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中文名称 英文名称 CAS号 化学式 结构式图片
—— benzyl N-[(4S,6S,13S)-6-[(tert-butoxycarbonyl)amino]-11,15-dimethyl-9,12,16-trioxo-2-oxa-8,11,15-triazatricyclo[15.3.1.0<sup>4,8</sup>]henicosa-1(21),17,19-trien-13-yl]carbamate 1264222-78-7 C32H41N5O8
benzyl N-[(4S,6S,13S)-6-[(tert-butoxycarbonyl)amino]-11,15-dimethyl-9,12,16-trioxo-2-oxa-8,11,15-triazatricyclo[15.3.1.0<sup>4,8</sup>]henicosa-1(21),17,19-trien-13-yl]carbamate
—— (R)-2-(3-fluorophenyl)-7-(3-dimethylaminopyrrolidin-1-yl)-2H-[1,2,3]triazolo[4,5-f]quinoline-9-carboxylic acid 1287793-76-3 C22H21FN6O2
(R)-2-(3-fluorophenyl)-7-(3-dimethylaminopyrrolidin-1-yl)-2H-[1,2,3]triazolo[4,5-f]quinoline-9-carboxylic acid
—— 2-aminoethanol 4-(3-chloro-5-isoxazolyl)-thiazole-2-oxamate salt 104777-20-0 C2H7NO*C8H4ClN3O4S
2-aminoethanol 4-(3-chloro-5-isoxazolyl)-thiazole-2-oxamate salt
—— 1-(2,6-dichloro-4-trifluoromethylphenyl)-3-cyano-4-dichlorofluoromethylsulfinyl-5-methoxypyrazole 130233-99-7 C13H5Cl4F4N3O2S
1-(2,6-dichloro-4-trifluoromethylphenyl)-3-cyano-4-dichlorofluoromethylsulfinyl-5-methoxypyrazole
—— 25-acetoxy-4,5-seco-D:A-friedoolean-5(10),7-diene-4,6-dione 129393-16-4 C32H48O4
25-acetoxy-4,5-seco-D:A-friedoolean-5(10),7-diene-4,6-dione
—— ethyl 4-[2-chloro-4-fluoro-5-(4-difluoromethyl-4,5-dihydro-3-methyl-5-oxo-1H-1,2,4-triazol-1-yl)phenoxy]phenylcarboxylate 141500-94-9 C19H15ClF3N3O4
ethyl 4-[2-chloro-4-fluoro-5-(4-difluoromethyl-4,5-dihydro-3-methyl-5-oxo-1H-1,2,4-triazol-1-yl)phenoxy]phenylcarboxylate
—— 6,8-dimethyl-3,4-dihydro-5-[2-(4-((cyclopropylmethoxy)carbonylamino)-1-piperidyl)ethoxy]carbostyril hydrochloride 141498-27-3 C23H33N3O4*ClH
6,8-dimethyl-3,4-dihydro-5-[2-(4-((cyclopropylmethoxy)carbonylamino)-1-piperidyl)ethoxy]carbostyril hydrochloride
—— 2-(4-(2,4-difluorophenyl)piperidin-1-yl)-N-(6-(4-(2-fluorophenylcarbamoyl)piperazin-1-yl)pyridin-3-yl)-4-(trifluoromethyl)oxazole-5-carboxamide 1228004-53-2 C32H29F6N7O3
2-(4-(2,4-difluorophenyl)piperidin-1-yl)-N-(6-(4-(2-fluorophenylcarbamoyl)piperazin-1-yl)pyridin-3-yl)-4-(trifluoromethyl)oxazole-5-carboxamide
—— N-(5-tert-butyl-3-methanesulphonylamino-2-methoxy-phenyl)-3-(2-chloro-pyrimidin-4-yloxy)-4-chloro-benzamide 1215030-45-7 C23H24Cl2N4O5S
N-(5-tert-butyl-3-methanesulphonylamino-2-methoxy-phenyl)-3-(2-chloro-pyrimidin-4-yloxy)-4-chloro-benzamide
—— 2-amino-5-m-tolyl-thiazole-4-carboxylic acid [2-(4-chloro-phenyl)-ethyl]-cyclopropylmethyl-amide 1223581-52-9 C23H24ClN3OS
