pyridin-6-yl)urea
—— (R)-2-fluoro-N-(1-(methyl(propyl)amino)propan-2-yl)-4-(5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl)benzamide 1418293-27-2 C17H20F4N4O2
(R)-2-fluoro-N-(1-(methyl(propyl)amino)propan-2-yl)-4-(5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl)benzamide
—— (E)-(5-fluoropyridin-2-yl)[6-(1H,1'H-spiro[furo[3,4-c]pyridine-3,4'-piperidin]-1'-ylmethyl)pyridin-3-yl]methanone O-methyloxime 1017599-59-5 C24H24FN5O2
(E)-(5-fluoropyridin-2-yl)[6-(1H,1'H-spiro[furo[3,4-c]pyridine-3,4'-piperidin]-1'-ylmethyl)pyridin-3-yl]methanone O-methyloxime
—— 2-cyclopropyl-N-[2-[4-(2-methylphenyl)piperazin-1-yl]-5-(1-phenylethylcarbamoyl)phenyl]-1,3-oxazole-4-carboxamide 1419868-98-6 C33H35N5O3
2-cyclopropyl-N-[2-[4-(2-methylphenyl)piperazin-1-yl]-5-(1-phenylethylcarbamoyl)phenyl]-1,3-oxazole-4-carboxamide
—— 2-[4-(5-chloropyridin-2-yl)piperazine-1-carbonyl]pyrrolo[1,2-a]quinazolin-5(4H)-one 1417561-99-9 C21H18ClN5O2
2-[4-(5-chloropyridin-2-yl)piperazine-1-carbonyl]pyrrolo[1,2-a]quinazolin-5(4H)-one
—— [4-(3-cyclopropyl-5-methylpyridin-2-yl)piperazin-1-yl](2-fluoro-4-iodophenyl)methanone 1346124-11-5 C20H21FIN3O
[4-(3-cyclopropyl-5-methylpyridin-2-yl)piperazin-1-yl](2-fluoro-4-iodophenyl)methanone
—— (R)-6-(5-chloro-2-methylphenyl)-2-(3-methyl-1H-indol-4-yl)-4-(3-methyl-4-(oxetan-3-yl)piperazin-1-yl)-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidine 1421250-95-4 C31H35ClN6O
(R)-6-(5-chloro-2-methylphenyl)-2-(3-methyl-1H-indol-4-yl)-4-(3-methyl-4-(oxetan-3-yl)piperazin-1-yl)-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidine
—— furan-2-carboxylic acid [5-(1-methanesulfonyl-piperidin-4-ylaminoformyl)-2-(4-o-tolueneyl-piperazin-1-yl)-phenyl]-amide 1419866-62-8 C29H35N5O5S
furan-2-carboxylic acid [5-(1-methanesulfonyl-piperidin-4-ylaminoformyl)-2-(4-o-tolueneyl-piperazin-1-yl)-phenyl]-amide
—— (R)-2-(2,4-Dichloro-phenyl)-N-((R)-2,3-dihydro-furo[2,3-b]pyridin-3-yl)-propionamide 1421619-71-7 C16H14Cl2N2O2
(R)-2-(2,4-Dichloro-phenyl)-N-((R)-2,3-dihydro-furo[2,3-b]pyridin-3-yl)-propionamide
—— 8-chloro-2-(3-fluorophenyl)-3-[(1S)-1-[(2-methyl-[1,3]thiazolo[5,4-d]pyrimidin-7-yl)amino]ethyl]isoquinolin-1-one 1420829-77-1 C23H17ClFN5OS
8-chloro-2-(3-fluorophenyl)-3-[(1S)-1-[(2-methyl-[1,3]thiazolo[5,4-d]pyrimidin-7-yl)amino]ethyl]isoquinolin-1-one
—— N-[5-[[3-[(dimethylamino)methyl]phenyl]methylcarbamoyl]-2-[4-(2-methylphenyl)piperazin-1-yl]phenyl]furan-2-carboxamide 1419868-82-8 C33H37N5O3
N-[5-[[3-[(dimethylamino)methyl]phenyl]methylcarbamoyl]-2-[4-(2-methylphenyl)piperazin-1-yl]phenyl]furan-2-carboxamide
—— 1-(1-(2-hydroxyethyl)-1H-indazol-4-yl)-3-((2-(4-methylpiperidin-1-yl)-6-(trifluoromethyl)pyridin-3-yl)methyl)urea 1421429-01-7 C23H27F3N6O2
1-(1-(2-hydroxyethyl)-1H-indazol-4-yl)-3-((2-(4-methylpiperidin-1-yl)-6-(trifluoromethyl)pyridin-3-yl)methyl)urea
