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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-(4-(thiophene-2-carbonylamino)piperidin-1-yl)ethyl 4-amino-5-chloro-2-methoxybenzoate 1148012-34-3 C20H24ClN3O4S
2-(4-(thiophene-2-carbonylamino)piperidin-1-yl)ethyl 4-amino-5-chloro-2-methoxybenzoate
—— (2-(2-phenylsulfonyl)phenylamino)-1-[1-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-octahydro-1H-pyrrolo[2,3-c]pyridin-6-yl]ethanone 1374239-98-1 C27H28N6O3S
(2-(2-phenylsulfonyl)phenylamino)-1-[1-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-octahydro-1H-pyrrolo[2,3-c]pyridin-6-yl]ethanone
—— 2-(2-methoxyphenoxy)-3-phenyl-6-[6-(trifluoromethyl)-1H-benzimidazol-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-one 1240709-68-5 C28H22F3N5O3
2-(2-methoxyphenoxy)-3-phenyl-6-[6-(trifluoromethyl)-1H-benzimidazol-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-one
—— 4-[2-amino-6-(dimethylamino)-4-pyrimidinyl]-2,6-difluorobenzaldehyde 1227910-21-5 C13H12F2N4O
4-[2-amino-6-(dimethylamino)-4-pyrimidinyl]-2,6-difluorobenzaldehyde
—— methyl 3-(5-cyano-3-ethyl-6-methylpyridin-2-yl)propanoate 1233244-50-2 C13H16N2O2
methyl 3-(5-cyano-3-ethyl-6-methylpyridin-2-yl)propanoate
—— (R)-1-((4-methyl-1-(2-(1-methyl-1H-indol-5-ylamino)pyrimidin-4-yl)-1H-pyrrol-3-yl)methyl) pyrrolidin-3-ol 1307802-06-7 C23H26N6O
(R)-1-((4-methyl-1-(2-(1-methyl-1H-indol-5-ylamino)pyrimidin-4-yl)-1H-pyrrol-3-yl)methyl) pyrrolidin-3-ol
—— (Z)-tert-butyl 3-(2-chloro-4-(N'-hydroxycarbamimidoyl)phenylsulfonamido)propanoate 1233477-87-6 C14H20ClN3O5S
(Z)-tert-butyl 3-(2-chloro-4-(N'-hydroxycarbamimidoyl)phenylsulfonamido)propanoate
—— N-[2-(tert-butylcarbamoyl)-4-cyano-6-methylphenyl]-2-(3-chloropyridin-2-yl)-5-[[4-chloro-6-(trifluoromethyl)benzotriazol-1-yl]methyl]pyrazole-3-carboxamide 1339949-27-7 C30H24Cl2F3N9O2
N-[2-(tert-butylcarbamoyl)-4-cyano-6-methylphenyl]-2-(3-chloropyridin-2-yl)-5-[[4-chloro-6-(trifluoromethyl)benzotriazol-1-yl]methyl]pyrazole-3-carboxamide
—— 1,4-Dichloro-5,8-dimethoxyisoquinoline 1001422-28-1 C11H9Cl2NO2
1,4-Dichloro-5,8-dimethoxyisoquinoline
—— [4-[2-Amino-6-methyl-5-[2-[6-(methylamino)pyridin-3-yl]ethynyl]pyrimidin-4-yl]-3-fluorophenyl]-(4-methylpiperazin-1-yl)methanone 1207349-05-0 C25H26FN7O
