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中文名称 英文名称 CAS号 化学式 结构式图片
—— (S)-3-tert-butoxycarbonylamino-4-oxo-5-(2,2,2-trifluoro-ethyl)-2,3,4,5-tetrahydro-benzo[b][1,4]diazepine-1-carboxylic acid 2,2,2-trifluoro-ethyl ester 1015085-77-4 C19H21F6N3O5
(S)-3-tert-butoxycarbonylamino-4-oxo-5-(2,2,2-trifluoro-ethyl)-2,3,4,5-tetrahydro-benzo[b][1,4]diazepine-1-carboxylic acid 2,2,2-trifluoro-ethyl ester
—— N-{2-[(3H-imidazol-4-ylmethyl)-phenyl-amino]-ethyl}-methanesulfonamide 1020814-89-4 C13H18N4O2S
N-{2-[(3H-imidazol-4-ylmethyl)-phenyl-amino]-ethyl}-methanesulfonamide
—— US10202379, Reference Example 284 1370240-16-6 C25H23F2N3O3
US10202379, Reference Example 284
—— 5-Chloro-2-[[(3,5-dimethoxy-4-methylbenzoyl)-(3-phenylpropyl)amino]methyl]-1,3-thiazole-4-carboxylic acid 1282551-17-0 C24H25ClN2O5S
5-Chloro-2-[[(3,5-dimethoxy-4-methylbenzoyl)-(3-phenylpropyl)amino]methyl]-1,3-thiazole-4-carboxylic acid
—— 2-(4-(5-bromo-2-(2-chloro-6-fluoro-phenyl)-1H-imidazol-4-yl)-phenyl)-1-cyclopropyl-6-methyl-1H-benzoimidazole 1038842-74-8 C26H19BrClFN4
2-(4-(5-bromo-2-(2-chloro-6-fluoro-phenyl)-1H-imidazol-4-yl)-phenyl)-1-cyclopropyl-6-methyl-1H-benzoimidazole
—— 5-(3-(trifluoromethyl)phenyl)-1-isopropyl-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxylic acid ((5-(N-cyano-S-(methyl)sulfonimidoyl)-1-oxypyridin-2-yl)methyl)amide 1570077-15-4 C25H24F3N5O4S
5-(3-(trifluoromethyl)phenyl)-1-isopropyl-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxylic acid ((5-(N-cyano-S-(methyl)sulfonimidoyl)-1-oxypyridin-2-yl)methyl)amide
—— 3-(((5S)-2'-amino-7-phenylspiro[chromeno[2,3-b]pyridine-5,4'-[1,3]oxazol]-3-yl)oxy)-2,2-dimethylpropanenitrile 1215870-29-3 C25H22N4O3
3-(((5S)-2'-amino-7-phenylspiro[chromeno[2,3-b]pyridine-5,4'-[1,3]oxazol]-3-yl)oxy)-2,2-dimethylpropanenitrile
—— 3-Hydroxyimino-1-[2-(3-methylthiophen-2-yl)-2-oxoethyl]-5-phenyl-1,4-benzodiazepin-2-one 145084-78-2 C22H17N3O3S
3-Hydroxyimino-1-[2-(3-methylthiophen-2-yl)-2-oxoethyl]-5-phenyl-1,4-benzodiazepin-2-one
—— (2E,4R,7R)-4-benzyloxy-1-chloro-7-(methoxycarbonyl)amino-8-(trityloxy)oct-2-ene 153198-39-1 C36H38ClNO4
(2E,4R,7R)-4-benzyloxy-1-chloro-7-(methoxycarbonyl)amino-8-(trityloxy)oct-2-ene
—— 2-(4-{[(9H-fluoren-9-yl)methoxy]carbonyl}-1,1-dioxo-1lambda6-thiomorpholin-3-yl)acetic acid 1503338-67-7 C21H21NO6S
2-(4-{[(9H-fluoren-9-yl)methoxy]carbonyl}-1,1-dioxo-1lambda6-thiomorpholin-3-yl)acetic acid
