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中文名称 英文名称 CAS号 化学式 结构式图片
—— 8-methyl-4-oxo-1-phenyl-5H-[1,2,4]triazolo[4,3-a]quinoxaline-7-carboxylic acid 1243162-98-2 C17H12N4O3
8-methyl-4-oxo-1-phenyl-5H-[1,2,4]triazolo[4,3-a]quinoxaline-7-carboxylic acid
—— 3-[2-[(1R)-1-[(2R)-2-hydroxy-3-[(2S)-2-[[4-(trifluoromethyl)phenyl]methyl]pyrrolidin-1-yl]propoxy]ethyl]phenyl]propanoic acid 1232831-46-7 C26H32F3NO4
3-[2-[(1R)-1-[(2R)-2-hydroxy-3-[(2S)-2-[[4-(trifluoromethyl)phenyl]methyl]pyrrolidin-1-yl]propoxy]ethyl]phenyl]propanoic acid
—— N-(4-((5S,7S,8R)-7-amino-8-hydroxy-8-methyl-4-oxaspiro[2.5]octan-5-yl)pyridin-3-yl)-6-(2,6-difluorophenyl)-5-fluoropicolinamide 1355010-22-8 C25H23F3N4O3
N-(4-((5S,7S,8R)-7-amino-8-hydroxy-8-methyl-4-oxaspiro[2.5]octan-5-yl)pyridin-3-yl)-6-(2,6-difluorophenyl)-5-fluoropicolinamide
—— 2-[(2-Chlorophenyl)methyl]-4-(hydroxymethyl)-4-methyl-3-isoxazolidinone 140360-36-7 C12H14ClNO3
2-[(2-Chlorophenyl)methyl]-4-(hydroxymethyl)-4-methyl-3-isoxazolidinone
—— (S)-1-(1,1-dioxo-1λ6-thiomorpholine-4-carbonyl)-piperidine-2-carboxylic acid [2-(2-chloro-6-fluoro-benzylsulfanyl)-ethyl]-amide 1240057-78-6 C20H27ClFN3O4S2
(S)-1-(1,1-dioxo-1λ6-thiomorpholine-4-carbonyl)-piperidine-2-carboxylic acid [2-(2-chloro-6-fluoro-benzylsulfanyl)-ethyl]-amide
—— N-methyl-N-[[1-(4-methylphenyl)piperidin-4-yl]methyl]-4-[4-nitro-3-(trifluoromethyl)anilino]piperidine-1-carboxamide 1247035-73-9 C27H34F3N5O3
N-methyl-N-[[1-(4-methylphenyl)piperidin-4-yl]methyl]-4-[4-nitro-3-(trifluoromethyl)anilino]piperidine-1-carboxamide
—— 7-(7-chloro-3,4-dihydro-1H-isoquinoline-2-carbonyl)-8-methyl-1-(oxan-4-yl)-5H-imidazo[1,5-a]quinoxalin-4-one 1243155-61-4 C26H25ClN4O3
7-(7-chloro-3,4-dihydro-1H-isoquinoline-2-carbonyl)-8-methyl-1-(oxan-4-yl)-5H-imidazo[1,5-a]quinoxalin-4-one
—— 2-(2,6-dichloro-phenylamino)-1-methyl-1H-benzimidazole-5-carboxylic acid (4,4-difluoro-cyclohexyl)amide 1219120-38-3 C21H20Cl2F2N4O
2-(2,6-dichloro-phenylamino)-1-methyl-1H-benzimidazole-5-carboxylic acid (4,4-difluoro-cyclohexyl)amide
—— (4-hydroxy-2-methyl-1,1-dioxo-1,2-dihydro-2H-benzo[e][1,2]thiazin-3-yl)-(1-phenyl-cyclopropyl)-methanone 1242133-92-1 C19H17NO4S
