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中文名称 英文名称 CAS号 化学式 结构式图片
—— (4R)-4-fIuoro-7-(2-fIuoro-3-pyridinyl)-2-methoxy-5,6-dihydrospiro[1,3-oxazine-4,9-xanthen]-2-amine 1335217-31-6 C22H17F2N3O3
(4R)-4-fIuoro-7-(2-fIuoro-3-pyridinyl)-2-methoxy-5,6-dihydrospiro[1,3-oxazine-4,9-xanthen]-2-amine
—— 3-((5R)-2-amino-3-(5,6-dihydro-2H-pyran-3-yl)-1-fluoro-5,6-dihydrospiro[chromeno[2,3-c]pyridine-5,4'-[1,3]oxazin]-7-yl)benzonitrile 1335217-80-5 C27H21FN4O3
3-((5R)-2-amino-3-(5,6-dihydro-2H-pyran-3-yl)-1-fluoro-5,6-dihydrospiro[chromeno[2,3-c]pyridine-5,4'-[1,3]oxazin]-7-yl)benzonitrile
—— N-cyclopropyl-3-fluoro-5-{2-(3-hydroxy-2,2-dimethylpropyl)-4-[(4-methylpiperazin-1-yl)methyl]-1-oxo-1,2-dihydroisoquinolin-6-yl}-4-methylbenzamide 1220228-26-1 C31H39FN4O3
N-cyclopropyl-3-fluoro-5-{2-(3-hydroxy-2,2-dimethylpropyl)-4-[(4-methylpiperazin-1-yl)methyl]-1-oxo-1,2-dihydroisoquinolin-6-yl}-4-methylbenzamide
—— methyl 4-{[(4-{3-(cyanomethyl)-3-[4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl]azetidin-1-yl}piperidin-1-yl)carbonyl]amino}-3-fluorobenzoate 1334301-10-8 C28H28FN9O3
methyl 4-{[(4-{3-(cyanomethyl)-3-[4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl]azetidin-1-yl}piperidin-1-yl)carbonyl]amino}-3-fluorobenzoate
—— tert-butyl 3-(3-methoxy-4-(1-(4-(trifluoromethyl)benzyl)piperidin-4-yloxy)benzamido)propylcarbamate 1037491-31-8 C29H38F3N3O5
tert-butyl 3-(3-methoxy-4-(1-(4-(trifluoromethyl)benzyl)piperidin-4-yloxy)benzamido)propylcarbamate
—— 5-{[(3S)-1-(cyclopropylcarbonyl)-3-pyrrolidinyl]methyl}-4-[2-fluoro-4-(7-quinazolinyl)phenyl]-2,4-dihydro-3H-1,2,4-triazol-3-one 1332332-54-3 C25H23FN6O2
5-{[(3S)-1-(cyclopropylcarbonyl)-3-pyrrolidinyl]methyl}-4-[2-fluoro-4-(7-quinazolinyl)phenyl]-2,4-dihydro-3H-1,2,4-triazol-3-one
—— N-ethyl-N-methyl-N'-{3-[2,2,2-trifluoro-1-(pyridin-3-yl)-ethoxy]quinoxalin-2-yl}-sulfuric diamide 1226505-99-2 C18H18F3N5O3S
N-ethyl-N-methyl-N'-{3-[2,2,2-trifluoro-1-(pyridin-3-yl)-ethoxy]quinoxalin-2-yl}-sulfuric diamide
—— 6,6'-[(methylimino)bis(propane-3,1-diylimino)]bis[2-(4-ethylphenyl)-1,3-benzoxazole-4,7-dione] 1348915-27-4 C37H37N5O6
6,6'-[(methylimino)bis(propane-3,1-diylimino)]bis[2-(4-ethylphenyl)-1,3-benzoxazole-4,7-dione]
—— 2-(2-chloro-6-fluorophenyl)-N-(6-(4-(oxetan-3-yl)piperazin-1-yl)pyrimidin-4-yl)-3H-imidazo[4,5-c]pyridin-4-amine 1334410-77-3 C23H22ClFN8O
2-(2-chloro-6-fluorophenyl)-N-(6-(4-(oxetan-3-yl)piperazin-1-yl)pyrimidin-4-yl)-3H-imidazo[4,5-c]pyridin-4-amine
—— (5-chloro-6-methoxypyridin-2-yl)[4-methyl-3-(trifluoromethyl)phenyl]methanone 1310947-59-1 C15H11ClF3NO2
(5-chloro-6-methoxypyridin-2-yl)[4-methyl-3-(trifluoromethyl)phenyl]methanone