2-amino-5-m-tolyl-thiazole-4-carboxylic acid [2-(4-chloro-phenyl)-ethyl]-cyclopropylmethyl-amide
—— 2,2,2-trifluoro-N-(4-fluoro-3-{1-[1-(2-hydroxy-ethyl)-7-trifluoromethoxy-1H-indole-3-carbonyl]-piperidin-4-yl}-benzyl)-acetamide 1313042-25-9 C26H24F7N3O4
2,2,2-trifluoro-N-(4-fluoro-3-{1-[1-(2-hydroxy-ethyl)-7-trifluoromethoxy-1H-indole-3-carbonyl]-piperidin-4-yl}-benzyl)-acetamide
—— 3-(4-isopropoxy-3-methylphenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1408088-62-9 C15H17N5O
3-(4-isopropoxy-3-methylphenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
—— 6-(4-fluoro-3-methylphenyl)-2-methyl-N-{1-[3-(1-methyl-1H-pyrazol-4-yl)phenyl]ethyl}pyrimidin-4-amine 1404107-14-7 C24H24FN5
6-(4-fluoro-3-methylphenyl)-2-methyl-N-{1-[3-(1-methyl-1H-pyrazol-4-yl)phenyl]ethyl}pyrimidin-4-amine
—— N-(3-(2-hydroxyamino-2-oxo-1-phenylethyl)phenyl)-3-methylbenzamide 1070678-87-3 C22H20N2O3
N-(3-(2-hydroxyamino-2-oxo-1-phenylethyl)phenyl)-3-methylbenzamide
—— 2-[2-[2-hydroxy-3-(octadecyloxy)propylthio]ethoxy]ethyl trityl ether 131958-06-0 C44H66O4S
2-[2-[2-hydroxy-3-(octadecyloxy)propylthio]ethoxy]ethyl trityl ether
—— 3-bromo-4-(1-hydroxytridecyl)-5-hydroxy-2(5H)-furanone 120755-41-1 C17H29BrO4
3-bromo-4-(1-hydroxytridecyl)-5-hydroxy-2(5H)-furanone
—— 6-(1,3-benzothiazol-6-yl)-2-methyl-N-[1-(3-{[2-(2-methyl-1H-imidazol-1-yl)ethyl]oxy}phenyl)ethyl]pyrimidin-4-amine 1404106-59-7 C26H26N6OS
6-(1,3-benzothiazol-6-yl)-2-methyl-N-[1-(3-{[2-(2-methyl-1H-imidazol-1-yl)ethyl]oxy}phenyl)ethyl]pyrimidin-4-amine
—— (8S,11S,14S,17S)-14-benzyl-10-[(2S)-4-methyl-2-[[(2S)-2-(methylamino)propanoyl]amino]pentanoyl]-12,15-dioxo-2-oxa-5,6,7,10,13,16-hexazatetracyclo[17.2.2.14,7.18,11]pentacosa-1(22),4(25),5,19(23),20-pentaene-17-carboxylic acid 1432734-49-0 C36H46N8O7
(8S,11S,14S,17S)-14-benzyl-10-[(2S)-4-methyl-2-[[(2S)-2-(methylamino)propanoyl]amino]pentanoyl]-12,15-dioxo-2-oxa-5,6,7,10,13,16-hexazatetracyclo[17.2.2.14,7.18,11]pentacosa-1(22),4(25),5,19(23),20-pentaene-17-carboxylic acid
—— 4-N-(3-chloro-2-propan-2-ylsulfonylphenyl)-2-N-[2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]quinazoline-2,4-diamine 1097917-76-4 C34H42ClN7O3S
4-N-(3-chloro-2-propan-2-ylsulfonylphenyl)-2-N-[2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]quinazoline-2,4-diamine
—— 4-(5-{5-[(3-fluorophenoxy)methyl]-1-methyl-1H-pyrazol-4-yl}-1,2,4-oxadiazol-3-yl)benzenesulfonamide 1359027-34-1 C19H16FN5O4S