(4-hydroxy-2-methyl-1,1-dioxo-1,2-dihydro-2H-benzo[e][1,2]thiazin-3-yl)-(1-phenyl-cyclopropyl)-methanone
—— 2-(4-chloro-3-fluorophenyl)-N-cyclohexylimidazo[1,2-a]pyridin-3-amine 1218933-55-1 C19H19ClFN3
2-(4-chloro-3-fluorophenyl)-N-cyclohexylimidazo[1,2-a]pyridin-3-amine
—— ethyl 3-(3-fluoro-4-hydroxyphenyl)-2,2,3,3-tetradeuteriopropanoate 1234846-22-0 C11H13FO3
ethyl 3-(3-fluoro-4-hydroxyphenyl)-2,2,3,3-tetradeuteriopropanoate
—— ethyl (2E)-3-{2-[(1R)-1-({(2R)-3-[(2S)-2-(3-fluoro-4-methylbenzyl)pyrrolidin-1-yl]-2-hydroxypropyl}oxy)ethyl]-4-methylphenyl}prop-2-enoate 1232829-04-7 C29H38FNO4
ethyl (2E)-3-{2-[(1R)-1-({(2R)-3-[(2S)-2-(3-fluoro-4-methylbenzyl)pyrrolidin-1-yl]-2-hydroxypropyl}oxy)ethyl]-4-methylphenyl}prop-2-enoate
—— 2-[(E)-2-phenylvinyl]-N-(pyrimidin-5-ylmethyl)pyrido[3,4-d]pyrimidin-4-amine 1352995-34-6 C20H16N6
2-[(E)-2-phenylvinyl]-N-(pyrimidin-5-ylmethyl)pyrido[3,4-d]pyrimidin-4-amine
—— N-((S)-1-Ethyl-pyrrolidin-2-ylmethyl)-2-hydroxy-6-methoxy-5-methyl-3-propyl-benzamide 129725-12-8 C19H30N2O3
N-((S)-1-Ethyl-pyrrolidin-2-ylmethyl)-2-hydroxy-6-methoxy-5-methyl-3-propyl-benzamide
—— 11β-(4-Dimethylaminophenyl)-3,3-ethylenedioxy-17α-(3-hydroxyprop-1(Z)-enyl)-9-estrene-5α,17β-diol 101771-83-9 C31H43NO5
11β-(4-Dimethylaminophenyl)-3,3-ethylenedioxy-17α-(3-hydroxyprop-1(Z)-enyl)-9-estrene-5α,17β-diol
—— 4-[4-(1-isopropyl-1H-imidazo[4,5-c]pyridin-6-ylamino)pyrimidin-2-yl]piperazin-2-one 1612165-68-0 C17H20N8O
4-[4-(1-isopropyl-1H-imidazo[4,5-c]pyridin-6-ylamino)pyrimidin-2-yl]piperazin-2-one
—— 4-(trifluoromethyl)-N-phenyl-2-aminopyridine 1448801-58-8 C12H9F3N2
4-(trifluoromethyl)-N-phenyl-2-aminopyridine
—— N-(N2-(((9H-fluoren-9-yl)methoxy)carbonyl)-N6-(tert-butoxycarbonyl)-L-lysyl)-N-benzylglycine 1582256-93-6 C35H41N3O7
N-(N2-(((9H-fluoren-9-yl)methoxy)carbonyl)-N6-(tert-butoxycarbonyl)-L-lysyl)-N-benzylglycine
—— (S)-4-(2-(2-phenylthiazol-4-yl)2-(4-(methoxycarbonyl)thiazole-5-ylamino)ethyl)phenylsulfamic acid ammonium salt 1235330-73-0 C22H20N4O5S3*H3N
(S)-4-(2-(2-phenylthiazol-4-yl)2-(4-(methoxycarbonyl)thiazole-5-ylamino)ethyl)phenylsulfamic acid ammonium salt
—— Lersivirine metabolite M17 1204578-43-7 C17H18N4O3
