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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-Chloro-2-cyclopropyl-4-(2,5-dimethylthiophen-3-yl)-1,4-dihydropyrimidine 1449704-89-5 C13H15ClN2S
5-Chloro-2-cyclopropyl-4-(2,5-dimethylthiophen-3-yl)-1,4-dihydropyrimidine
—— 2-[7-(4-Bromopiperidin-1-yl)-5-methyl-2-phenylpyrazolo[1,5-a]pyrimidin-6-yl]-2-[(2-methylpropan-2-yl)oxy]acetic acid 1451006-49-7 C24H29BrN4O3
2-[7-(4-Bromopiperidin-1-yl)-5-methyl-2-phenylpyrazolo[1,5-a]pyrimidin-6-yl]-2-[(2-methylpropan-2-yl)oxy]acetic acid
—— 1-((E)-1-Methyl-3-trimethylsilanyloxy-allyl)-pyridinium; iodide 113345-48-5 C12H20NOSi*I
1-((E)-1-Methyl-3-trimethylsilanyloxy-allyl)-pyridinium; iodide
—— 2-chloro-5-(2,2,2-trifluoroethyl)spiro[8H-pteridine-7,1'-cyclobutane]-6-one 1452229-27-4 C11H10ClF3N4O
2-chloro-5-(2,2,2-trifluoroethyl)spiro[8H-pteridine-7,1'-cyclobutane]-6-one
—— (2S)-2-(tert-butoxy)-2-(2-(2'-fluoro-[1,1'-biphenyl]-3-yl)-5-methyl-7-(6-methyl-3-azabicyclo[4.1.0]heptan-3-yl)pyrazolo[1,5-a]pyrimidin-6-yl)acetic acid 1451006-91-9 C32H35FN4O3
(2S)-2-(tert-butoxy)-2-(2-(2'-fluoro-[1,1'-biphenyl]-3-yl)-5-methyl-7-(6-methyl-3-azabicyclo[4.1.0]heptan-3-yl)pyrazolo[1,5-a]pyrimidin-6-yl)acetic acid
—— 2-amino-N-[6-[2-(1,3-thiazol-5-yl)ethynyl]pyridin-2-yl]propanamide 1452572-85-8 C13H12N4OS
2-amino-N-[6-[2-(1,3-thiazol-5-yl)ethynyl]pyridin-2-yl]propanamide
—— 5-bromo-2-methoxy-N-(5-(thiazol-5-yl)pyridin-3-yl)benzenesulfonamide 1451272-32-4 C15H12BrN3O3S2
5-bromo-2-methoxy-N-(5-(thiazol-5-yl)pyridin-3-yl)benzenesulfonamide
—— ethyl 3-(4'-(2,6-difluorobenzamido)-6-methyl-[1,1'-biphenyl]-3-yl)-4,4-dimethyl-4,5-dihydroisoxazole-5-carboxylate 1373938-68-1 C28H26F2N2O4
ethyl 3-(4'-(2,6-difluorobenzamido)-6-methyl-[1,1'-biphenyl]-3-yl)-4,4-dimethyl-4,5-dihydroisoxazole-5-carboxylate
—— 5-[7-[5-[(4,5-dichloro-2-hydroxyphenyl)carbamoyl]-5-methyl-4H-1,2-oxazol-3-yl]-3-(4-fluorophenyl)-4-oxoquinazolin-2-yl]pentanoic acid 1373276-01-7 C30H25Cl2FN4O6
5-[7-[5-[(4,5-dichloro-2-hydroxyphenyl)carbamoyl]-5-methyl-4H-1,2-oxazol-3-yl]-3-(4-fluorophenyl)-4-oxoquinazolin-2-yl]pentanoic acid
—— 7-benzyl-6,7,8,9,10,11,12,14-octahydro-6,14-dioxo-5-phenyl[1,4]diazonino[2,1-g] [1,7]naphthyridine 183550-07-4 C27H25N3O2
7-benzyl-6,7,8,9,10,11,12,14-octahydro-6,14-dioxo-5-phenyl[1,4]diazonino[2,1-g] [1,7]naphthyridine
—— methyl 5-[4-(3,4-methylenedioxybenzylamino)-5,6-dimethylthieno[2,3-d]pyrimidin-2-yl]valerate 1098996-80-5 C22H25N3O4S
methyl 5-[4-(3,4-methylenedioxybenzylamino)-5,6-dimethylthieno[2,3-d]pyrimidin-2-yl]valerate
—— 3-[2'(S)-benzyl-3'-mercaptopropionyl]-4(R)-carboxy-5,5-dimethylthiazolidine 188636-45-5 C16H21NO3S2