4-(5-{5-[(3-fluorophenoxy)methyl]-1-methyl-1H-pyrazol-4-yl}-1,2,4-oxadiazol-3-yl)benzenesulfonamide
—— 6-(3-Chloro-4-fluoroanilino)-4-azatricyclo[6.2.2.02,7]dodeca-2(7),5-dien-3-one 1357188-88-5 C17H16ClFN2O
6-(3-Chloro-4-fluoroanilino)-4-azatricyclo[6.2.2.02,7]dodeca-2(7),5-dien-3-one
—— 4-({3-[1-(2,2-dimethylpropyl)-3-methyl-2-oxo-2,3-dihydro-1H-benzimidazol-5-yl]phenoxy}methyl)benzonitrile 1359759-85-5 C27H27N3O2
4-({3-[1-(2,2-dimethylpropyl)-3-methyl-2-oxo-2,3-dihydro-1H-benzimidazol-5-yl]phenoxy}methyl)benzonitrile
—— 1,5-anhydro-2,3-dideoxy-4-O-methyl-3-{[(1R,3S)-3-(2,2,2-trifluoroethyl)-3-({(1S,4S)-5-[6-(trifluoromethyl)pyridin-2-yl]-2,5-diazabicyclo[2.2.1]hept-2-yl}carbonyl)cyclopentyl]amino}-D-erythro-pentitol 1228111-86-1 C25H32F6N4O3
1,5-anhydro-2,3-dideoxy-4-O-methyl-3-{[(1R,3S)-3-(2,2,2-trifluoroethyl)-3-({(1S,4S)-5-[6-(trifluoromethyl)pyridin-2-yl]-2,5-diazabicyclo[2.2.1]hept-2-yl}carbonyl)cyclopentyl]amino}-D-erythro-pentitol
—— 2-[6-bromo-9-(cyclopropylmethoxy)-1H-phenanthro[9,10-d]imidazol-2-yl]isophthalonitrile 1057385-02-0 C27H17BrN4O
2-[6-bromo-9-(cyclopropylmethoxy)-1H-phenanthro[9,10-d]imidazol-2-yl]isophthalonitrile
—— 2,2,2-trifluoro-N-(4-fluoro-3-{1-[7-methyl-1-(2-morpholin-4-yl-ethyl)-1H-indole-3-carbonyl]piperidin-4-yl}-benzyl)-acetamide 1313041-49-4 C30H34F4N4O3
2,2,2-trifluoro-N-(4-fluoro-3-{1-[7-methyl-1-(2-morpholin-4-yl-ethyl)-1H-indole-3-carbonyl]piperidin-4-yl}-benzyl)-acetamide
—— 1,3-Dimethyl-6-(4-[3-(2-phenyl-4-oxo-4H-1-benzopyran-8-yl)oxypropyl]piperazine-1-yl)-2,4(1H,3H)-pyrimidinedione oxalate 135653-41-7 C2H2O4*C28H30N4O5
1,3-Dimethyl-6-(4-[3-(2-phenyl-4-oxo-4H-1-benzopyran-8-yl)oxypropyl]piperazine-1-yl)-2,4(1H,3H)-pyrimidinedione oxalate
—— N-hydroxy-2-phenyl-2-(3-(2-(thiophen-2-yl)acetamido)phenyl)acetamide 1070678-94-2 C20H18N2O3S
N-hydroxy-2-phenyl-2-(3-(2-(thiophen-2-yl)acetamido)phenyl)acetamide
—— MeOCO-Thr-DL-N(Ph(3-F))Phg(2-Cl)-Unk 1448309-68-9 C24H25ClF3N3O5
MeOCO-Thr-DL-N(Ph(3-F))Phg(2-Cl)-Unk
—— 2-[3-[1-(4-Iodophenyl)cyclobutyl]indol-1-yl]acetic acid 1448611-19-5 C20H18INO2
2-[3-[1-(4-Iodophenyl)cyclobutyl]indol-1-yl]acetic acid
—— rac-2-amino-6-bromo-7-[1-(4-chloropyridine-3-sulfonylamino)ethyl]-[1,8]naphthyridine-3-carboxylic acid amide 1438254-47-7 C16H14BrClN6O3S
rac-2-amino-6-bromo-7-[1-(4-chloropyridine-3-sulfonylamino)ethyl]-[1,8]naphthyridine-3-carboxylic acid amide