Lersivirine metabolite M17
—— 3-[2-[4-[(2S,3R)-2-[4-[3,4-dihydroxy-3-(hydroxymethyl)butyl]phenyl]-3-[(3S)-3-(4-fluorophenyl)-3-hydroxypropyl]-4-oxoazetidin-1-yl]phenyl]ethyl]pyrazine-2-carboxamide 1025467-69-9 C36H39FN4O6
3-[2-[4-[(2S,3R)-2-[4-[3,4-dihydroxy-3-(hydroxymethyl)butyl]phenyl]-3-[(3S)-3-(4-fluorophenyl)-3-hydroxypropyl]-4-oxoazetidin-1-yl]phenyl]ethyl]pyrazine-2-carboxamide
—— 3-[5-(2,4-difluorophenyl)-4,5-diazatricyclo[5.2.1.0(2,6)]deca-2(6),3-dien-3-yl]phenylmethanol 1024004-49-6 C21H18F2N2O
3-[5-(2,4-difluorophenyl)-4,5-diazatricyclo[5.2.1.0(2,6)]deca-2(6),3-dien-3-yl]phenylmethanol
—— 5-chloro-2-{[7-(1-ethylpropyl)-4-methoxy-1-methyl-1H-benzimidazol-2-yl]oxy}benzenesulfonamide 1022248-98-1 C20H24ClN3O4S
5-chloro-2-{[7-(1-ethylpropyl)-4-methoxy-1-methyl-1H-benzimidazol-2-yl]oxy}benzenesulfonamide
—— 2-(4-methoxy-9H-xanthen-9-yl)-2-methyl-N-{4-[4-(4-pyridinyl)benzyl]-1,3-thiazol-2-yl}propanamide 1008114-07-5 C33H29N3O3S
2-(4-methoxy-9H-xanthen-9-yl)-2-methyl-N-{4-[4-(4-pyridinyl)benzyl]-1,3-thiazol-2-yl}propanamide
—— 4-[2-(1-(3,4-dichlorophenyl)-5-methyl-1H-1,2,4-triazol-3-yloxy)ethyl]morpholine oxalate 1025011-44-2 C2H2O4*C15H18Cl2N4O2
4-[2-(1-(3,4-dichlorophenyl)-5-methyl-1H-1,2,4-triazol-3-yloxy)ethyl]morpholine oxalate
—— (3,4-dimethoxy-phenyl)-(6-pyrazol-1-yl-pyridin-2-yl)-amine 1043893-72-6 C16H16N4O2
(3,4-dimethoxy-phenyl)-(6-pyrazol-1-yl-pyridin-2-yl)-amine
—— 6-(3,4-dimethoxy-phenyl)-2-methyl-3-[4-(3-trifluoromethyl-pyrazol-1-yl)-phenyl]-imidazo[1,2-b]pyridazine 1023716-21-3 C25H20F3N5O2
6-(3,4-dimethoxy-phenyl)-2-methyl-3-[4-(3-trifluoromethyl-pyrazol-1-yl)-phenyl]-imidazo[1,2-b]pyridazine
—— 1-O-methyl-2,3-O-dibenzoyl-4-O-isobutyryl-5-methyl-α-rhamnose 112398-14-8 C26H30O8
1-O-methyl-2,3-O-dibenzoyl-4-O-isobutyryl-5-methyl-α-rhamnose
—— 5'-d(TXTTTTTT)-3'; X = 2'-deoxy-5-[3-({4-[(2,2-difluorocyclooct-3-yn-1-yl)methyl]benzoyl}amino)prop-1-yn-1-yl]uridine 1289361-06-3 C98H120F2N17O55P7
5'-d(TXTTTTTT)-3'; X = 2'-deoxy-5-[3-({4-[(2,2-difluorocyclooct-3-yn-1-yl)methyl]benzoyl}amino)prop-1-yn-1-yl]uridine
—— 3β-acetoxy-5-keto-5,6-secostigmastan-6-oic acid 14958-42-0 C31H52O5
3β-acetoxy-5-keto-5,6-secostigmastan-6-oic acid
