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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-chloro-4-[3-(3-chloro-4-isopropoxy-phenyl)-[1,2,4]oxadiazol-5-yl]-pyridine 1035214-23-3 C16H13Cl2N3O2
2-chloro-4-[3-(3-chloro-4-isopropoxy-phenyl)-[1,2,4]oxadiazol-5-yl]-pyridine
—— N-hydroxy-4-methoxy-4-(4-(trifluoromethyl)phenyl)butanamide 1100155-95-0 C12H14F3NO3
N-hydroxy-4-methoxy-4-(4-(trifluoromethyl)phenyl)butanamide
—— 3-(4-Ethoxyanilino)-1-naphthalen-2-ylpropan-1-ol 1146191-05-0 C21H23NO2
3-(4-Ethoxyanilino)-1-naphthalen-2-ylpropan-1-ol
—— N-benzyl-N'-{2-[5-[2-(2-furyl)-1-methyl-1H-benzimidazol-5-yl]-2-oxo-2H-1,3,4-thiadiazin-3(6H)-yl]ethyl}urea 1151821-58-7 C25H24N6O3S
N-benzyl-N'-{2-[5-[2-(2-furyl)-1-methyl-1H-benzimidazol-5-yl]-2-oxo-2H-1,3,4-thiadiazin-3(6H)-yl]ethyl}urea
—— 1-methyl-N-[1-[3-(1-methylbenzimidazol-2-yl)phenyl]piperidin-4-yl]piperidine-4-carboxamide 1160831-28-6 C26H33N5O
1-methyl-N-[1-[3-(1-methylbenzimidazol-2-yl)phenyl]piperidin-4-yl]piperidine-4-carboxamide
—— N-[(4-chlorophenyl)methyl]-2-{4-[2-hydroxy-3-(2-methylbenzothiazol-5-yloxy)propyl]piperazinyl}acetamide 1082297-49-1 C24H29ClN4O3S
N-[(4-chlorophenyl)methyl]-2-{4-[2-hydroxy-3-(2-methylbenzothiazol-5-yloxy)propyl]piperazinyl}acetamide
—— (1R,2R)-1-hydroxy-2-methyl-1-(3,4,5-trifluorophenyl)pentan-3-one 1126928-37-7 C12H13F3O2
(1R,2R)-1-hydroxy-2-methyl-1-(3,4,5-trifluorophenyl)pentan-3-one
—— 3-(2-fluorobenzyl)-5-hexyl-1,3-oxazolidin-2-one 1174338-38-5 C16H22FNO2
3-(2-fluorobenzyl)-5-hexyl-1,3-oxazolidin-2-one
—— 1-oxo-2-(4-trifluoromethoxy-phenyl)-2,8-diaza-spiro[4.5]decane-8-carboxylic acid diethylamide 1255714-81-8 C20H26F3N3O3
1-oxo-2-(4-trifluoromethoxy-phenyl)-2,8-diaza-spiro[4.5]decane-8-carboxylic acid diethylamide
—— (Z)-3-cyclohexyl-5-{[5-(3,4-difluorophenyl)furan-2-yl]methylene}imidazolidine-2,4-dione 1149337-77-8 C20H18F2N2O3
(Z)-3-cyclohexyl-5-{[5-(3,4-difluorophenyl)furan-2-yl]methylene}imidazolidine-2,4-dione
—— N-(4-piperazin-1-ylpyridin-3-yl)-2-pyridin-3-ylpyrimidine-4-carboxamide 1107624-93-0 C19H19N7O
N-(4-piperazin-1-ylpyridin-3-yl)-2-pyridin-3-ylpyrimidine-4-carboxamide
—— N-(2-chloro-5-(2-(methylamino)-1,3-benzothiazol-6-yl)-3-pyridinyl)-2-fluorobenzenesulfonamide 1112982-41-8 C19H14ClFN4O2S2
N-(2-chloro-5-(2-(methylamino)-1,3-benzothiazol-6-yl)-3-pyridinyl)-2-fluorobenzenesulfonamide
—— (S)-3-[3-(1H-tetrazol-1-yl)propionyl]amino-1-(4-chloro-5-isoquinolinesulfonyl)pyrrolidine 1055266-76-6 C17H18ClN7O3S
(S)-3-[3-(1H-tetrazol-1-yl)propionyl]amino-1-(4-chloro-5-isoquinolinesulfonyl)pyrrolidine
—— (R)-(4-(4-(4-fluorophenyl)phthalazin-1-yl)-3-methylpiperazin-1-yl)(phenyl)methanone 1095638-22-4 C26H23FN4O
(R)-(4-(4-(4-fluorophenyl)phthalazin-1-yl)-3-methylpiperazin-1-yl)(phenyl)methanone