—— N-(4-((2S,4R,5S,6R)-4-amino-5-hydroxy-6-isopropyltetrahydro-2H-pyran-2-yl)pyridin-3-yl)-6-(2,6-difluoro-4-(2-methoxyethoxy)phenyl)-5-fluoropicolinamide 1355010-71-7 C28H31F3N4O5
N-(4-((2S,4R,5S,6R)-4-amino-5-hydroxy-6-isopropyltetrahydro-2H-pyran-2-yl)pyridin-3-yl)-6-(2,6-difluoro-4-(2-methoxyethoxy)phenyl)-5-fluoropicolinamide
—— 6-[2-Chloro-4-(2-methylpyridin-3-yl)phenyl]-8-methyl-2-(4-piperidin-4-ylanilino)pyrido[2,3-d]pyrimidin-7-one 1428760-41-1 C31H29ClN6O
6-[2-Chloro-4-(2-methylpyridin-3-yl)phenyl]-8-methyl-2-(4-piperidin-4-ylanilino)pyrido[2,3-d]pyrimidin-7-one
—— 2-bromo-6-(4-chloro-phenyl)-5-(1,3-dimethyl-2-oxo-hexahydro-pyrimidin-5-yl)-1-isopropyl-5,6-dihydro-1H-pyrrolo[3,4-d]imidazol-4-one 1448871-44-0 C20H23BrClN5O2
2-bromo-6-(4-chloro-phenyl)-5-(1,3-dimethyl-2-oxo-hexahydro-pyrimidin-5-yl)-1-isopropyl-5,6-dihydro-1H-pyrrolo[3,4-d]imidazol-4-one
—— 1-(cyclohexylmethyl)-5-(3,5-ditert-butylphenyl)-2-methyl-N-(2-morpholin-4-ylethyl)pyrrole-3-carboxamide 1442423-69-9 C33H51N3O2
1-(cyclohexylmethyl)-5-(3,5-ditert-butylphenyl)-2-methyl-N-(2-morpholin-4-ylethyl)pyrrole-3-carboxamide
—— (2S)-N-(1-(2-chlorophenyl)-2-((3,3-difluorocyclobutyl)amino)-2-oxoethyl)-1-(4-cyanopyridin-2-yl)-N-(3-(methylsulfonyl)phenyl)-5-oxopyrrolidine-2-carboxamide 1448346-68-6 C30H26ClF2N5O5S
(2S)-N-(1-(2-chlorophenyl)-2-((3,3-difluorocyclobutyl)amino)-2-oxoethyl)-1-(4-cyanopyridin-2-yl)-N-(3-(methylsulfonyl)phenyl)-5-oxopyrrolidine-2-carboxamide
—— {4-[1-(3,4-dichlorophenyl)-3-methyl-1H-pyrazol-5-yl]piperidin-1-yl}[(3S,4R)-4-(2,4-difluorophenyl)-pyrrolidin-3-yl]methanone trifluoroacetate 1352245-88-5 C2HF3O2*C26H26Cl2F2N4O
{4-[1-(3,4-dichlorophenyl)-3-methyl-1H-pyrazol-5-yl]piperidin-1-yl}[(3S,4R)-4-(2,4-difluorophenyl)-pyrrolidin-3-yl]methanone trifluoroacetate
—— 7-[(4-Cyclopropylpiperazin-1-yl)methyl]-6-(ethoxymethyl)-5-(7-methoxy-5-methyl-1-benzothiophen-2-yl)pyrrolo[2,1-f][1,2,4]triazin-4-amine 1443531-28-9 C27H34N6O2S
7-[(4-Cyclopropylpiperazin-1-yl)methyl]-6-(ethoxymethyl)-5-(7-methoxy-5-methyl-1-benzothiophen-2-yl)pyrrolo[2,1-f][1,2,4]triazin-4-amine
—— 2-bromo-5-[(5-chloro-2-methyl-phenylamino)-(4-chloro-phenyl)-methyl]-1-((R)-1-methyl-2-triisopropylsilanyloxy-ethyl)-1H-imidazole-4-carboxylic acid 1448870-82-3 C30H40BrCl2N3O3Si
2-bromo-5-[(5-chloro-2-methyl-phenylamino)-(4-chloro-phenyl)-methyl]-1-((R)-1-methyl-2-triisopropylsilanyloxy-ethyl)-1H-imidazole-4-carboxylic acid