—— (2aR,6aS,7R,10aS,10bR,10cR)-3,7,10a-Trimethyl-1,2,2a,6,6a,7,8,9,10,10a,10b,10c-dodecahydro-benzo[f]cyclopenta[cd]azulene-7-carboxylic acid methyl ester 142669-93-0 C21H30O2
(2aR,6aS,7R,10aS,10bR,10cR)-3,7,10a-Trimethyl-1,2,2a,6,6a,7,8,9,10,10a,10b,10c-dodecahydro-benzo[f]cyclopenta[cd]azulene-7-carboxylic acid methyl ester
—— 2-[2-hydroxyethyl-[2-[[(16E)-14-oxa-5,7,19,28-tetrazapentacyclo[17.5.2.12,6.18,12.022,26]octacosa-1(25),2(28),3,5,8(27),9,11,16,20,22(26),23-undecaen-11-yl]oxy]ethyl]amino]ethanol 1027635-57-9 C29H33N5O4
2-[2-hydroxyethyl-[2-[[(16E)-14-oxa-5,7,19,28-tetrazapentacyclo[17.5.2.12,6.18,12.022,26]octacosa-1(25),2(28),3,5,8(27),9,11,16,20,22(26),23-undecaen-11-yl]oxy]ethyl]amino]ethanol
—— 4-{4-[2,5-difluoro-4-(3-propylureido)phenyl]cyclohexylideneaminooxy}piperidine-1-carboxylic acid phenyl ester 1393685-16-9 C28H34F2N4O4
4-{4-[2,5-difluoro-4-(3-propylureido)phenyl]cyclohexylideneaminooxy}piperidine-1-carboxylic acid phenyl ester
—— —— 1456596-14-7 C23H16F3N5O
—— —— 1456596-25-0 C25H17F5N4O
—— US10202379, Reference Example 269 1370240-01-9 C25H25N3O5S
US10202379, Reference Example 269
—— N-[1-(4-trifluoromethylphenyl)-3-(4-fluorophenylthio)-2-propenylidene]-4-trifluoromethylaniline 1140914-82-4 C23H14F7NS
N-[1-(4-trifluoromethylphenyl)-3-(4-fluorophenylthio)-2-propenylidene]-4-trifluoromethylaniline
—— 6-((1-(cyclopropanecarbonyl)azetidin-3-yl)methyl)-5-(2-fluoro-4-(7-fluoronaphthalen-2-yl)phenyl)-4,6-diazaspiro[2.4]hept-4-en-7-one 1579518-39-0 C29H25F2N3O2
6-((1-(cyclopropanecarbonyl)azetidin-3-yl)methyl)-5-(2-fluoro-4-(7-fluoronaphthalen-2-yl)phenyl)-4,6-diazaspiro[2.4]hept-4-en-7-one
—— tert-butyl (1R,2R)-2-(benzyloxycarbonyl)amino-2-(diethoxyphosphoryl)-1-phenylethylcarbamate 1228746-91-5 C25H35N2O7P
tert-butyl (1R,2R)-2-(benzyloxycarbonyl)amino-2-(diethoxyphosphoryl)-1-phenylethylcarbamate
—— diethyl (4aR,9aR)-7-methoxy-4a-methyl-1-methylene-4,4a,9,9a-tetrahydro-1H-xanthene-3,3(2H)-dicarboxylate 1233027-61-6 C22H28O6
diethyl (4aR,9aR)-7-methoxy-4a-methyl-1-methylene-4,4a,9,9a-tetrahydro-1H-xanthene-3,3(2H)-dicarboxylate
—— 5-methyl-N-[4-(4-methylpiperazin-1-yl)phenyl]-2,2-dioxo-3,4-dihydro-1H-thiopyrano[4,3-b]indol-8-amine 1342810-13-2 C23H28N4O2S
5-methyl-N-[4-(4-methylpiperazin-1-yl)phenyl]-2,2-dioxo-3,4-dihydro-1H-thiopyrano[4,3-b]indol-8-amine
—— methyl {(5Z)-5-[(1-{[2,4-bis(trifluoromethyl)phenyl]methyl}-1H-indol-5-yl)methylidene]-2,4-dioxo-1,3-thiazolidin-3-yl}acetate 1351568-93-8 C24H16F6N2O4S