—— 4-{[4-({2-[(methylsulfonyl)amino]benzyl}amino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}benzamide 1073156-34-9 C20H19F3N6O3S
4-{[4-({2-[(methylsulfonyl)amino]benzyl}amino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}benzamide
—— 1-[5-({4-[3-(6-methylpyridin-2-yl)prop-2-ynylidene]piperidin-1-yl}carbonyl)thien-2-yl]ethanone 1107618-83-6 C21H20N2O2S
1-[5-({4-[3-(6-methylpyridin-2-yl)prop-2-ynylidene]piperidin-1-yl}carbonyl)thien-2-yl]ethanone
—— [(1R)-1-[[(2S)-6-amino-2-[[(2S)-2-[[(2S)-6-amino-2-[[(2S)-3-amino-2-[[4-(4-chlorophenyl)benzoyl]amino]propanoyl]amino]hexanoyl]amino]propanoyl]amino]hexanoyl]amino]ethyl]boronic acid 1451205-72-3 C33H50BClN8O7
[(1R)-1-[[(2S)-6-amino-2-[[(2S)-2-[[(2S)-6-amino-2-[[(2S)-3-amino-2-[[4-(4-chlorophenyl)benzoyl]amino]propanoyl]amino]hexanoyl]amino]propanoyl]amino]hexanoyl]amino]ethyl]boronic acid
—— 5-(2-chloro-pyridin-4-yl)-4-chloromethyl-3-methyl-isoxazole 1030122-27-0 C10H8Cl2N2O
5-(2-chloro-pyridin-4-yl)-4-chloromethyl-3-methyl-isoxazole
—— 2-methyl-4-({4-[({3-[methyl(methylsulfonyl)amino]pyridin-2-yl}methyl)amino]-5-(trifluoromethyl)pyrimidin-2-yl}amino)benzamide 1073158-76-5 C21H22F3N7O3S
2-methyl-4-({4-[({3-[methyl(methylsulfonyl)amino]pyridin-2-yl}methyl)amino]-5-(trifluoromethyl)pyrimidin-2-yl}amino)benzamide
—— ((2S,5R)-4-(4-(4-chloro-2-fluorophenyl)phthalazin-1-yl)-2,5-dimethylpiperazin-1-yl)(phenyl)methanone 1095638-64-4 C27H24ClFN4O
((2S,5R)-4-(4-(4-chloro-2-fluorophenyl)phthalazin-1-yl)-2,5-dimethylpiperazin-1-yl)(phenyl)methanone
—— (4-chloro-3-methyl-phenyl)-[2-(4-trifluoromethyl-phenyl)-ethyl]-amine 1111734-69-0 C16H15ClF3N
(4-chloro-3-methyl-phenyl)-[2-(4-trifluoromethyl-phenyl)-ethyl]-amine
—— (+/-)-2-(2-amino-cyclobutyl)-8-chloro-4,5-dihydro-1H-pyrrolo[2,3-f]isoquinoline-3-carboxylic acid lactam 1105663-63-5 C16H14ClN3O
(+/-)-2-(2-amino-cyclobutyl)-8-chloro-4,5-dihydro-1H-pyrrolo[2,3-f]isoquinoline-3-carboxylic acid lactam
—— 4-(5-Ethyl-2-thiophen-3-yl-1,3-thiazol-4-yl)-2,2,6,6-tetramethyloxane-3,5-dione 1094621-60-9 C18H21NO3S2
4-(5-Ethyl-2-thiophen-3-yl-1,3-thiazol-4-yl)-2,2,6,6-tetramethyloxane-3,5-dione
—— 1-{8-[6-(thiazolo[4,5-b]pyridin-2-yloxy)-benzofuran-3-ylmethyl]-2,8-diaza-spiro[4.5]dec-2-yl}-ethanone 1256104-38-7 C25H26N4O3S
1-{8-[6-(thiazolo[4,5-b]pyridin-2-yloxy)-benzofuran-3-ylmethyl]-2,8-diaza-spiro[4.5]dec-2-yl}-ethanone
—— [3-(4-methoxybenzyloxy)-2-methylphenyl]-(1-methyl-1H-imidazo[4,5-c]pyridin-6-yl)amine 1449515-62-1 C22H22N4O2
[3-(4-methoxybenzyloxy)-2-methylphenyl]-(1-methyl-1H-imidazo[4,5-c]pyridin-6-yl)amine
—— 1-(2,2-dimethylpropyl)-3-methyl-5-[2-methyl-5-(piperazin-1-ylmethyl)phenyl]-1,3-dihydro-2H-imidazo[4,5-b]pyridin-2-one 1352426-61-9 C24H33N5O