—— 4-(3-furyl)phenyl 5-thio-β-D-xylopyranoside 1011721-88-2 C15H16O5S
4-(3-furyl)phenyl 5-thio-β-D-xylopyranoside
—— (S)-tert-butyl 2-(6-ethynyl-1H-benzo[d]imidazol-2-yl)-4-cyclopropyl-2,5-dihydro-1H-pyrrole-1-carboxylate 1352393-21-5 C21H23N3O2
(S)-tert-butyl 2-(6-ethynyl-1H-benzo[d]imidazol-2-yl)-4-cyclopropyl-2,5-dihydro-1H-pyrrole-1-carboxylate
—— 4-Iodo-2'-t-butyl-4',6'-dinitrodiphenylamine 109825-57-2 C16H16IN3O4
4-Iodo-2'-t-butyl-4',6'-dinitrodiphenylamine
—— 1-(3-(4-(pyridine-3-carbonyl)piperazine-1-carbonyl)benzyl)quinazoline-2,4(1H,3H)-dione 1401681-74-0 C26H23N5O4
1-(3-(4-(pyridine-3-carbonyl)piperazine-1-carbonyl)benzyl)quinazoline-2,4(1H,3H)-dione
—— 2-benzyl-6-[(3-fluorophenyl)sulfonyl]-1,2,4,5,6,7-hexahydro-3H-pyrazolo[3,4-c]pyridin-3-one 1331738-63-6 C19H18FN3O3S
2-benzyl-6-[(3-fluorophenyl)sulfonyl]-1,2,4,5,6,7-hexahydro-3H-pyrazolo[3,4-c]pyridin-3-one
—— 2-{5-(4-fluorophenyl)-6-methyl-4-[(pyridin-2-ylmethyl)-amino]-thieno[2,3-d]pyrimidin-2-yl}-ethanol 1056054-77-3 C21H19FN4OS
2-{5-(4-fluorophenyl)-6-methyl-4-[(pyridin-2-ylmethyl)-amino]-thieno[2,3-d]pyrimidin-2-yl}-ethanol
—— (S)-N-[1-benzyl-2-(4-dimethylamino-piperidin-1-yl)-2-oxo-ethyl]-N-(4-pyridin-2-yl-benzyl)-3-(1,3,5-trimethyl-1H-pyrazol-4-yl)-acrylamide 1227791-20-9 C37H44N6O2
(S)-N-[1-benzyl-2-(4-dimethylamino-piperidin-1-yl)-2-oxo-ethyl]-N-(4-pyridin-2-yl-benzyl)-3-(1,3,5-trimethyl-1H-pyrazol-4-yl)-acrylamide
—— (S)-N-[1-benzyl-2-(4-dimethylamino-piperidin-1-yl)-2-oxo-ethyl]-N-(4-pyridin-2-yl-benzyl)-3-(4-trifluoromethyl-phenyl)-acrylamide 1227791-17-4 C38H39F3N4O2
(S)-N-[1-benzyl-2-(4-dimethylamino-piperidin-1-yl)-2-oxo-ethyl]-N-(4-pyridin-2-yl-benzyl)-3-(4-trifluoromethyl-phenyl)-acrylamide
—— 6-(3-chloro-4-fluorobenzyl)-2-(2-morpholin-4-ylethyl)-1,2,4,5,6,7-hexahydro-3H-pyrazolo[3,4-c]pyridin-3-one 1331738-02-3 C19H24ClFN4O2
6-(3-chloro-4-fluorobenzyl)-2-(2-morpholin-4-ylethyl)-1,2,4,5,6,7-hexahydro-3H-pyrazolo[3,4-c]pyridin-3-one
—— 4-{3-(cyanomethyl)-3-[4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl]azetidin-1-yl}-N-(2,6-dichlorophenyl)piperidine-1-carboxamide 1334300-61-6 C26H25Cl2N9O
4-{3-(cyanomethyl)-3-[4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl]azetidin-1-yl}-N-(2,6-dichlorophenyl)piperidine-1-carboxamide
—— 4-[4-(1,3-benzothiazol-5-yl)phenyl]-5-{[(3S)-1-(cyclopropylcarbonyl)-3-pyrrolidinyl]methyl}-2,4-dihydro-3H-1,2,4-triazol-3-one 1332332-01-0 C24H23N5O2S
4-[4-(1,3-benzothiazol-5-yl)phenyl]-5-{[(3S)-1-(cyclopropylcarbonyl)-3-pyrrolidinyl]methyl}-2,4-dihydro-3H-1,2,4-triazol-3-one
—— N-(2-(2,6-dichlorophenyl)-3H-imidazo[4,5-c]pyridin-4-yl)-5-methylisoxazol-3-amine 1334408-48-8 C16H11Cl2N5O