—— (E)-3-(4-bromophenyl)-1-(4-((E)-3-[4-(trifluoromethyl)phenyl]-2-propenoyl)piperazino)-2-propen-1-one 1352051-02-5 C23H20BrF3N2O2
(E)-3-(4-bromophenyl)-1-(4-((E)-3-[4-(trifluoromethyl)phenyl]-2-propenoyl)piperazino)-2-propen-1-one
—— (E)-1-tosyl-4-((trimethylsilyl)methylene)pyrrolidin-3-ol 1427798-20-6 C15H23NO3SSi
(E)-1-tosyl-4-((trimethylsilyl)methylene)pyrrolidin-3-ol
—— 6,7-Dihydro-2-methyl-7-(4-nitrobenzoyl)-5H-pyrimido-[5,4-d][1]benzazepine 169879-00-9 C20H16N4O3
6,7-Dihydro-2-methyl-7-(4-nitrobenzoyl)-5H-pyrimido-[5,4-d][1]benzazepine
—— 1-(2,2-dioxido-1,2,3-oxathiazolidin-3-yl)hexadecan-1-one 1569834-07-6 C18H35NO4S
1-(2,2-dioxido-1,2,3-oxathiazolidin-3-yl)hexadecan-1-one
—— 1'-(1H-indazol-5-ylcarbonyl)-6,7-dimethylspiro[chromene-2,4'-piperidin]-4(3H)-one 1031413-14-5 C23H23N3O3
1'-(1H-indazol-5-ylcarbonyl)-6,7-dimethylspiro[chromene-2,4'-piperidin]-4(3H)-one
—— 2-[(3S)-1-[5-(cyclohexylcarbamoyl)-6-(2-pyrazin-2-ylethylsulfanyl)pyridin-2-yl]-3-piperidyl]acetic acid 1024035-73-1 C25H33N5O3S
2-[(3S)-1-[5-(cyclohexylcarbamoyl)-6-(2-pyrazin-2-ylethylsulfanyl)pyridin-2-yl]-3-piperidyl]acetic acid
—— N-[2,6-dichloro-4-(trifluoromethoxy)phenyl]-7-(1-ethylpropyl)-4-methoxy-1-methyl-1H-benzimidazol-2-amine 1022250-22-1 C21H22Cl2F3N3O2
N-[2,6-dichloro-4-(trifluoromethoxy)phenyl]-7-(1-ethylpropyl)-4-methoxy-1-methyl-1H-benzimidazol-2-amine
—— 1-{4-[3-(1-methyl-1H-pyrazol-3-yl)-9-phenyl[1,2,4]triazolo[3,4-f]-1,6-naphthyridin-8-yl]phenyl}cyclobutanamine 1032526-88-7 C29H25N7
1-{4-[3-(1-methyl-1H-pyrazol-3-yl)-9-phenyl[1,2,4]triazolo[3,4-f]-1,6-naphthyridin-8-yl]phenyl}cyclobutanamine
—— (S)-N-(5-chlorothiazol-2-yl)-2-(4-(cyclopentylsulfonyl)-6-methyl-2-oxopyridin-1(2H)-yl)-3-(tetrahydro-2H-pyran-4-yl)propanamide 1036205-65-8 C22H28ClN3O5S2
(S)-N-(5-chlorothiazol-2-yl)-2-(4-(cyclopentylsulfonyl)-6-methyl-2-oxopyridin-1(2H)-yl)-3-(tetrahydro-2H-pyran-4-yl)propanamide
—— adamantane-1-carboxylic acid N'-[2-(1-benzenesulfonyl-piperidin-3-yl)-acetyl]-hydrazide 1040878-82-7 C24H33N3O4S
adamantane-1-carboxylic acid N'-[2-(1-benzenesulfonyl-piperidin-3-yl)-acetyl]-hydrazide