methyl {(5Z)-5-[(1-{[2,4-bis(trifluoromethyl)phenyl]methyl}-1H-indol-5-yl)methylidene]-2,4-dioxo-1,3-thiazolidin-3-yl}acetate
—— 1-{4-[3-phenyl-5-(2-piperidin-1-ylethoxy)-1,6-naphthyridin-2-yl]phenyl}methanamine 1238318-73-4 C28H30N4O
1-{4-[3-phenyl-5-(2-piperidin-1-ylethoxy)-1,6-naphthyridin-2-yl]phenyl}methanamine
—— 4-((6-(3-fluoro-4-methoxybenzyl)-1,4-oxazepan-4-yl)carbonyl)-N-1,3-thiazol-2-ylbenzenesulfonamide 1063728-18-6 C23H24FN3O5S2
4-((6-(3-fluoro-4-methoxybenzyl)-1,4-oxazepan-4-yl)carbonyl)-N-1,3-thiazol-2-ylbenzenesulfonamide
—— 1-((2-(trimethylsilyl)ethoxy)methyl)-1H-benzo[d]imidazole-5-carbaldehyde 1185767-48-9 C14H20N2O2Si
1-((2-(trimethylsilyl)ethoxy)methyl)-1H-benzo[d]imidazole-5-carbaldehyde
—— 3-chloro-4-[(1,3-thiazol-2-ylamino)sulfonyl]-N-[3-fluoro-4-(trifluoromethyl)benzyl]benzamide 1063730-18-6 C18H12ClF4N3O3S2
3-chloro-4-[(1,3-thiazol-2-ylamino)sulfonyl]-N-[3-fluoro-4-(trifluoromethyl)benzyl]benzamide
—— ethyl 2-[[(3S)-3-[[(2S)-3-cyclohexyl-2-[(2-thiophen-2-ylacetyl)amino]propanoyl]amino]-2-oxo-4-phenylmethoxybutanoyl]amino]acetate 1229294-47-6 C30H39N3O7S
ethyl 2-[[(3S)-3-[[(2S)-3-cyclohexyl-2-[(2-thiophen-2-ylacetyl)amino]propanoyl]amino]-2-oxo-4-phenylmethoxybutanoyl]amino]acetate
—— N-[4-methyl-2-[3-(3-oxopiperazin-1-yl)prop-1-ynyl]phenyl]-6-(trifluoromethoxy)-3,4-dihydro-2H-1,4-benzoxazine-2-carboxamide 1233530-10-3 C24H23F3N4O4
N-[4-methyl-2-[3-(3-oxopiperazin-1-yl)prop-1-ynyl]phenyl]-6-(trifluoromethoxy)-3,4-dihydro-2H-1,4-benzoxazine-2-carboxamide
—— N-[4-(2-{[3-(4-methylpiperazin-1-yl)propyl]amino}-5,6-dihydrobenzo[h]quinazolin-6-yl)phenyl]-2-(methylsulfonyl)benzenesulfonamide 1234355-37-3 C33H38N6O4S2
N-[4-(2-{[3-(4-methylpiperazin-1-yl)propyl]amino}-5,6-dihydrobenzo[h]quinazolin-6-yl)phenyl]-2-(methylsulfonyl)benzenesulfonamide
—— 6-[(E)-2-(2-cyclopentyloxy-3-methoxyphenyl)vinyl]-N-[4-(trifluoromethyl)-1,3-thiazol-2-yl]imidazo[2,1-b][1,3]thiazole-5-carboxamide 1228828-87-2 C24H21F3N4O3S2
6-[(E)-2-(2-cyclopentyloxy-3-methoxyphenyl)vinyl]-N-[4-(trifluoromethyl)-1,3-thiazol-2-yl]imidazo[2,1-b][1,3]thiazole-5-carboxamide
—— [Pt(PEt<sub>3</sub>)<sub>2</sub>(N-ethoxycarbonylpyrrole-2-thiocarboxamide)] 1498381-80-8 C20H40N2O2P2PtS
[Pt(PEt<sub>3</sub>)<sub>2</sub>(N-ethoxycarbonylpyrrole-2-thiocarboxamide)]
—— —— 1078727-77-1 C17H11BN4O8
—— 1-(6-acetoxy-3-methyl-benzofuran-2-yl)-propan-1-one 106475-94-9 C14H14O4