[4-[2-Amino-6-methyl-5-[2-[6-(methylamino)pyridin-3-yl]ethynyl]pyrimidin-4-yl]-3-fluorophenyl]-(4-methylpiperazin-1-yl)methanone
—— N-[2-[2-amino-5-[2-(6-aminopyridin-3-yl)ethynyl]-6-methylpyrimidin-4-yl]phenyl]acetamide 1207349-61-8 C20H18N6O
N-[2-[2-amino-5-[2-(6-aminopyridin-3-yl)ethynyl]-6-methylpyrimidin-4-yl]phenyl]acetamide
—— (1S,3'R,4'S,5'S,6'R)-6-[(4-acetylphenyl)methyl]-5-chloro-3',4',5',6'-tetrahydro-6'-(hydroxymethyl)-spiro[isobenzofuran-1(3H),2'-[2H]pyran]-3',4',5'-triol 1005142-07-3 C22H23ClO7
(1S,3'R,4'S,5'S,6'R)-6-[(4-acetylphenyl)methyl]-5-chloro-3',4',5',6'-tetrahydro-6'-(hydroxymethyl)-spiro[isobenzofuran-1(3H),2'-[2H]pyran]-3',4',5'-triol
—— 4((4-(trifluoromethyl)phenyl)ethynyl)-1H-pyrrolo[2,3-b]pyridine 1174297-55-2 C16H9F3N2
4((4-(trifluoromethyl)phenyl)ethynyl)-1H-pyrrolo[2,3-b]pyridine
—— 5-(4-carbamoyl-pyridin-2-yl)-1H-indole-2-carboxylic acid ethyl ester 1222173-78-5 C17H15N3O3
5-(4-carbamoyl-pyridin-2-yl)-1H-indole-2-carboxylic acid ethyl ester
—— 2-(3-chloropyridin-2-yl)-N-[2,4-dichloro-6-(propan-2-ylcarbamoyl)phenyl]-5-[[4-(1,1,1,2,3,3,3-heptafluoropropan-2-yl)triazol-2-yl]methyl]pyrazole-3-carboxamide 1339951-06-2 C25H18Cl3F7N8O2
2-(3-chloropyridin-2-yl)-N-[2,4-dichloro-6-(propan-2-ylcarbamoyl)phenyl]-5-[[4-(1,1,1,2,3,3,3-heptafluoropropan-2-yl)triazol-2-yl]methyl]pyrazole-3-carboxamide
—— 2-chloro-5-methoxy-4-[[4-[(7-methyl-3-oxo-1,2-dihydroinden-4-yl)oxy]-5-(trifluoromethyl)pyrimidin-2-yl]amino]-N-[(3R)-1-methylpyrrolidin-3-yl]benzamide 1227947-98-9 C28H27ClF3N5O4
2-chloro-5-methoxy-4-[[4-[(7-methyl-3-oxo-1,2-dihydroinden-4-yl)oxy]-5-(trifluoromethyl)pyrimidin-2-yl]amino]-N-[(3R)-1-methylpyrrolidin-3-yl]benzamide
—— (2R)-2-[[2-hydroxy-2-[4-(trifluoromethyl)phenyl]ethyl]amino]propan-1-ol 1350769-40-2 C12H16F3NO2
(2R)-2-[[2-hydroxy-2-[4-(trifluoromethyl)phenyl]ethyl]amino]propan-1-ol
—— 4-N-(1-ethylpiperidin-4-yl)-6-iodoquinoline-3,4-diamine 1350733-76-4 C16H21IN4
4-N-(1-ethylpiperidin-4-yl)-6-iodoquinoline-3,4-diamine
—— N'-(3,5-dimethoxyphenyl)-N'-[3-(1H-pyrazol-4-yl)quinoxalin-6-yl]-N-(2,2,2-trifluoroethyl)propane-1,3-diamine 1346243-06-8 C24H25F3N6O2
N'-(3,5-dimethoxyphenyl)-N'-[3-(1H-pyrazol-4-yl)quinoxalin-6-yl]-N-(2,2,2-trifluoroethyl)propane-1,3-diamine
—— ethyl N-[[(5S)-3-[3-fluoro-4-[4-[2-(pyridine-3-carbonylamino)acetyl]piperazin-1-yl]phenyl]-2-oxo-1,3-oxazolidin-5-yl]methyl]carbamate 1227687-20-8 C25H29FN6O6
