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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-(2-fluoro-phenyl)-5-[3-(4-methoxy-phenyl)-isoxazol-5-ylmethyl]-5H-imidazo[4,5-d]pyridazine 1105058-82-9 C22H16FN5O2
2-(2-fluoro-phenyl)-5-[3-(4-methoxy-phenyl)-isoxazol-5-ylmethyl]-5H-imidazo[4,5-d]pyridazine
—— 2-(3-fluoro-4-methylbenzyl)-4,5-dihydroxyisoindoline-1,3-dione 1123213-65-9 C16H12FNO4
2-(3-fluoro-4-methylbenzyl)-4,5-dihydroxyisoindoline-1,3-dione
—— N-cyclohexyl 4-(1-(4-(methylsulfonyl)phenyl)-2-oxo-1,2-dihydropyridin-4-yloxy)piperidine-1-carboxamide 1104446-30-1 C24H31N3O5S
N-cyclohexyl 4-(1-(4-(methylsulfonyl)phenyl)-2-oxo-1,2-dihydropyridin-4-yloxy)piperidine-1-carboxamide
—— 6-{[(4-bromophenyl)methyl]amino}-5-(4-fluorophenyl)-1-methyl-1H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one 1123783-99-2 C19H15BrFN5O
6-{[(4-bromophenyl)methyl]amino}-5-(4-fluorophenyl)-1-methyl-1H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
—— N-(2-chloro-benzyl)-2-(3,4-dichloro-phenyl)-4-[4-(ethyl-methanesulfonyl-amino)-piperidin-1-yl]-2,N-dimethyl-butyramide 1131738-21-0 C27H36Cl3N3O3S
N-(2-chloro-benzyl)-2-(3,4-dichloro-phenyl)-4-[4-(ethyl-methanesulfonyl-amino)-piperidin-1-yl]-2,N-dimethyl-butyramide
—— N-((6-tert.-butyl-2-(4-methylpiperidin-1-yl)pyridin-3-yl)methyl)-2-(2-thioxo-2,3-dihydrobenzo[d]thiazol-6-yl)propanamide 1072149-39-3 C26H34N4OS2
N-((6-tert.-butyl-2-(4-methylpiperidin-1-yl)pyridin-3-yl)methyl)-2-(2-thioxo-2,3-dihydrobenzo[d]thiazol-6-yl)propanamide
—— 6-[[4-[[(3R)-pyrrolidin-3-yl]amino]pyrrolidin-3-yl]methyl]pyridin-2-amine 1111394-12-7 C14H23N5
6-[[4-[[(3R)-pyrrolidin-3-yl]amino]pyrrolidin-3-yl]methyl]pyridin-2-amine
—— N-[2-[[2-[4-[bis(2-hydroxyethyl)amino]anilino]-5-chloropyrimidin-4-yl]amino]phenyl]cyclopropanecarboxamide 1035561-13-7 C24H27ClN6O3
N-[2-[[2-[4-[bis(2-hydroxyethyl)amino]anilino]-5-chloropyrimidin-4-yl]amino]phenyl]cyclopropanecarboxamide
—— 2-bromo-3-(4-pentylamino-phenyl)-4,5,6,6a-tetrahydro-3aH-pentalen-1-one 1104634-17-4 C19H24BrNO
2-bromo-3-(4-pentylamino-phenyl)-4,5,6,6a-tetrahydro-3aH-pentalen-1-one
—— N-(2-{5-methoxy-2-[(2,3-dihydro-1H-indol-1-yl)-methyl]-1H-indol-3-yl}ethyl)acetamide 1338474-10-4 C22H25N3O2
N-(2-{5-methoxy-2-[(2,3-dihydro-1H-indol-1-yl)-methyl]-1H-indol-3-yl}ethyl)acetamide
—— N3-[(1S,2R)-1-benzyl-2-hydroxy-3-{[3-(trifluoromethyl)benzyl]amino}propyl]-1-ethyl-N5-hexyl-N5-methyl-1H-pyrazole-3,5-dicarboxamide 1106668-43-2 C32H42F3N5O3
N3-[(1S,2R)-1-benzyl-2-hydroxy-3-{[3-(trifluoromethyl)benzyl]amino}propyl]-1-ethyl-N5-hexyl-N5-methyl-1H-pyrazole-3,5-dicarboxamide
—— 4-(2-fluorodibenzo[b,f][1,4]oxazepin-11-yl)-N-hydroxybenzamide 1024007-26-8 C20H13FN2O3