3-[2'(S)-benzyl-3'-mercaptopropionyl]-4(R)-carboxy-5,5-dimethylthiazolidine
—— [((3S)-3-amino-3-carboxy)propyl][(4-phosphonomethoxyphenyl)hydroxymethyl]phosphinic acid 1413405-51-2 C12H19NO9P2
[((3S)-3-amino-3-carboxy)propyl][(4-phosphonomethoxyphenyl)hydroxymethyl]phosphinic acid
—— 5-{3-[bis(2-methoxyethyl)amino]prop-1-yn-1-yl}thiophene-2-sulfonamide 1599442-29-1 C13H20N2O4S2
5-{3-[bis(2-methoxyethyl)amino]prop-1-yn-1-yl}thiophene-2-sulfonamide
—— (1R,5R)-5-Benzyloxy-5-methyl-3-vinyl-cyclohex-2-enol 166757-87-5 C16H20O2
(1R,5R)-5-Benzyloxy-5-methyl-3-vinyl-cyclohex-2-enol
—— 2-amino-N-[6-[2-(furan-3-yl)ethynyl]pyridin-2-yl]propanamide 1452572-86-9 C14H13N3O2
2-amino-N-[6-[2-(furan-3-yl)ethynyl]pyridin-2-yl]propanamide
—— 4-(2,5-Dimethylthiophen-3-yl)-7-fluoro-2-methyl-1,4-dihydroquinazoline 1449705-03-6 C15H15FN2S
4-(2,5-Dimethylthiophen-3-yl)-7-fluoro-2-methyl-1,4-dihydroquinazoline
—— (7-bromo-5-chloro-6-((2,4-dichlorobenzyl)oxy)-1-benzofuran-3-yl)acetic acid 1452477-78-9 C17H10BrCl3O4
(7-bromo-5-chloro-6-((2,4-dichlorobenzyl)oxy)-1-benzofuran-3-yl)acetic acid
—— 5-[5-[1-[(benzo[b]thien-3-yl)methyl]-(3R)-piperidinyl]-1H-1,3,4-oxadiazol-2-yl]-3-(2-methyl-4-pyridinyl)-1H-indazole 1374352-51-8 C29H26N6OS
5-[5-[1-[(benzo[b]thien-3-yl)methyl]-(3R)-piperidinyl]-1H-1,3,4-oxadiazol-2-yl]-3-(2-methyl-4-pyridinyl)-1H-indazole
—— 2-(6-methyl-2-oxo-5-(6-(trifluoromethyl)-1H-indazol-4-yl)pyridin-1(2H)-yl)acetonitrile 1454299-02-5 C16H11F3N4O
2-(6-methyl-2-oxo-5-(6-(trifluoromethyl)-1H-indazol-4-yl)pyridin-1(2H)-yl)acetonitrile
—— 1-Amino-3-[4-chloro-2-fluoro-5-(6-chloro-5-nitro-4-pyrimidyloxy)phenyl]-6-trifluoro-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione 1099379-16-4 C15H6Cl2F4N6O5
1-Amino-3-[4-chloro-2-fluoro-5-(6-chloro-5-nitro-4-pyrimidyloxy)phenyl]-6-trifluoro-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
—— N-[4-(2-pyrrolidin-1-ylethoxy)phenyl]-5-[1-(thiophen-2-ylmethyl)pyrazol-4-yl]-[1,2,4]triazolo[1,5-a]pyridin-2-amine 1142941-81-8 C26H27N7OS
N-[4-(2-pyrrolidin-1-ylethoxy)phenyl]-5-[1-(thiophen-2-ylmethyl)pyrazol-4-yl]-[1,2,4]triazolo[1,5-a]pyridin-2-amine
—— 8-(2-chloro-benzenesulfonyl)-2-(3-chloro-4-trifluoromethyl-phenyl)-2,8-diaza-spiro[4.5]decan-1-one 1255714-42-1 C21H19Cl2F3N2O3S
8-(2-chloro-benzenesulfonyl)-2-(3-chloro-4-trifluoromethyl-phenyl)-2,8-diaza-spiro[4.5]decan-1-one
—— 4-[4-[[4-(cyclopropylamino)-3-methylsulfonyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl]amino]phenyl]-N,N-dimethylbenzenesulfonamide 1037478-91-3 C23H25N7O4S2
4-[4-[[4-(cyclopropylamino)-3-methylsulfonyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl]amino]phenyl]-N,N-dimethylbenzenesulfonamide