ethyl N-[[(5S)-3-[3-fluoro-4-[4-[2-(pyridine-3-carbonylamino)acetyl]piperazin-1-yl]phenyl]-2-oxo-1,3-oxazolidin-5-yl]methyl]carbamate
—— N-carbamoylmethyl-3-methanesulfonyl-N-(2-methoxy-[3,4']bipyridinyl-3'-yl)-5-trifluoromethyl-benzamide 1395413-90-7 C22H19F3N4O5S
N-carbamoylmethyl-3-methanesulfonyl-N-(2-methoxy-[3,4']bipyridinyl-3'-yl)-5-trifluoromethyl-benzamide
—— 5-(2-Pyridin-3-ylethynyl)-6-[3-(trifluoromethoxy)phenyl]pyrimidine-2,4-diamine 1207347-93-0 C18H12F3N5O
5-(2-Pyridin-3-ylethynyl)-6-[3-(trifluoromethoxy)phenyl]pyrimidine-2,4-diamine
—— 2-Chloro-5-[3-(3-hydroxy-2,2,6,6-tetramethyl-5-oxopyran-4-yl)-4-methylphenyl]benzonitrile 1033758-53-0 C23H22ClNO3
2-Chloro-5-[3-(3-hydroxy-2,2,6,6-tetramethyl-5-oxopyran-4-yl)-4-methylphenyl]benzonitrile
—— 3'-phenylcarbamoyl-[1,1']bi[tricyclodecyl]-3-carboxylic acid 1206697-67-7 C28H35NO3
3'-phenylcarbamoyl-[1,1']bi[tricyclodecyl]-3-carboxylic acid
—— 3-(Propan-2-yloxy)propane-1-sulfonyl chloride 1339066-35-1 C6H13ClO3S
3-(Propan-2-yloxy)propane-1-sulfonyl chloride
—— —— 1307294-12-7 C24H28N2S2
—— N-[(4,6-dimethyl-2-oxo-1,2-dihydro-3-pyridinyl)methyl]-3-methyl-1-(1-methylethyl)-6-(4-pyrimidinyl)-1H-indole-4-carboxamide 1346574-12-6 C25H27N5O2
N-[(4,6-dimethyl-2-oxo-1,2-dihydro-3-pyridinyl)methyl]-3-methyl-1-(1-methylethyl)-6-(4-pyrimidinyl)-1H-indole-4-carboxamide
—— N-[1-[4-[4-[(5S)-5-(acetamidomethyl)-2-oxo-1,3-oxazolidin-3-yl]-2,6-difluorophenyl]piperazine-1-carbonyl]cyclopentyl]imidazo[1,2-a]pyrazine-2-carboxamide 1227685-82-6 C29H32F2N8O5
N-[1-[4-[4-[(5S)-5-(acetamidomethyl)-2-oxo-1,3-oxazolidin-3-yl]-2,6-difluorophenyl]piperazine-1-carbonyl]cyclopentyl]imidazo[1,2-a]pyrazine-2-carboxamide
—— 5-cyclopropyl-2-[4-[2-methyl-5-(1-propylsulfonyl-3,6-dihydro-2H-pyridin-4-yl)-3H-1-benzofuran-2-yl]piperidin-1-yl]pyrimidine 1346529-38-1 C29H38N4O3S
5-cyclopropyl-2-[4-[2-methyl-5-(1-propylsulfonyl-3,6-dihydro-2H-pyridin-4-yl)-3H-1-benzofuran-2-yl]piperidin-1-yl]pyrimidine
—— 6-(2-chlorophenyl)-2-[(2'-methyl-2',3'-dihydro-1'H-spiro[cyclopropane-1,4'-isoquinolin]-7'-yl)amino]imidazo[1,2-a]pyrimido[5,4-e]pyrimidin-5(6H)-one 1395026-31-9 C26H22ClN7O
6-(2-chlorophenyl)-2-[(2'-methyl-2',3'-dihydro-1'H-spiro[cyclopropane-1,4'-isoquinolin]-7'-yl)amino]imidazo[1,2-a]pyrimido[5,4-e]pyrimidin-5(6H)-one