1-(6-acetoxy-3-methyl-benzofuran-2-yl)-propan-1-one
—— (3E,4Z)-1-methoxy-4-[3-(phenylsulfanylmethylene)-4-(p-tolyl-2-propynylidene)tetrahydrofuran-2-yl]benzene 1380676-42-5 C28H24O2S
(3E,4Z)-1-methoxy-4-[3-(phenylsulfanylmethylene)-4-(p-tolyl-2-propynylidene)tetrahydrofuran-2-yl]benzene
—— (Z)-4-methyl-3-(2-oxo-2-phenylethylidene)indolin-2-one 1608112-09-9 C17H13NO2
(Z)-4-methyl-3-(2-oxo-2-phenylethylidene)indolin-2-one
—— 1,3-di-tert-butyl-2-fluoro-2-(di-tert-butyl-phenyl-silylamino)-4,4-dimethyl-1,3-diaza-2,4-disilacyclobutane 1360457-13-1 C24H48FN3Si3
1,3-di-tert-butyl-2-fluoro-2-(di-tert-butyl-phenyl-silylamino)-4,4-dimethyl-1,3-diaza-2,4-disilacyclobutane
—— —— 1160371-43-6 C12H23BrOSi
—— —— 1312615-91-0 C17H24O4
—— [(3-bromorophenyl)CaI(tetrahydrofuran)<sub>4</sub>] 1415220-00-6 C22H36BrCaIO4
[(3-bromorophenyl)CaI(tetrahydrofuran)<sub>4</sub>]
—— —— 17211-15-3 C7H9Na11O24P6
—— N-(5-(benzyloxy)pyrimidin-2-yl)benzamide 1361235-68-8 C18H15N3O2
N-(5-(benzyloxy)pyrimidin-2-yl)benzamide
—— ethyl (1S,2S,5S)-2-hydroxy-5-methoxy-6-oxabicyclo<3.2.1>octane-1-carboxylate 127484-11-1 C11H18O5
ethyl (1S,2S,5S)-2-hydroxy-5-methoxy-6-oxabicyclo<3.2.1>octane-1-carboxylate
—— [Fe((2-methoxyethyl)bis(pyrid-2-ylmethyl)amine)Cl3] 1325743-87-0 C15H19Cl3FeN3O
[Fe((2-methoxyethyl)bis(pyrid-2-ylmethyl)amine)Cl3]
—— 3-(5-(2-(((2'-chloro-4'-fluoro-[1,1'-biphenyl]-4-yl)amino)methyl)-5-(trifluoromethyl)phenyl)picolinamido)propanoic acid 1415127-59-1 C29H22ClF4N3O3
3-(5-(2-(((2'-chloro-4'-fluoro-[1,1'-biphenyl]-4-yl)amino)methyl)-5-(trifluoromethyl)phenyl)picolinamido)propanoic acid
—— dimethyl 7-(tert-butylamino)-2,3-dicyano-5H-benzo[h]pyrano[3,2-f]quinoxaline-5,6-dicarboxylate 1359092-37-7 C25H21N5O5
dimethyl 7-(tert-butylamino)-2,3-dicyano-5H-benzo[h]pyrano[3,2-f]quinoxaline-5,6-dicarboxylate
—— —— 1408288-17-4 C34H49ClN6O7Si
—— [Ru(bpy)2(bpy-ph-NHCO-trpy)Ru(bpy)(H2O)](4+) 1380114-97-5 C64H52N12O2Ru2
[Ru(bpy)2(bpy-ph-NHCO-trpy)Ru(bpy)(H2O)](4+)
—— (2S)-2-[[2-(3-chlorophenyl)-2-hydroxyethyl]amino]propan-1-ol 1350768-87-4 C11H16ClNO2
(2S)-2-[[2-(3-chlorophenyl)-2-hydroxyethyl]amino]propan-1-ol
—— 1-(2,4-bis-benzyloxy-3-iodophenyl)-2-cyclopropylethanone 1204737-75-6 C25H23IO3
1-(2,4-bis-benzyloxy-3-iodophenyl)-2-cyclopropylethanone
—— (2R)-3-(3,4-diacetyloxyphenyl)-2-hydroxypropanoic acid 1339947-18-0 C13H14O7
(2R)-3-(3,4-diacetyloxyphenyl)-2-hydroxypropanoic acid