—— 3-methoxy-5,8-bis((methoxymethoxy)methyl)-6,7-bis(3-(methoxymethoxy)prop-1-yn-1-yl)isoquinoline 1224954-39-5 C26H33NO9
3-methoxy-5,8-bis((methoxymethoxy)methyl)-6,7-bis(3-(methoxymethoxy)prop-1-yn-1-yl)isoquinoline
—— 4-methoxy-2,6-bis(2-phenylsulfinyl-2-propenyl)phenol 139371-11-2 C25H24O4S2
4-methoxy-2,6-bis(2-phenylsulfinyl-2-propenyl)phenol
—— ethyl 7-amino-2-(4-methoxyphenyl)-5-phenyl-3,4-dihydroimidazo[1,5-b]pyridazine-4-carboxylate 1106668-19-2 C22H22N4O3
ethyl 7-amino-2-(4-methoxyphenyl)-5-phenyl-3,4-dihydroimidazo[1,5-b]pyridazine-4-carboxylate
—— 1-isoquinolin-5-ylmethanamine hydrochloride 1001906-56-4 C10H10N2*ClH
1-isoquinolin-5-ylmethanamine hydrochloride
—— tert-butyl 4-(2-((tert-butyldimethylsilyloxy)methyl)quinolin-7-yl)piperazine-1-carboxylate 1352640-57-3 C25H39N3O3Si
tert-butyl 4-(2-((tert-butyldimethylsilyloxy)methyl)quinolin-7-yl)piperazine-1-carboxylate
—— (1R,5R)-3,5,8,8-Tetramethyl-2-oxo-3-aza-bicyclo[3.2.1]octane-1-carboxylic acid 183850-83-1 C12H19NO3
(1R,5R)-3,5,8,8-Tetramethyl-2-oxo-3-aza-bicyclo[3.2.1]octane-1-carboxylic acid
—— (2S,5S)-5-isopropyl-2-(naphthalen-2-yl)-1-(3-oxobutyl)-3-(pyridin-2-yl)imidazolidin-4-one 1222985-79-6 C25H27N3O2
(2S,5S)-5-isopropyl-2-(naphthalen-2-yl)-1-(3-oxobutyl)-3-(pyridin-2-yl)imidazolidin-4-one
—— 5-methyl-3,6-diphenyl-5H-isoxazolo[5,4-d]pyrimidin-4-one 14246-73-2 C18H13N3O2
5-methyl-3,6-diphenyl-5H-isoxazolo[5,4-d]pyrimidin-4-one
—— 1,2-Difluoro-4-nitro-5-prop-1-en-2-ylbenzene 1449199-78-3 C9H7F2NO2
1,2-Difluoro-4-nitro-5-prop-1-en-2-ylbenzene
—— 2-chloro-5-(oxetan-3-yl)spiro[8H-pteridine-7,3'-oxolane]-6-one 1452229-02-5 C12H13ClN4O3
2-chloro-5-(oxetan-3-yl)spiro[8H-pteridine-7,3'-oxolane]-6-one
—— 2-[1-(2,2-dimethylpropyl)-3-methyl-2-oxo-2,3-dihydro-1H-imidazo[4,5-b]pyridin-5-yl]-4-[[4-hydroxypiperidin-1-yl]methyl]benzonitrile 1352422-45-7 C25H31N5O2
2-[1-(2,2-dimethylpropyl)-3-methyl-2-oxo-2,3-dihydro-1H-imidazo[4,5-b]pyridin-5-yl]-4-[[4-hydroxypiperidin-1-yl]methyl]benzonitrile
—— 3-(2-furyl)-4-(trifluoromethoxy)-1H-pyrazole 1450829-26-1 C8H5F3N2O2
3-(2-furyl)-4-(trifluoromethoxy)-1H-pyrazole
—— 2-methylsulfanyl-8-propan-2-yl-N-[[2-(1,2,4-triazol-1-yl)phenyl]methyl]pyrazolo[1,5-a][1,3,5]triazin-4-amine 1453835-28-3 C18H20N8S
2-methylsulfanyl-8-propan-2-yl-N-[[2-(1,2,4-triazol-1-yl)phenyl]methyl]pyrazolo[1,5-a][1,3,5]triazin-4-amine
—— 2-fluoro-N-[5-(1-methyl-1-phenylethyl)-1,3,4-thiadiazol-2-yl]-5-{[(2,2,2-trifluoroethyl)amino]sulfonyl}benzamide 1032463-14-1 C20H18F4N4O3S2
2-fluoro-N-[5-(1-methyl-1-phenylethyl)-1,3,4-thiadiazol-2-yl]-5-{[(2,2,2-trifluoroethyl)amino]sulfonyl}benzamide
