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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-[bis(diethylamino)phosphanyl]-N,N-diethyl-6-methyl-[1,2,4,3]triazaphospholo[5,4-b][1,3]benzothiazol-1-amine 131471-69-7 C20H36N6P2S
2-[bis(diethylamino)phosphanyl]-N,N-diethyl-6-methyl-[1,2,4,3]triazaphospholo[5,4-b][1,3]benzothiazol-1-amine
—— 4-[(3-chloro-4-fluorophenyl)amino]-6-[4-((1-methyl-4-piperidinylamino)carbonyl)cyclohexylamino]pyrimido[5,4-d]pyrimidine 1230872-60-2 C25H30ClFN8O
4-[(3-chloro-4-fluorophenyl)amino]-6-[4-((1-methyl-4-piperidinylamino)carbonyl)cyclohexylamino]pyrimido[5,4-d]pyrimidine
—— 3-benzylsulfanyl-1-ethyl-5-phenyl-6-(trideuteriomethoxy)-6H-1,2,4-triazine 146539-68-6 C19H21N3OS
3-benzylsulfanyl-1-ethyl-5-phenyl-6-(trideuteriomethoxy)-6H-1,2,4-triazine
—— 2-(2,4-Dimethoxy-phenyl)-3-p-tolyl-1-(2,2,2-trifluoro-acetyl)-2,3-dihydro-1H-quinazolin-4-one 136009-56-8 C25H21F3N2O4
2-(2,4-Dimethoxy-phenyl)-3-p-tolyl-1-(2,2,2-trifluoro-acetyl)-2,3-dihydro-1H-quinazolin-4-one
—— 5'-(pyrrolidin-1-ylsulfonyl)-1'-(4,4,4-trifluorobutyl)spiro[1,3-dioxane-2,3'-indol]-2'(1'H)-one 1234337-66-6 C19H23F3N2O5S
5'-(pyrrolidin-1-ylsulfonyl)-1'-(4,4,4-trifluorobutyl)spiro[1,3-dioxane-2,3'-indol]-2'(1'H)-one
—— diethyl (4-methyl-5-oxopentan-2-yl) phosphite 130279-56-0 C10H21O4P
diethyl (4-methyl-5-oxopentan-2-yl) phosphite
—— 2-Methyl-2-p-tolyl-6,6-bis-trifluoromethyl-tetrahydro-pyran 141207-59-2 C15H16F6O
2-Methyl-2-p-tolyl-6,6-bis-trifluoromethyl-tetrahydro-pyran
—— (2E,4Z)-ethyl 6-tetrahydropyranyloxy-2,4-hexadienoate 150919-17-8 C13H20O4
(2E,4Z)-ethyl 6-tetrahydropyranyloxy-2,4-hexadienoate
—— ethyl 9-(2-fluoroethyl)-6-hydroxy-2,3,4,9-tetrahydro-1H-carbazole-4-carboxylate 1360060-85-0 C17H20FNO3
ethyl 9-(2-fluoroethyl)-6-hydroxy-2,3,4,9-tetrahydro-1H-carbazole-4-carboxylate
—— S-(3-mercaptopropyl) 3-acetyl-4-oxo-2-trifluoromethylpentanethioate 1225456-70-1 C11H15F3O3S2
S-(3-mercaptopropyl) 3-acetyl-4-oxo-2-trifluoromethylpentanethioate
—— 1-[4-[[5'-(4-acetylphenoxy)-1,1,1',1'-tetramethyl-3,3'-spirobi[2H-indene]-5-yl]oxy]phenyl]ethanone 133387-18-5 C37H36O4
1-[4-[[5'-(4-acetylphenoxy)-1,1,1',1'-tetramethyl-3,3'-spirobi[2H-indene]-5-yl]oxy]phenyl]ethanone
—— triethyl(3-methoxyphenoxy)silane 18406-23-0 C13H22O2Si
triethyl(3-methoxyphenoxy)silane