—— 5-bromo-N-{3-(2-cyano-1H-pyrrol-1-yl)-1-[(4-methylpiperidin-1-yl)carbonyl]propyl}-2-methoxybenzenesulfonamide 1191032-00-4 C22H27BrN4O4S
5-bromo-N-{3-(2-cyano-1H-pyrrol-1-yl)-1-[(4-methylpiperidin-1-yl)carbonyl]propyl}-2-methoxybenzenesulfonamide
—— N-[4-chloro-2-methyl-6-(methylcarbamoyl)phenyl]-2-(3-chloropyridin-2-yl)-5-[(4-propan-2-yltriazol-2-yl)methyl]pyrazole-3-carboxamide 1339948-36-5 C24H24Cl2N8O2
N-[4-chloro-2-methyl-6-(methylcarbamoyl)phenyl]-2-(3-chloropyridin-2-yl)-5-[(4-propan-2-yltriazol-2-yl)methyl]pyrazole-3-carboxamide
—— —— 1307294-03-6 C26H25NS2
—— 4-(3-Fluoro-4-methoxyphenyl)-6-methyl-5-(2-pyridin-3-ylethynyl)pyrimidin-2-amine 1207346-93-7 C19H15FN4O
4-(3-Fluoro-4-methoxyphenyl)-6-methyl-5-(2-pyridin-3-ylethynyl)pyrimidin-2-amine
—— 2-[5-(4-Chloro-3-fluorophenyl)-2-ethylphenyl]-3-hydroxycyclopent-2-en-1-one 1235109-80-4 C19H16ClFO2
2-[5-(4-Chloro-3-fluorophenyl)-2-ethylphenyl]-3-hydroxycyclopent-2-en-1-one
—— 2-((2S)-1-(4-((2'-fluoro-5'-methoxy-2-methylbiphenyl-4-yl)methoxy)phenyl)pyrrolidin-2-yl)acetic acid trifluoroacetic acid salt 1283143-31-6 C2HF3O2*C27H28FNO4
2-((2S)-1-(4-((2'-fluoro-5'-methoxy-2-methylbiphenyl-4-yl)methoxy)phenyl)pyrrolidin-2-yl)acetic acid trifluoroacetic acid salt
—— tert-butyl {(3,5-dichlorophenylsulphonyl)-[5-(5-morpholin-4-ylmethyl-[1,2,4]oxadiazol-3-yl)naphthalen-2-yl]amino}acetate 1192208-95-9 C29H30Cl2N4O6S
tert-butyl {(3,5-dichlorophenylsulphonyl)-[5-(5-morpholin-4-ylmethyl-[1,2,4]oxadiazol-3-yl)naphthalen-2-yl]amino}acetate
—— ethyl 1-(((5-(4-(benzo[d]thiazol-2-ylamino)-2-fluorophenyl)pyrimidin-2-yl)oxy)methyl)cyclopropanecarboxylate 1431302-26-9 C24H21FN4O3S
ethyl 1-(((5-(4-(benzo[d]thiazol-2-ylamino)-2-fluorophenyl)pyrimidin-2-yl)oxy)methyl)cyclopropanecarboxylate
—— ethyl 1-(((5-(4-((4,6-dichlorobenzo[d]thiazol-2-yl)amino)phenyl)pyrimidin-2-yl)oxy)methyl)cyclohexanecarboxylate 1431301-99-3 C27H26Cl2N4O3S
ethyl 1-(((5-(4-((4,6-dichlorobenzo[d]thiazol-2-yl)amino)phenyl)pyrimidin-2-yl)oxy)methyl)cyclohexanecarboxylate
—— methyl 3-((5-(4-(benzo[d]thiazol-2-ylamino)-2,5-difluorophenyl)pyrimidin-2-yl)oxy)-2,2-dimethylpropanoate 1431301-30-2 C23H20F2N4O3S
methyl 3-((5-(4-(benzo[d]thiazol-2-ylamino)-2,5-difluorophenyl)pyrimidin-2-yl)oxy)-2,2-dimethylpropanoate