—— 6-(2-methoxy-phenylethynyl)-2H-chromene-8-carboxylic acid [(R)-1-hydroxymethyl-2-(1H-indol-3-yl)-ethyl]-amide 1033763-46-0 C30H26N2O4
6-(2-methoxy-phenylethynyl)-2H-chromene-8-carboxylic acid [(R)-1-hydroxymethyl-2-(1H-indol-3-yl)-ethyl]-amide
—— 3,6-bis(1-methyl-1H-pyrazol-4-yl)-4-{2-[(2S)-piperidin-2-yl]ethoxy}quinoline 1021911-71-6 C24H28N6O
3,6-bis(1-methyl-1H-pyrazol-4-yl)-4-{2-[(2S)-piperidin-2-yl]ethoxy}quinoline
—— 6-{[1-(4-fluorophenyl)-1H-indazol-4-yl]amino}-9,9-dimethyl-7-(trifluoromethyl)-6,7,8,9-tetrahydro-naphtho[1,2-d]-1,3-dioxol-7-ol 1021536-78-6 C27H23F4N3O3
6-{[1-(4-fluorophenyl)-1H-indazol-4-yl]amino}-9,9-dimethyl-7-(trifluoromethyl)-6,7,8,9-tetrahydro-naphtho[1,2-d]-1,3-dioxol-7-ol
—— (R)-4-benzyl-3-(3-bromophenethyl)-1-(4-((S)-3-(3-fluorophenethyl)-2-iminoimidazolidin-4-yl)butyl)imidazolidin-2-imine 1510811-18-3 C33H40BrFN6
(R)-4-benzyl-3-(3-bromophenethyl)-1-(4-((S)-3-(3-fluorophenethyl)-2-iminoimidazolidin-4-yl)butyl)imidazolidin-2-imine
—— N-(naphthalen-1-yl)sulfonyl-3-amino-4-oxo-5-(5-(2,6-dichlorophenylmethyl)tetrazol-2-yl)pentanoic acid 192460-04-1 C23H19Cl2N5O5S
N-(naphthalen-1-yl)sulfonyl-3-amino-4-oxo-5-(5-(2,6-dichlorophenylmethyl)tetrazol-2-yl)pentanoic acid
—— 3'-(3-(1-(4-(tert-butyl)benzyl)-4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)propyl)-[1,1'-biphenyl]-3-carboxylic acid 1616372-38-3 C31H35N3O3
3'-(3-(1-(4-(tert-butyl)benzyl)-4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)propyl)-[1,1'-biphenyl]-3-carboxylic acid
—— 2-[(2R)-2-(4-chlorophenyl)piperazin-1-yl]-5-(2-hydroxyethyl)benzonitrile 1427711-63-4 C19H20ClN3O
2-[(2R)-2-(4-chlorophenyl)piperazin-1-yl]-5-(2-hydroxyethyl)benzonitrile
—— tert-Butyl [1-(2-benzoyl benzyl)-5-methyl-3-phenyl-1H-pyrazol-4-yl]acetate 1379446-02-2 C30H30N2O3
tert-Butyl [1-(2-benzoyl benzyl)-5-methyl-3-phenyl-1H-pyrazol-4-yl]acetate
—— 5-(Methoxymethyl)-3-(2-piperazin-1-ylpyrimidin-4-yl)-1,2,4-oxadiazole;hydrochloride 1177093-11-6 C12H17ClN6O2
5-(Methoxymethyl)-3-(2-piperazin-1-ylpyrimidin-4-yl)-1,2,4-oxadiazole;hydrochloride
—— N-(1-{[7-(3-hydroxypropyl)-2-naphthyl]methyl}piperidin-4-yl)-3-methoxybenzamide 1018072-70-2 C27H32N2O3
N-(1-{[7-(3-hydroxypropyl)-2-naphthyl]methyl}piperidin-4-yl)-3-methoxybenzamide