—— 1-benzyl-3-(4-chlorophenyl)-N-methyl-N-[(5-methyl-isoxazol-3-yl)-methyl]-5-(trifluoromethyl)-1H-pyrrole-2-carboxylic acid amide 1574115-18-6 C25H21ClF3N3O2
1-benzyl-3-(4-chlorophenyl)-N-methyl-N-[(5-methyl-isoxazol-3-yl)-methyl]-5-(trifluoromethyl)-1H-pyrrole-2-carboxylic acid amide
—— 1-isopropyl-6-methyl-4-oxo-5-(3-(trifluoromethyl)phenyl)-1,4-dihydropyridine-3-carboxylic acid ((5-methanesulfonylthiophen-2-yl)methyl)amide 1569648-70-9 C23H23F3N2O4S2
1-isopropyl-6-methyl-4-oxo-5-(3-(trifluoromethyl)phenyl)-1,4-dihydropyridine-3-carboxylic acid ((5-methanesulfonylthiophen-2-yl)methyl)amide
—— (4-cyclobutyl-[1,4]diazepan-1-yl)-[5-(pyridin-4-ylsulfanyl)-pyridin-3-yl]-methanone 1153654-51-3 C20H24N4OS
(4-cyclobutyl-[1,4]diazepan-1-yl)-[5-(pyridin-4-ylsulfanyl)-pyridin-3-yl]-methanone
—— 2-([(1R)-1-methylbutyl]oxy)-8-(methyloxy)-9-[3-(tetrahydro-2H-pyran-4-yl)propyl]-9h-purin-6-amine 1050498-80-0 C19H31N5O3
2-([(1R)-1-methylbutyl]oxy)-8-(methyloxy)-9-[3-(tetrahydro-2H-pyran-4-yl)propyl]-9h-purin-6-amine
—— 3-(1-(7H-pyrrolo[2,3-d]pyrimidin-4-yloxy)but-3-enyl)-2-(2-chlorophenyl)-8-methylquinoline 1065478-32-1 C26H21ClN4O
3-(1-(7H-pyrrolo[2,3-d]pyrimidin-4-yloxy)but-3-enyl)-2-(2-chlorophenyl)-8-methylquinoline
—— 2-(pyridin-2-yl)benzofuran-5-carboxylic acid 1154060-90-8 C14H9NO3
2-(pyridin-2-yl)benzofuran-5-carboxylic acid
—— N-(3-aminopropyl)-N-(1-{7-chloro-3-[(2,5-difluorophenyl)amino]-4-oxo-3,4-dihydroquinazolin-2-yl}propyl)-4-methylbenzamide 1095253-91-0 C28H28ClF2N5O2
N-(3-aminopropyl)-N-(1-{7-chloro-3-[(2,5-difluorophenyl)amino]-4-oxo-3,4-dihydroquinazolin-2-yl}propyl)-4-methylbenzamide
—— 2,3,4-tri-O-benzoyl-5-C-[1-(4-methoxybenzyl)-1H-tetrazol-5-yl]-α-D-xylopyranosyde trichloroacetimidate 1228578-44-6 C37H30Cl3N5O9
2,3,4-tri-O-benzoyl-5-C-[1-(4-methoxybenzyl)-1H-tetrazol-5-yl]-α-D-xylopyranosyde trichloroacetimidate
—— —— 1462845-27-7 C15H22F2N4O
—— 2-pyrazinecarboxylic acid 5-[2-(4-fluorophenyl)-5-iodo-4-oxazolyl]-methyl ester 1262656-82-5 C15H9FIN3O3
2-pyrazinecarboxylic acid 5-[2-(4-fluorophenyl)-5-iodo-4-oxazolyl]-methyl ester
—— 1,2-dibromo-1-cyclopropylidenethane 182629-59-0 C5H6Br2
1,2-dibromo-1-cyclopropylidenethane
—— [2-[(2,4-dimethylphenyl)methyl-methylamino]-2,3,4,5,6,6a-hexahydro-1H-pentalen-3a-yl]-[3-(trifluoromethyl)-7,8-dihydro-5H-1,6-naphthyridin-6-yl]methanone 1138085-67-2 C28H34F3N3O
[2-[(2,4-dimethylphenyl)methyl-methylamino]-2,3,4,5,6,6a-hexahydro-1H-pentalen-3a-yl]-[3-(trifluoromethyl)-7,8-dihydro-5H-1,6-naphthyridin-6-yl]methanone