1-(2,2-dimethylpropyl)-3-methyl-5-[2-methyl-5-(piperazin-1-ylmethyl)phenyl]-1,3-dihydro-2H-imidazo[4,5-b]pyridin-2-one
—— methyl 3-amino-4-{[(3,5-dichloro-2-pyridinyl)methyl]amino}benzoate 1168138-80-4 C14H13Cl2N3O2
methyl 3-amino-4-{[(3,5-dichloro-2-pyridinyl)methyl]amino}benzoate
—— methyl (1R,2R)-2-aminocyclobutane-1-carboxylate;2,2,2-trifluoroacetic acid 1453222-25-7 C2HF3O2*C6H11NO2
methyl (1R,2R)-2-aminocyclobutane-1-carboxylate;2,2,2-trifluoroacetic acid
—— (2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[4-(4-butylphenyl)benzoyl]amino]-6-[(2-methylpropan-2-yl)oxycarbonylamino]hexanoyl]amino]-6-[(2-methylpropan-2-yl)oxycarbonylamino]hexanoyl]amino]propanoyl]amino]-4-oxo-4-(tritylamino)butanoic acid 1451204-43-5 C65H83N7O11
(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[4-(4-butylphenyl)benzoyl]amino]-6-[(2-methylpropan-2-yl)oxycarbonylamino]hexanoyl]amino]-6-[(2-methylpropan-2-yl)oxycarbonylamino]hexanoyl]amino]propanoyl]amino]-4-oxo-4-(tritylamino)butanoic acid
—— 1-[4-(5'-chloro-5-fluoro-3-methyl-2,4'-bipyridin-2'-yl)piperazin-1-yl]-3-(methylsulfonyl)propan-1-one 1373615-71-4 C19H22ClFN4O3S
1-[4-(5'-chloro-5-fluoro-3-methyl-2,4'-bipyridin-2'-yl)piperazin-1-yl]-3-(methylsulfonyl)propan-1-one
—— N-[1-[(3,5-difluoropyridin-2-yl)methyl]pyrazol-3-yl]acetamide 1372891-73-0 C11H10F2N4O
N-[1-[(3,5-difluoropyridin-2-yl)methyl]pyrazol-3-yl]acetamide
—— (R)-tert-butyl 3-(2-(6-fluoroimidazo[1,2-a]pyridin-3-yl)-5-methoxypyrimidin-4-ylamino)piperidine-1-carboxylate 1313279-86-5 C22H27FN6O3
(R)-tert-butyl 3-(2-(6-fluoroimidazo[1,2-a]pyridin-3-yl)-5-methoxypyrimidin-4-ylamino)piperidine-1-carboxylate
—— 8-iodo-1-[(3S)-pyrrolidin-3-yl]imidazo[4,5-c]quinoline 1350734-15-4 C14H13IN4
8-iodo-1-[(3S)-pyrrolidin-3-yl]imidazo[4,5-c]quinoline
—— [1-fluoro-2-[5-(1H-indazol-4-yl)pyridin-2-yl]-1-phosphonoethyl]phosphonic acid 1254582-18-7 C14H14FN3O6P2
[1-fluoro-2-[5-(1H-indazol-4-yl)pyridin-2-yl]-1-phosphonoethyl]phosphonic acid
—— 3-[1-(5-fluoro-2-methoxypyridin-3-yl)ethoxy]-5-(5-methyl-1H-pyrazol-4-yl)pyridin-2-amine 1346815-27-7 C17H18FN5O2
3-[1-(5-fluoro-2-methoxypyridin-3-yl)ethoxy]-5-(5-methyl-1H-pyrazol-4-yl)pyridin-2-amine
—— N-(3,4-dimethoxyphenyl)-3-(4-methylpiperazin-1-yl)-3-oxo-2-phenyl-N-[2-(4-trifluoromethylphenyl)ethyl]propionamide 1059182-20-5 C31H34F3N3O4
N-(3,4-dimethoxyphenyl)-3-(4-methylpiperazin-1-yl)-3-oxo-2-phenyl-N-[2-(4-trifluoromethylphenyl)ethyl]propionamide
—— (3-chloro-4-difluoromethoxy-phenyl)-[2-(4-trifluoromethyl-phenyl)-ethyl]-amine 1111735-42-2 C16H13ClF5NO
(3-chloro-4-difluoromethoxy-phenyl)-[2-(4-trifluoromethyl-phenyl)-ethyl]-amine
—— (RS)-N-[(3-chlorophenyl)(1,3-thiazol-2-yl)methyl]-2-oxo-2-(1'H,3H-spiro[2-benzofuran-1,4'-piperidin]-1'-yl)ethanamine 1039166-11-4 C24H24ClN3O2S