N-(2-(2,6-dichlorophenyl)-3H-imidazo[4,5-c]pyridin-4-yl)-5-methylisoxazol-3-amine
—— 3,5-dichloro-4-(4-(6-(4-methylpiperazin-1-yl)pyrimidin-4-ylamino)-3H-imidazo[4,5-c]pyridin-2-yl)benzonitrile 1334407-89-4 C22H19Cl2N9
3,5-dichloro-4-(4-(6-(4-methylpiperazin-1-yl)pyrimidin-4-ylamino)-3H-imidazo[4,5-c]pyridin-2-yl)benzonitrile
—— (S)-N-(1-{[2-(furan-3-ylmethyl-methyl-amino)-ethyl]-methyl-carbamoyl}-2-phenyl-ethyl)-N-(4-pyridin-2-yl-benzyl)-3-(4-trifluoromethyl-phenyl)-acrylamide 1227793-47-6 C40H39F3N4O3
(S)-N-(1-{[2-(furan-3-ylmethyl-methyl-amino)-ethyl]-methyl-carbamoyl}-2-phenyl-ethyl)-N-(4-pyridin-2-yl-benzyl)-3-(4-trifluoromethyl-phenyl)-acrylamide
—— 4-(4-bromophenyl)-5-{[(3S)-1-(2-methylpropanoyl)-3-pyrrolidinyl]methyl}-2,4-dihydro-3H-1,2,4-triazol-3-one 1332333-85-3 C17H21BrN4O2
4-(4-bromophenyl)-5-{[(3S)-1-(2-methylpropanoyl)-3-pyrrolidinyl]methyl}-2,4-dihydro-3H-1,2,4-triazol-3-one
—— 3-(4-fluorophenyl)-4-phenyl-5-(2-(tetrahydro-2H-pyran-2-yloxy)ethylthio)-1H-pyrazole 1231308-85-2 C22H23FN2O2S
3-(4-fluorophenyl)-4-phenyl-5-(2-(tetrahydro-2H-pyran-2-yloxy)ethylthio)-1H-pyrazole
—— {1-{1-[(1,2-dimethyl-1H-imidazol-4-yl)sulfonyl]piperidin-4-yl}-3-[4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl]azetidin-3-yl}acetonitrile 1334301-61-9 C24H28N10O2S
{1-{1-[(1,2-dimethyl-1H-imidazol-4-yl)sulfonyl]piperidin-4-yl}-3-[4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl]azetidin-3-yl}acetonitrile
—— 5-(3,4-dimethyl-phenyl)-thiazole-4-carboxylic acid cyclopropylmethyl-[2-(5-fluoro-1H-indol-3-yl)-ethyl]-amide 1223586-11-5 C26H26FN3OS
5-(3,4-dimethyl-phenyl)-thiazole-4-carboxylic acid cyclopropylmethyl-[2-(5-fluoro-1H-indol-3-yl)-ethyl]-amide
—— 2-[2-(4-methylphenyl)-2-oxoethyl]-1,3,4-thiazidin-5-one 1187371-78-3 C12H14N2O2S
2-[2-(4-methylphenyl)-2-oxoethyl]-1,3,4-thiazidin-5-one
—— di-tert-butyl 2,2'-((3-(1,3-dioxoisoindolin-2-yl)propyl)azanediyl)diacetate 1354023-17-8 C23H32N2O6
di-tert-butyl 2,2'-((3-(1,3-dioxoisoindolin-2-yl)propyl)azanediyl)diacetate
—— 3,3'-[2-(4-fluorophenyl)-2-oxoethylidene]bis[4-hydroxy-2H-1-benzopyran-2-one] 1619260-30-8 C26H15FO7
3,3'-[2-(4-fluorophenyl)-2-oxoethylidene]bis[4-hydroxy-2H-1-benzopyran-2-one]
—— —— 14886-32-9 C21H34ClNO
—— —— 1592601-45-0 Br*C8H11N2
—— —— 1527527-88-3 C22H22O5
—— 3,4-Dimethyl-1-phenyl-Δ<sup>2</sup>-pyrazolin 19212-65-8 C11H14N2
3,4-Dimethyl-1-phenyl-Δ<sup>2</sup>-pyrazolin
—— 6-hexanoyl-7-methoxy-1-methyl-3,4-dihydro-β-carboline 1215093-41-6 C19H24N2O2
6-hexanoyl-7-methoxy-1-methyl-3,4-dihydro-β-carboline
—— 9,10-dimethoxy-15-(3-nitrophenyl)-12,13-dihydro-7aH,15H-naphtho[1',2':5,6][1,3]oxazino[2,3-a]-isoquinoline 1346683-16-6 C28H24N2O5