—— 5-(3-((7-methoxyquinolin-4-yloxy)methyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl)-3-methylthiophene-2-carbonyl chloride 1002308-88-4 C22H16ClN5O3S
5-(3-((7-methoxyquinolin-4-yloxy)methyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl)-3-methylthiophene-2-carbonyl chloride
—— 4-Hydroxy-2,3-dimethylbutanal 133782-35-1 C6H12O2
4-Hydroxy-2,3-dimethylbutanal
—— (3-methoxy-4-((5-(1-(2-methoxyethyl)-1H-pyrazol-4-yl)isoquinolin-3-yl)amino)phenyl)(3-methoxyazetidin-1-yl)methanone 1578243-55-6 C27H29N5O4
(3-methoxy-4-((5-(1-(2-methoxyethyl)-1H-pyrazol-4-yl)isoquinolin-3-yl)amino)phenyl)(3-methoxyazetidin-1-yl)methanone
—— (5S)-3-(trimethylsilylethynyl)-7-(3-pyridinyl)-spiro[chromeno[2,3-b]pyridine-5,4'-[1,3]oxazol]-2'-amine 1215869-75-2 C24H22N4O2Si
(5S)-3-(trimethylsilylethynyl)-7-(3-pyridinyl)-spiro[chromeno[2,3-b]pyridine-5,4'-[1,3]oxazol]-2'-amine
—— 4-{cyclopropyl-[4-(5-methanesulfonyl-pyridin-2-yl)-benzoyl]-amino}-piperidine-1-carboxylic acid tert-butyl ester 1578188-30-3 C26H33N3O5S
4-{cyclopropyl-[4-(5-methanesulfonyl-pyridin-2-yl)-benzoyl]-amino}-piperidine-1-carboxylic acid tert-butyl ester
—— 1-(4-(((tert-butyldimethylsilyl)oxy)methyl)-3-methoxyphenyl)-3-(4-cyclopropylphenoxy)-1H-pyrrol-2(5H)-one 1574542-70-3 C27H35NO4Si
1-(4-(((tert-butyldimethylsilyl)oxy)methyl)-3-methoxyphenyl)-3-(4-cyclopropylphenoxy)-1H-pyrrol-2(5H)-one
—— 6-(1,5-dimethyl-1H-pyrazol-4-yl)-2-methoxypyridin-3-amine 1578247-21-8 C11H14N4O
6-(1,5-dimethyl-1H-pyrazol-4-yl)-2-methoxypyridin-3-amine
—— US10138229, Example 47 1558036-78-4 C25H26N4O3
US10138229, Example 47
—— ethyl N-[6-[3-({[(1,1-dimethylethyl)oxy]carbonyl}amino)-1-pyrrolidinyl]-2-(2-pyridinyl)-4-pyrimidinyl]-3-alaninate 1373423-67-6 C23H32N6O4
ethyl N-[6-[3-({[(1,1-dimethylethyl)oxy]carbonyl}amino)-1-pyrrolidinyl]-2-(2-pyridinyl)-4-pyrimidinyl]-3-alaninate
—— —— 1462836-79-8 C17H23F2N3O
—— —— 1462845-14-2 C16H21F4N3O
—— —— 1454712-13-0 C25H32N4O3
—— —— 1509946-44-4 C16H22BrNO
—— N-tert-butoxycarbonyl-1-amino-2-[1-(4-fluorophenyl)-2-methyl-5-(4-methylsulphonylphenyl)-3-[2-(2-(tetrahydro-2H-pyran-2-yl)oxy)propyloxyl]ethyl]-1H-pyrrole 1363375-86-3 C33H43FN2O7S
N-tert-butoxycarbonyl-1-amino-2-[1-(4-fluorophenyl)-2-methyl-5-(4-methylsulphonylphenyl)-3-[2-(2-(tetrahydro-2H-pyran-2-yl)oxy)propyloxyl]ethyl]-1H-pyrrole