(RS)-N-[(3-chlorophenyl)(1,3-thiazol-2-yl)methyl]-2-oxo-2-(1'H,3H-spiro[2-benzofuran-1,4'-piperidin]-1'-yl)ethanamine
—— 4-[3-{6-[3-bromo-5-(1,3-dimethyl-2,4-dioxo-1,2,3,4-tetrahydro-pyrimidin-5-yl)-phenoxy]-hexyl}-(2-(2-ethoxycarbonyl-ethyl)-phenoxy)]-butyric acid ethyl ester 1123158-51-9 C35H45BrN2O8
4-[3-{6-[3-bromo-5-(1,3-dimethyl-2,4-dioxo-1,2,3,4-tetrahydro-pyrimidin-5-yl)-phenoxy]-hexyl}-(2-(2-ethoxycarbonyl-ethyl)-phenoxy)]-butyric acid ethyl ester
—— rac-[4-(tetrahydro-furan-3-yloxy)-cyclohexyl]-acetic acid methyl ester 1114554-20-9 C13H22O4
rac-[4-(tetrahydro-furan-3-yloxy)-cyclohexyl]-acetic acid methyl ester
—— 1-[(2R)-2-[{2-oxo-2-(1'H,3H-spiro[2-benzofuran-1,4'-piperidin]-1'-yl)ethyl}amino]-2-phenylacetyl]pyrrolidin-3-ol 1039166-42-1 C26H31N3O4
1-[(2R)-2-[{2-oxo-2-(1'H,3H-spiro[2-benzofuran-1,4'-piperidin]-1'-yl)ethyl}amino]-2-phenylacetyl]pyrrolidin-3-ol
—— 2-methyl-8-nitro-4-(3-(trifluoromethyl)phenoxy)quinazoline 1449737-29-4 C16H10F3N3O3
2-methyl-8-nitro-4-(3-(trifluoromethyl)phenoxy)quinazoline
—— 2,6,12,16-tetramethylheptadecan-9-yl methanesulfonate 1450889-52-7 C22H46O3S
2,6,12,16-tetramethylheptadecan-9-yl methanesulfonate
—— 1-amino-7-(3-fluorophenyl)-N-[2-(4-hydroxy-1-piperidyl)ethyl]isoquinoline-4-carboxamide 1449277-42-2 C23H25FN4O2
1-amino-7-(3-fluorophenyl)-N-[2-(4-hydroxy-1-piperidyl)ethyl]isoquinoline-4-carboxamide
—— 2-(methylamino)-N-[6-[2-(4-methylphenyl)ethynyl]-5-(quinolin-5-yl)pyridin-2-yl]propanamide 1452571-88-8 C27H24N4O
2-(methylamino)-N-[6-[2-(4-methylphenyl)ethynyl]-5-(quinolin-5-yl)pyridin-2-yl]propanamide
—— N-(5-bromopyrazine-2-yl)-2,4,5-trifluorobenzamide 1373940-45-4 C11H5BrF3N3O
N-(5-bromopyrazine-2-yl)-2,4,5-trifluorobenzamide
—— 6-(3-methylbenzyl)-2-(methylthio)pyrido[4,3-d]pyrimidin-5(6H)-one 1452230-03-3 C16H15N3OS
6-(3-methylbenzyl)-2-(methylthio)pyrido[4,3-d]pyrimidin-5(6H)-one
—— 4-[(1R,3R,4R)-4-{[bis(4-fluorophenyl)methyl]carbamoyl}-3-(2-fluorophenyl)cyclohexyl]morpholine trifluoroacetate 1350710-92-7 C2HF3O2*C30H31F3N2O2
4-[(1R,3R,4R)-4-{[bis(4-fluorophenyl)methyl]carbamoyl}-3-(2-fluorophenyl)cyclohexyl]morpholine trifluoroacetate
—— 5-[7-[(5R)-5-(6-chloro-1,3-benzoxazol-2-yl)-4,5-dihydro-1,2-oxazol-3-yl]-3-(4-fluorophenyl)-4-oxoquinazolin-2-yl]pentanoic acid 1373275-89-8 C29H22ClFN4O5
5-[7-[(5R)-5-(6-chloro-1,3-benzoxazol-2-yl)-4,5-dihydro-1,2-oxazol-3-yl]-3-(4-fluorophenyl)-4-oxoquinazolin-2-yl]pentanoic acid
—— methyl 4-[1-[2,2-dimethylpropyl]-3-methyl-2-oxo-2,3-dihydro-1H-imidazo[4,5-b]pyridin-5-yl]-3-fluorobenzoate 1352421-91-0 C20H22FN3O3
methyl 4-[1-[2,2-dimethylpropyl]-3-methyl-2-oxo-2,3-dihydro-1H-imidazo[4,5-b]pyridin-5-yl]-3-fluorobenzoate