—— [3-(4-methylpiperazin-1-yl)azetidin-1-yl]-[5-[(4-pyridin-2-ylpyrimidin-2-yl)amino]-1H-indol-2-yl]methanone 1391600-57-9 C26H28N8O
[3-(4-methylpiperazin-1-yl)azetidin-1-yl]-[5-[(4-pyridin-2-ylpyrimidin-2-yl)amino]-1H-indol-2-yl]methanone
—— N-(adamantane-2-yl)-2-methyl-2-(2-bromophenylsulfonamido)propanamide 1422024-45-0 C20H27BrN2O3S
N-(adamantane-2-yl)-2-methyl-2-(2-bromophenylsulfonamido)propanamide
—— 2-[4-(4-trifluoromethylphenyl)piperazine-1-carbonyl]pyrrolo[1,2-a]quinazolin-5(4H)-one 1417561-98-8 C23H19F3N4O2
2-[4-(4-trifluoromethylphenyl)piperazine-1-carbonyl]pyrrolo[1,2-a]quinazolin-5(4H)-one
—— 5-(2-aminopyrimidin-4-yl)-2-(5-chloro-2-methylphenyl)-4-({4-[(4-methylpiperazin-1-yl)carbonyl]phenyl}ethynyl)-1H-pyrrole-3-carboxamide 1421582-39-9 C30H28ClN7O2
5-(2-aminopyrimidin-4-yl)-2-(5-chloro-2-methylphenyl)-4-({4-[(4-methylpiperazin-1-yl)carbonyl]phenyl}ethynyl)-1H-pyrrole-3-carboxamide
—— 2-(2-(3,5-dimethylisoxazol-4-yl)-1H-benzo[d]imidazol-6-yl)-N-((2,4-dimethylphenyl)(phenyl)methyl)acetamide 1422167-98-3 C29H28N4O2
2-(2-(3,5-dimethylisoxazol-4-yl)-1H-benzo[d]imidazol-6-yl)-N-((2,4-dimethylphenyl)(phenyl)methyl)acetamide
—— 2-Cyclopropyl-oxazole-4-carboxylic acid [5-(3-propionylamino-propylcarbamoyl)-2-(4-o-tolyl-piperazin-1-yl)-phenyl]-amide 1419869-97-8 C31H38N6O4
2-Cyclopropyl-oxazole-4-carboxylic acid [5-(3-propionylamino-propylcarbamoyl)-2-(4-o-tolyl-piperazin-1-yl)-phenyl]-amide
—— 4-amino-N-(3-methoxybenzyl)-7-(2-methoxy-4-pyridinyl)pyrrolo[2,1-f][1,2,4]triazine-5-carboxamide 1338049-65-2 C21H20N6O3
4-amino-N-(3-methoxybenzyl)-7-(2-methoxy-4-pyridinyl)pyrrolo[2,1-f][1,2,4]triazine-5-carboxamide
—— 2-(2-((R)-(2-amino-2-methylpropoxy)(3,5-dimethylisoxazol-4-yl)methyl)benzofuran-5-yl)-N-((S)-(3,5-dimethylpyridin-2-yl)(phenyl)methyl)acetamide 1422167-61-0 C34H38N4O4
2-(2-((R)-(2-amino-2-methylpropoxy)(3,5-dimethylisoxazol-4-yl)methyl)benzofuran-5-yl)-N-((S)-(3,5-dimethylpyridin-2-yl)(phenyl)methyl)acetamide
—— ethyl 3-(5-(2-(((S)-(2,4-dimethylphenyl)(phenyl)methyl)amino)-2-oxoethyl)benzofuran-2-yl)-3-(pyridin-4-yl)propanoate 1422170-96-4 C35H34N2O4
ethyl 3-(5-(2-(((S)-(2,4-dimethylphenyl)(phenyl)methyl)amino)-2-oxoethyl)benzofuran-2-yl)-3-(pyridin-4-yl)propanoate
—— 3-[(4-{[tert-butyl(dimethyl)silyl]oxy}phenyl)amino]-4-nitrobenzonitrile 1345688-19-8 C19H23N3O3Si
3-[(4-{[tert-butyl(dimethyl)silyl]oxy}phenyl)amino]-4-nitrobenzonitrile
—— [(2S,3S,4S,4aR)-3,4,7-trihydroxy-6-oxo-3,4,4a,5-tetrahydro-2H-[1,3]dioxolo[4,5-j]phenanthridin-2-yl] (4Z,7Z,10Z,13Z,16Z,19Z)-docosa-4,7,10,13,16,19-hexaenoate 1417784-11-2 C36H43NO8
[(2S,3S,4S,4aR)-3,4,7-trihydroxy-6-oxo-3,4,4a,5-tetrahydro-2H-[1,3]dioxolo[4,5-j]phenanthridin-2-yl] (4Z,7Z,10Z,13Z,16Z,19Z)-docosa-4,7,10,13,16,19-hexaenoate