4-(2-fluorodibenzo[b,f][1,4]oxazepin-11-yl)-N-hydroxybenzamide
—— N,N-diisobutyl-[α,α,β,β-d4]-tryptamine 1174656-41-7 C18H28N2
N,N-diisobutyl-[α,α,β,β-d4]-tryptamine
—— N3-[(1S,2R)-1-(3,5-difluorobenzyl)-2-hydroxy-3-{[(1S)-7-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl]amino}propyl]-1-ethyl-N5-heptyl-N5-methyl-1H-pyrazole-3,5-dicarboxamide 1106668-48-7 C36H49F2N5O4
N3-[(1S,2R)-1-(3,5-difluorobenzyl)-2-hydroxy-3-{[(1S)-7-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl]amino}propyl]-1-ethyl-N5-heptyl-N5-methyl-1H-pyrazole-3,5-dicarboxamide
—— 4-(dibenzo[b,f][1,4]oxazepin-11-yl)-2-fluoro-N-hydroxy-benzamide 1024007-48-4 C20H13FN2O3
4-(dibenzo[b,f][1,4]oxazepin-11-yl)-2-fluoro-N-hydroxy-benzamide
—— N-[(2S)-6-[(oxan-4-ylmethylamino)methyl]-1,2,3,4-tetrahydronaphthalen-2-yl]-4-[[(2S)-oxolan-2-yl]methoxy]benzamide 1119018-75-5 C29H38N2O4
N-[(2S)-6-[(oxan-4-ylmethylamino)methyl]-1,2,3,4-tetrahydronaphthalen-2-yl]-4-[[(2S)-oxolan-2-yl]methoxy]benzamide
—— 4-chloro-1-pyrimidin-2-yl-1H-indole-3-carboxylic acid [2-(4-bromo-phenyl)-ethyl]-amide 1119282-28-8 C21H16BrClN4O
4-chloro-1-pyrimidin-2-yl-1H-indole-3-carboxylic acid [2-(4-bromo-phenyl)-ethyl]-amide
—— 2-(4-(5-(4-(difluoromethoxy)phenyl)pyrimidin-2-ylamino)phenyl)-3-hydroxy-1-(4-methylpiperazin-1-yl)propan-1-one 1123513-88-1 C25H27F2N5O3
2-(4-(5-(4-(difluoromethoxy)phenyl)pyrimidin-2-ylamino)phenyl)-3-hydroxy-1-(4-methylpiperazin-1-yl)propan-1-one
—— 1-{4-[1-(1-benzylpiperidin-4-yl)-4-morpholin-4-yl-1H-pyrazolo[3,4-d]pyrimidin-6-yl]phenyl}-3-(1-methylpiperidin-4-yl)urea 1062162-93-9 C34H43N9O2
1-{4-[1-(1-benzylpiperidin-4-yl)-4-morpholin-4-yl-1H-pyrazolo[3,4-d]pyrimidin-6-yl]phenyl}-3-(1-methylpiperidin-4-yl)urea
—— 1-(4-(3-methoxybenzyl)thiazol-2-yl)-4-(pyridin-3-ylsulfonyl)piperazine 1114770-41-0 C20H22N4O3S2
1-(4-(3-methoxybenzyl)thiazol-2-yl)-4-(pyridin-3-ylsulfonyl)piperazine
—— Ethyl 4-isobutyl-5-methyl-6-oxo-2-(trifluoromethyl)-1,4,5,6-tetrahydropyridine-3-carboxylate 1130345-41-3 C14H20F3NO3
Ethyl 4-isobutyl-5-methyl-6-oxo-2-(trifluoromethyl)-1,4,5,6-tetrahydropyridine-3-carboxylate
—— [4-[[(4-cyanophenyl)methylidenehydrazinylidene]methyl]-2-methylphenyl] prop-2-enoate 1050428-24-4 C19H15N3O2
[4-[[(4-cyanophenyl)methylidenehydrazinylidene]methyl]-2-methylphenyl] prop-2-enoate
—— N-(4-((2-(3-(3-fluorobenzyl)ureido)thiazol-4-yl)methylsulfonyl)phenyl)acetamide 1108651-98-4 C20H19FN4O4S2
N-(4-((2-(3-(3-fluorobenzyl)ureido)thiazol-4-yl)methylsulfonyl)phenyl)acetamide
—— N-[((2R,4R)-1-cyano-4-{[(2,5-dibromophenyl)sulfonyl]amino}-2-pyrrolidinyl)methyl]-4-fluorobenzamide 1123308-09-7 C19H17Br2FN4O3S
N-[((2R,4R)-1-cyano-4-{[(2,5-dibromophenyl)sulfonyl]amino}-2-pyrrolidinyl)methyl]-4-fluorobenzamide