—— N-[1-(2-methylphenyl)-3-(3-bromophenylthio)-2-propenylidene]aniline 1140913-97-8 C22H18BrNS
N-[1-(2-methylphenyl)-3-(3-bromophenylthio)-2-propenylidene]aniline
—— 5-bromo-N-[[4-(N-cyano-S-methylsulfonimidoyl)phenyl]methyl]-6-methyl-1-(4-methylpyridin-3-yl)-4-oxopyridine-3-carboxamide 1570083-95-2 C22H20BrN5O3S
5-bromo-N-[[4-(N-cyano-S-methylsulfonimidoyl)phenyl]methyl]-6-methyl-1-(4-methylpyridin-3-yl)-4-oxopyridine-3-carboxamide
—— (3R,4R)-1-(5-bromo-4-methylpyrimidin-2-yl)pyrrolidine-3,4-diol 1578253-51-6 C9H12BrN3O2
(3R,4R)-1-(5-bromo-4-methylpyrimidin-2-yl)pyrrolidine-3,4-diol
—— 3-((6-oxo-3-(3-(4-(trifluoromethoxy)phenyl)-1,2,4-oxadiazol-5-yl)pyridazin-1(6H)-yl)methyl)benzonitrile 1571025-59-6 C21H12F3N5O3
3-((6-oxo-3-(3-(4-(trifluoromethoxy)phenyl)-1,2,4-oxadiazol-5-yl)pyridazin-1(6H)-yl)methyl)benzonitrile
—— 1-cyclopentyl-6-methyl-4-oxo-5-(3-trifluoromethyl-phenyl)-1,4-dihydro-pyridine-3-caarboxylic acid (5-methyl-[1,3,4]oxadiazol-2-ylmethyl)-amide 1569645-69-7 C23H23F3N4O3
1-cyclopentyl-6-methyl-4-oxo-5-(3-trifluoromethyl-phenyl)-1,4-dihydro-pyridine-3-caarboxylic acid (5-methyl-[1,3,4]oxadiazol-2-ylmethyl)-amide
—— —— 1571142-89-6 C48H48O4
—— 2,3,6-tri-(thiophenyl)benzoquinone 171820-61-4 C24H16O2S3
2,3,6-tri-(thiophenyl)benzoquinone
—— (1S,2R,6S,7R,8S,8aR)-6,7,8-tris(benzyloxy)octahydroindolizine-1,2-diyl diacetate 1550202-24-8 C33H37NO7
(1S,2R,6S,7R,8S,8aR)-6,7,8-tris(benzyloxy)octahydroindolizine-1,2-diyl diacetate
—— 1H-Isoindole-1,3(2H)-dione,2-[4-hydroxy-3-[[(tributylstannyl)oxy]carbonyl]phenyl]- 139257-36-6 C27H35NO5Sn
1H-Isoindole-1,3(2H)-dione,2-[4-hydroxy-3-[[(tributylstannyl)oxy]carbonyl]phenyl]-
—— 3,3a,4,5-tetrahydro-3,3-dimethyl-1-(3-methyl-2-butenyl)-10-methoxymethyleneoxy-1,5-dimethylene-1H,7H-furan[3,4-d]xanthene-7,13-diketone 1338230-37-7 C25H28O6
3,3a,4,5-tetrahydro-3,3-dimethyl-1-(3-methyl-2-butenyl)-10-methoxymethyleneoxy-1,5-dimethylene-1H,7H-furan[3,4-d]xanthene-7,13-diketone
—— 4-(Ethyl-d5)phenol 134334-12-6 C8H10O
4-(Ethyl-d5)phenol
—— 4-[[(1R,2S,3R,4R)-2,3-dihydroxy-4-(hydroxymethyl)cyclopentyl]amino]-5-(4-methyl-1,3-thiazol-2-yl)-2-[4-(trifluoromethyl)piperidin-1-yl]-1H-pyrimidin-6-one;hydrochloride 1433150-01-6 C20H26F3N5O4S*ClH
4-[[(1R,2S,3R,4R)-2,3-dihydroxy-4-(hydroxymethyl)cyclopentyl]amino]-5-(4-methyl-1,3-thiazol-2-yl)-2-[4-(trifluoromethyl)piperidin-1-yl]-1H-pyrimidin-6-one;hydrochloride