—— —— 1380420-79-0 C15H17NO5
—— —— 1331482-29-1 C15H19F2IO3
—— 1-{[(2S,1R,4R,5R)-4-(6-chloropurin-9-yl)-7,7-dimethyl-3,6,8-trioxabicyclo[3.3.0]oct-2-yl]methylthio}-2,4-difluorobenzene 1056617-02-7 C19H17ClF2N4O3S
1-{[(2S,1R,4R,5R)-4-(6-chloropurin-9-yl)-7,7-dimethyl-3,6,8-trioxabicyclo[3.3.0]oct-2-yl]methylthio}-2,4-difluorobenzene
—— 2-(3-butoxyphenyl)-N-hydroxy-2-phenylacetamide 1070674-62-2 C18H21NO3
2-(3-butoxyphenyl)-N-hydroxy-2-phenylacetamide
—— 5-[4'-[[5-isobutyl-3-(1,1-difluoropropyl)-1H-1,2,4-triazol-yl]methyl][1,1'-biphenyl]-2-yl]-1H-tetrazole 140124-52-3 C23H25F2N7
5-[4'-[[5-isobutyl-3-(1,1-difluoropropyl)-1H-1,2,4-triazol-yl]methyl][1,1'-biphenyl]-2-yl]-1H-tetrazole
—— methyl 4-[(4-methyl-6-{[4-(trifluoromethyl)pyridin-2-yl]amino}-2,3'-bipyridin-6'-yl)carbonyl]cyclohexanecarboxylate 1411772-85-4 C26H25F3N4O3
methyl 4-[(4-methyl-6-{[4-(trifluoromethyl)pyridin-2-yl]amino}-2,3'-bipyridin-6'-yl)carbonyl]cyclohexanecarboxylate
—— 2-fluoro-N-[(6S,7aS)-3-oxo-2-(4-trifluoromethoxy-phenyl)-hexahydro-pyrrolo[1,2-c]imidazol-6-yl]-benzenesulfonamide 1408313-85-8 C19H17F4N3O4S
2-fluoro-N-[(6S,7aS)-3-oxo-2-(4-trifluoromethoxy-phenyl)-hexahydro-pyrrolo[1,2-c]imidazol-6-yl]-benzenesulfonamide
—— N-[(6R,7aS)-3-oxo-2-(4-trifluoromethoxy-phenyl)-hexahydro-pyrrolo[1,2-c]imidazol-6-yl]-2-phenoxy-acetamide 1408313-82-5 C21H20F3N3O4
N-[(6R,7aS)-3-oxo-2-(4-trifluoromethoxy-phenyl)-hexahydro-pyrrolo[1,2-c]imidazol-6-yl]-2-phenoxy-acetamide
—— 4-(4-methyl-piperazin-1-yl)-N-[6-(2-phenoxy-ethoxy)-1H-indazol-3-yl]-benzamide 1409989-39-4 C27H29N5O3
4-(4-methyl-piperazin-1-yl)-N-[6-(2-phenoxy-ethoxy)-1H-indazol-3-yl]-benzamide
—— 5-chloro-2-[5-(2-isopropyl-imidazol-1-ylmethyl)-pyridin-3-yl]-2,3-dihydro-isoindol-1-one 1440515-33-2 C20H19ClN4O
5-chloro-2-[5-(2-isopropyl-imidazol-1-ylmethyl)-pyridin-3-yl]-2,3-dihydro-isoindol-1-one
—— (E)-ethyl 3-(5-((Z)-(3-(decahydronaphthalen-2-yl)-4-oxo-2-thioxothiazolidin-5-ylidene)methyl)-furan-2-yl)acrylate 1352735-82-0 C23H27NO4S2
(E)-ethyl 3-(5-((Z)-(3-(decahydronaphthalen-2-yl)-4-oxo-2-thioxothiazolidin-5-ylidene)methyl)-furan-2-yl)acrylate
—— (S)-3,5-dichloro-4-(2-(3-(cyclopropylmethoxy)-4-(difluoromethoxy)phenyl)-2-(2-(5,6-dimethoxy-1H-indol-1-yl)acetoxy)ethyl)pyridine 1-oxide 1431565-36-4 C30H28Cl2F2N2O7
(S)-3,5-dichloro-4-(2-(3-(cyclopropylmethoxy)-4-(difluoromethoxy)phenyl)-2-(2-(5,6-dimethoxy-1H-indol-1-yl)acetoxy)ethyl)pyridine 1-oxide