—— 1'-isobutyl-piperidin-4'-yl-spiro(6-(pyridin-2-ylcarboxamido)-2H-benzopyran-2-yl) 1124313-30-9 C23H27N3O2
1'-isobutyl-piperidin-4'-yl-spiro(6-(pyridin-2-ylcarboxamido)-2H-benzopyran-2-yl)
—— N-[5-(3-furyl)[1,2,4]triazolo[1,5-a]pyridin-2-yl]-4-isobutylbenzamide 1124381-23-2 C21H20N4O2
N-[5-(3-furyl)[1,2,4]triazolo[1,5-a]pyridin-2-yl]-4-isobutylbenzamide
—— 5-(4-methyl-5-trifluoromethyl-isoxazol-3-yl)-thiophene-2-carboxylic acid cyclohexylamide 1124198-47-5 C16H17F3N2O2S
5-(4-methyl-5-trifluoromethyl-isoxazol-3-yl)-thiophene-2-carboxylic acid cyclohexylamide
—— 4-(5-ethyl-5H-dibenzo[b,e][1,4]diazepin-11-yl)-N-hydroxybenzamide 1024007-44-0 C22H19N3O2
4-(5-ethyl-5H-dibenzo[b,e][1,4]diazepin-11-yl)-N-hydroxybenzamide
—— 5-(4-methyl-5-trifluoromethyl-isoxazol-3-yl)-thiophene-2-carboxylic acid methylprop-2-ynyl-amide 1124198-31-7 C14H11F3N2O2S
5-(4-methyl-5-trifluoromethyl-isoxazol-3-yl)-thiophene-2-carboxylic acid methylprop-2-ynyl-amide
—— 6-{[(1R)-1-cyclobutylethyl]amino}-8-[2-methoxy-5-(1-methylethyl)phenyl]-7-[4-(trifluoromethyl)benzyl]-7H-purine-2-carboxylic acid 1621539-24-9 C30H32F3N5O3
6-{[(1R)-1-cyclobutylethyl]amino}-8-[2-methoxy-5-(1-methylethyl)phenyl]-7-[4-(trifluoromethyl)benzyl]-7H-purine-2-carboxylic acid
—— [(R)-2-(5-fluoro-7-(tetrahydropyran-4-yl)amino-1H-indol-2-yl)-4,5-dihydro-thiazol-4-yl]-acetic acid 1120342-86-0 C18H20FN3O3S
[(R)-2-(5-fluoro-7-(tetrahydropyran-4-yl)amino-1H-indol-2-yl)-4,5-dihydro-thiazol-4-yl]-acetic acid
—— (S)-6-chloro-N4-(3-fluoro-4-(morpholin-2-yl)phenyl)pyridine-2,4-dicarboxamide hydrochloride 1415757-17-3 C17H16ClFN4O3*ClH
(S)-6-chloro-N4-(3-fluoro-4-(morpholin-2-yl)phenyl)pyridine-2,4-dicarboxamide hydrochloride
—— 6-(1-allyl-2-benzyl-3-oxo-2,3-dihydro-1H-indazol-5-yl)-4-chloro-7,8-dihydropyrimido[5,4-f][1,4]oxazepin-5(6H)-one 1415345-31-1 C24H20ClN5O3
6-(1-allyl-2-benzyl-3-oxo-2,3-dihydro-1H-indazol-5-yl)-4-chloro-7,8-dihydropyrimido[5,4-f][1,4]oxazepin-5(6H)-one
—— tert-butyl 2-(6-(3-chlorophenyl)-5-methylpyridin-3-ylamino)-5-methylbenzoate 1119091-02-9 C24H25ClN2O2
tert-butyl 2-(6-(3-chlorophenyl)-5-methylpyridin-3-ylamino)-5-methylbenzoate
—— 1-(Cyclobutylidenemethyl)-3-nitrobenzene 1114779-90-6 C11H11NO2
1-(Cyclobutylidenemethyl)-3-nitrobenzene
—— 3-[(R)-2-(7-cyclopentylamino-1H-indol-2-yl)-4,5-dihydro-thiazol-4-yl]-propionic acid 1120343-24-9 C19H23N3O2S
3-[(R)-2-(7-cyclopentylamino-1H-indol-2-yl)-4,5-dihydro-thiazol-4-yl]-propionic acid
—— 5-[4-({4-[3-(2-furyl)-1H-1,2,4-triazol-5-yl]piperidin-1-yl}methyl)phenyl]-6-phenylpyrazolo[1,5-a]pyrimidine 1116117-98-6 C30H27N7O
5-[4-({4-[3-(2-furyl)-1H-1,2,4-triazol-5-yl]piperidin-1-yl}methyl)phenyl]-6-phenylpyrazolo[1,5-a]pyrimidine