—— (1R,2R,4S)-4-(2-chloro-4-bromo-benzenesulfonyl)-2-(3,3-difluoro-pyrrolidine-1-carbonyl)-cyclopentanecarboxylic acid 1258452-57-1 C17H17BrClF2NO5S
(1R,2R,4S)-4-(2-chloro-4-bromo-benzenesulfonyl)-2-(3,3-difluoro-pyrrolidine-1-carbonyl)-cyclopentanecarboxylic acid
—— —— 1078159-63-3 C14H25NO9S
—— [1-(5-acetyl-thiophen-2-ylmethyl)-1H-pyrazol-4-yl]-carbamic acid 2-chloro-benzyl ester 1163258-97-6 C18H16ClN3O3S
[1-(5-acetyl-thiophen-2-ylmethyl)-1H-pyrazol-4-yl]-carbamic acid 2-chloro-benzyl ester
—— {1-[5-(1,1-difluoro-ethyl)-furan-2-ylmethyl]-1H-pyrazol-3-yl}-carbamic acid 3-chloro-benzyl ester 1163258-12-5 C18H16ClF2N3O3
{1-[5-(1,1-difluoro-ethyl)-furan-2-ylmethyl]-1H-pyrazol-3-yl}-carbamic acid 3-chloro-benzyl ester
—— [1-(6-acetyl-pyridin-2-ylmethyl)-1H-pyrazol-3-yl]-carbamic acid 2-chloro-benzyl ester 1163259-50-4 C19H17ClN4O3
[1-(6-acetyl-pyridin-2-ylmethyl)-1H-pyrazol-3-yl]-carbamic acid 2-chloro-benzyl ester
—— N-(3-((4-cyanobenzyl)(4-(3-(2-(pyridin-3-yl)ethoxy)phenoxy)benzyl)amino)phenyl)methanesulfonamide 1264835-15-5 C35H32N4O4S
N-(3-((4-cyanobenzyl)(4-(3-(2-(pyridin-3-yl)ethoxy)phenoxy)benzyl)amino)phenyl)methanesulfonamide
—— 1-(2-chlorophenyl)-N-(imidazolidin-2-ylidene)-2-(pyridin-4-yl)ethanamine 1173172-35-4 C16H17ClN4
1-(2-chlorophenyl)-N-(imidazolidin-2-ylidene)-2-(pyridin-4-yl)ethanamine
—— 4-((S)-4-carboxy-2-{[1-(3-chloro-2-methylphenyl)-5-(1-ethoxycarbonylcyclobutoxy)-1H-pyrazole-3-carbonyl]amino}butyryl)piperazine-1-carboxylic acid ethyl ester 1164336-83-7 C30H38ClN5O9
4-((S)-4-carboxy-2-{[1-(3-chloro-2-methylphenyl)-5-(1-ethoxycarbonylcyclobutoxy)-1H-pyrazole-3-carbonyl]amino}butyryl)piperazine-1-carboxylic acid ethyl ester
—— 5-(4-chloro-phenyl)-2-methyl-oxazole-4-carboxylic acid [1-(5-oxo-hexyl)-1H-pyrazol-4-yl]-amide 1163257-60-0 C20H21ClN4O3
5-(4-chloro-phenyl)-2-methyl-oxazole-4-carboxylic acid [1-(5-oxo-hexyl)-1H-pyrazol-4-yl]-amide
—— rel-(3S,5S)-trans-6,7-Methylenedioxy-5-(2-cyclopropylethenyl)-1,5-dihydro-3-ethyl-5-(trifluoromethyl)-4,1-benzoxazepin-2(3H)-one 1175577-06-6 C18H18F3NO4
rel-(3S,5S)-trans-6,7-Methylenedioxy-5-(2-cyclopropylethenyl)-1,5-dihydro-3-ethyl-5-(trifluoromethyl)-4,1-benzoxazepin-2(3H)-one
—— 4-amino-1-(2-trifluoromethyl-benzyl)-piperidine-4-carboxylic acid (4-ethyl-phenyl)-amide 1262988-42-0 C22H26F3N3O
4-amino-1-(2-trifluoromethyl-benzyl)-piperidine-4-carboxylic acid (4-ethyl-phenyl)-amide
—— 5-(4-chloro-phenyl)-oxazole-4-carboxylic acid [1-(5-acetyl-furan-2-ylmethyl)-1H-pyrazol-4-yl]-amide 1163258-86-3 C20H15ClN4O4
5-(4-chloro-phenyl)-oxazole-4-carboxylic acid [1-(5-acetyl-furan-2-ylmethyl)-1H-pyrazol-4-yl]-amide