9,10-dimethoxy-15-(3-nitrophenyl)-12,13-dihydro-7aH,15H-naphtho[1',2':5,6][1,3]oxazino[2,3-a]-isoquinoline
—— (1S,4aS,5R,6R)-(-)-1,2,3,4,4a,5,6,7-octahydro-5-[2-(t-butyldiphenylsiloxy)ethyl]-1-(4-methyl-4-pentenyl)-1,5,6-trimethylnaphthalene 199525-15-0 C37H54OSi
(1S,4aS,5R,6R)-(-)-1,2,3,4,4a,5,6,7-octahydro-5-[2-(t-butyldiphenylsiloxy)ethyl]-1-(4-methyl-4-pentenyl)-1,5,6-trimethylnaphthalene
—— trans-7,8-tetradecanediol 16000-65-0 C14H30O2
trans-7,8-tetradecanediol
—— 8-(2',3'-dihydroxypropyl)-8-phenylmethoxycarbonylamino-1,4-dioxaspiro[4.5]decane 159638-80-9 C19H27NO6
8-(2',3'-dihydroxypropyl)-8-phenylmethoxycarbonylamino-1,4-dioxaspiro[4.5]decane
—— 2-ethyl-4-[5-(2-ethyl-6-methyl-pyridin-4-yl)-[1,2,4]oxadiazol-3-yl]-6-methyl-phenol 1011261-54-3 C19H21N3O2
2-ethyl-4-[5-(2-ethyl-6-methyl-pyridin-4-yl)-[1,2,4]oxadiazol-3-yl]-6-methyl-phenol
—— (1R,2S,4S)-5,6-Dimethylene-7-oxa-bicyclo[2.2.1]heptane-2-carbonitrile 105064-80-0 C9H9NO
(1R,2S,4S)-5,6-Dimethylene-7-oxa-bicyclo[2.2.1]heptane-2-carbonitrile
—— tert-butyl (5-((benzyloxy)methyl)-4-(tert-butoxy)-7-((2R,4S,5R)-4-hydroxy-5-(hydroxymethyl)tetrahydrofuran-2-yl)-7H-pyrrolo[2,3-d]pyrimidin-2-yl)carbamate 1159510-06-1 C28H38N4O7
tert-butyl (5-((benzyloxy)methyl)-4-(tert-butoxy)-7-((2R,4S,5R)-4-hydroxy-5-(hydroxymethyl)tetrahydrofuran-2-yl)-7H-pyrrolo[2,3-d]pyrimidin-2-yl)carbamate
—— N-Boc-α-dehydro-Ala-L-Val-L-Thr(O-TBDPS)-OMe 1033722-46-1 C34H49N3O7Si
N-Boc-α-dehydro-Ala-L-Val-L-Thr(O-TBDPS)-OMe
—— 11(R)-hydroxy-12(R)-methoxy-11,12-dihydro-3-methylcholanthrene 110455-91-9 C22H20O2
11(R)-hydroxy-12(R)-methoxy-11,12-dihydro-3-methylcholanthrene
—— 3-[(2E,6E)-9-(3,3-Dimethyl-oxiranyl)-3,7-dimethyl-nona-2,6-dienyl]-1,3-dihydro-indol-2-one 102720-38-7 C23H31NO2
3-[(2E,6E)-9-(3,3-Dimethyl-oxiranyl)-3,7-dimethyl-nona-2,6-dienyl]-1,3-dihydro-indol-2-one
—— 1-(2-hydroxy-1,3,9,10-tetramethoxy-5H-dibenzo[c,e]azepin-6(7H)-yl)ethanone 1426853-69-1 C20H23NO6
1-(2-hydroxy-1,3,9,10-tetramethoxy-5H-dibenzo[c,e]azepin-6(7H)-yl)ethanone
—— N-[(3R,4S)-3-{[tert-butyl(dimethyl)silyl]oxy}tetrahydro-2H-pyran-4-yl]-4-[hydroxy(6-methoxypyridin-3-yl)methyl]quinoline-2-carboxamide 1314141-63-3 C28H37N3O5Si
N-[(3R,4S)-3-{[tert-butyl(dimethyl)silyl]oxy}tetrahydro-2H-pyran-4-yl]-4-[hydroxy(6-methoxypyridin-3-yl)methyl]quinoline-2-carboxamide
—— 1-[3-(Cyclopropylmethoxy)-4-fluorophenyl]ethanol 1198223-42-5 C12H15FO2
1-[3-(Cyclopropylmethoxy)-4-fluorophenyl]ethanol
—— ethyl-5-hydroxy-4-(4-methoxyphenylazo)-4-methylpentanoate 1221689-32-2 C15H22N2O4
ethyl-5-hydroxy-4-(4-methoxyphenylazo)-4-methylpentanoate