—— N-{[2-(5-{[(2S)-3-methyl-1-(methylamino)-1-oxobutan-2-yl]carbamoyl}furan-2-yl)pyridin-4-yl]methyl}pyridine-2-carboxamide 1227191-01-6 C23H25N5O4
N-{[2-(5-{[(2S)-3-methyl-1-(methylamino)-1-oxobutan-2-yl]carbamoyl}furan-2-yl)pyridin-4-yl]methyl}pyridine-2-carboxamide
—— 6-[4-(4-chlorophenoxycarbonyloxy)-2-methoxyphenyl]-5-(5-fluoro-2-methylphenoxymethyl)-2,2,4-trimethyl-1,2-dihydroquinoline 1027100-60-2 C34H31ClFNO5
6-[4-(4-chlorophenoxycarbonyloxy)-2-methoxyphenyl]-5-(5-fluoro-2-methylphenoxymethyl)-2,2,4-trimethyl-1,2-dihydroquinoline
—— (trans-4-{4-[4-amino-2-(2-methylpropoxy)-5-oxo-7,8-dihydropyrimido[5,4-f][1,4]oxazepin-6(5H)-yl]phenyl}cyclohexyl)acetic acid trifluoroacetate 1398551-88-6 C2HF3O2*C25H32N4O5
(trans-4-{4-[4-amino-2-(2-methylpropoxy)-5-oxo-7,8-dihydropyrimido[5,4-f][1,4]oxazepin-6(5H)-yl]phenyl}cyclohexyl)acetic acid trifluoroacetate
—— —— 1393884-14-4 C10H19O4S*C17H19O3S
—— N-{3-(2-cyano-1H-pyrrol-1-yl)-1-[(4-pyrimidin-2-ylpiperazin-1-yl)carbonyl]propyl}-1H-indole-4-sulfonamide 1191104-85-4 C25H26N8O3S
N-{3-(2-cyano-1H-pyrrol-1-yl)-1-[(4-pyrimidin-2-ylpiperazin-1-yl)carbonyl]propyl}-1H-indole-4-sulfonamide
—— 4-(2,6-dichlorophenyl)-N-[(2,4-dimethoxyphenyl)methyl]-5-oxotetrazole-1-carboxamide 1346565-87-4 C17H15Cl2N5O4
4-(2,6-dichlorophenyl)-N-[(2,4-dimethoxyphenyl)methyl]-5-oxotetrazole-1-carboxamide
—— —— 1307293-38-4 C22H22ClNS2
—— (2,3-dihydro-[1,4]dioxino[2,3-c]pyridin-7-ylmethyl)-[(1α,5α,6α)-3-((1RS)-8-methoxy-1,2-dihydro-3-oxa-5,9-diaza-cyclopenta[a]naphthalen-1-ylmethyl)-3-aza-bicyclo[3.1.0]hex-6-yl]-amine 1192282-00-0 C25H27N5O4
(2,3-dihydro-[1,4]dioxino[2,3-c]pyridin-7-ylmethyl)-[(1α,5α,6α)-3-((1RS)-8-methoxy-1,2-dihydro-3-oxa-5,9-diaza-cyclopenta[a]naphthalen-1-ylmethyl)-3-aza-bicyclo[3.1.0]hex-6-yl]-amine
—— 2-(3-chloropyridin-2-yl)-N-[4-cyano-2-methyl-6-(methylcarbamoyl)phenyl]-5-[(4-cyclopropyltriazol-2-yl)methyl]pyrazole-3-carboxamide 1339948-51-4 C25H22ClN9O2
2-(3-chloropyridin-2-yl)-N-[4-cyano-2-methyl-6-(methylcarbamoyl)phenyl]-5-[(4-cyclopropyltriazol-2-yl)methyl]pyrazole-3-carboxamide
—— 3-Phenyl-4-thia-1-azapentacyclo[9.7.1.02,6.07,19.012,17]nonadeca-2,5,7,9,11(19),12,14,16-octaen-18-one 1346571-19-4 C23H13NOS
3-Phenyl-4-thia-1-azapentacyclo[9.7.1.02,6.07,19.012,17]nonadeca-2,5,7,9,11(19),12,14,16-octaen-18-one