—— {4-[4-(ethyloxy)-1,3-dioxo-9-(2-methylpropyl)-1,3-dihydro-2H-benzo[f]isoindol-2-yl]phenyl}acetic acid 1114974-17-2 C26H25NO5
{4-[4-(ethyloxy)-1,3-dioxo-9-(2-methylpropyl)-1,3-dihydro-2H-benzo[f]isoindol-2-yl]phenyl}acetic acid
—— 13-cyclohexyl-6-[4-(3,7-dioxa-9-azabicyclo[3.3.1]non-9-ylcarbonyl)-1-methyl-1H-pyrazol-5-yl]-3-methoxy-N-[(1-methylethyl)sulfonyl]-7H-indolo[2,1-a][2]benzazepine-10-carboxamide 1127235-61-3 C39H45N5O7S
13-cyclohexyl-6-[4-(3,7-dioxa-9-azabicyclo[3.3.1]non-9-ylcarbonyl)-1-methyl-1H-pyrazol-5-yl]-3-methoxy-N-[(1-methylethyl)sulfonyl]-7H-indolo[2,1-a][2]benzazepine-10-carboxamide
—— 1-ethyl-4-(3-methoxyphenyl)-4H-[1,2,4]triazolo[4,3-a]quinazolin-5-one 1105576-14-4 C18H16N4O2
1-ethyl-4-(3-methoxyphenyl)-4H-[1,2,4]triazolo[4,3-a]quinazolin-5-one
—— 1-(4-(azetidine-1-ylcarbonyl)-5-(2-fluoro-4-iodophenylamino)-1-methyl-1H-pyrrol-2-yl)ethanone 1023742-38-2 C17H17FIN3O2
1-(4-(azetidine-1-ylcarbonyl)-5-(2-fluoro-4-iodophenylamino)-1-methyl-1H-pyrrol-2-yl)ethanone
—— 4'-{[methyl-(3-methyl-butyl)amino]methyl}-biphenyl-3-carboxylic acid amide 1131794-63-2 C20H26N2O
4'-{[methyl-(3-methyl-butyl)amino]methyl}-biphenyl-3-carboxylic acid amide
—— 1-(3-fluorobenzyl)-3-(4-(methylsulfonylmethyl)thiazol-2-yl)urea 1108651-91-7 C13H14FN3O3S2
1-(3-fluorobenzyl)-3-(4-(methylsulfonylmethyl)thiazol-2-yl)urea
—— 4-[3-[(1-acetylpyrrolidin-3-yl)methyl]-7-methylimidazo[1,2-a]pyridin-2-yl]-N,3-dimethylbenzamide 1621165-07-8 C24H28N4O2
4-[3-[(1-acetylpyrrolidin-3-yl)methyl]-7-methylimidazo[1,2-a]pyridin-2-yl]-N,3-dimethylbenzamide
—— 4-chloro-N-[2-(4-chlorophenyl)-4-methylpentyl]-1-[2-(dimethylamino)ethyl]-1H-indole-3-carboxamide 1119281-88-7 C25H31Cl2N3O
4-chloro-N-[2-(4-chlorophenyl)-4-methylpentyl]-1-[2-(dimethylamino)ethyl]-1H-indole-3-carboxamide
—— N-[4-(4-fluorophenyl)-2,2,5-trimethyl-2H-chromen-7-yl]methanesulfonamide 1110663-68-7 C19H20FNO3S
N-[4-(4-fluorophenyl)-2,2,5-trimethyl-2H-chromen-7-yl]methanesulfonamide
—— {4-[2-(4-trifluoromethylphenyl)-pyrimidin-4-yl-methoxy]-phenoxy}-acetic acid 1104759-26-3 C20H15F3N2O4
{4-[2-(4-trifluoromethylphenyl)-pyrimidin-4-yl-methoxy]-phenoxy}-acetic acid
—— N-((2-(3-(3-fluorobenzyl)ureido)thiazol-4-yl)methyl)-N-methylquinoxaline-2-carboxamide 1108707-50-1 C22H19FN6O2S
N-((2-(3-(3-fluorobenzyl)ureido)thiazol-4-yl)methyl)-N-methylquinoxaline-2-carboxamide
—— 3-chloro-6-thiophen-2-yl-8-trifluoromethyl-imidazo[1,2-a]pyridine-2-carboxylic acid (thiophen-2-ylmethyl)-amide 1121051-71-5 C18H11ClF3N3OS2
3-chloro-6-thiophen-2-yl-8-trifluoromethyl-imidazo[1,2-a]pyridine-2-carboxylic acid (thiophen-2-ylmethyl)-amide
—— (S)-3-(1H-indol-3-yl)-N1-propylpropane-1,2-diamine 1116686-81-7 C14H21N3
(S)-3-(1H-indol-3-yl)-N1-propylpropane-1,2-diamine