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中文名称 英文名称 CAS号 化学式 结构式图片
—— ethyl 4-[4-oxo-2-[(2-oxoindol-3-yl)hydrazinylidene]-1,3-thiazolidin-3-yl]benzoate 1292780-49-4 C20H16N4O4S
ethyl 4-[4-oxo-2-[(2-oxoindol-3-yl)hydrazinylidene]-1,3-thiazolidin-3-yl]benzoate
—— 5-(3,5-dibromo-4-hydroxyphenyl)-N-(3-(trifluoromethoxy)benzyl)-1,2,4-oxadiazole-3-carboxamide 1191252-71-7 C17H10Br2F3N3O4
5-(3,5-dibromo-4-hydroxyphenyl)-N-(3-(trifluoromethoxy)benzyl)-1,2,4-oxadiazole-3-carboxamide
—— 6-Bromo-N-methylpyridine-3-sulfonamide 1215943-03-5 C6H7BrN2O2S
6-Bromo-N-methylpyridine-3-sulfonamide
—— 4-{3-[3-({[(2R)-1-ethylpyrrolidin-2-yl]methyl}amino)-3-oxopropyl]-5-(3-fluorophenyl)-1H-pyrazol-1-yl}benzoic acid 1353545-19-3 C26H29FN4O3
4-{3-[3-({[(2R)-1-ethylpyrrolidin-2-yl]methyl}amino)-3-oxopropyl]-5-(3-fluorophenyl)-1H-pyrazol-1-yl}benzoic acid
—— 2-{[3-fluoro-4-(4-hydroxypiperidino)]phenylamino}-6-[(2-methyl-4,5-dihydro)imidazol-1-yl]-3-nitropyridine 1229015-85-3 C20H23FN6O3
2-{[3-fluoro-4-(4-hydroxypiperidino)]phenylamino}-6-[(2-methyl-4,5-dihydro)imidazol-1-yl]-3-nitropyridine
—— 7-(2-methoxyethoxy)-N-(1-((tetrahydro-2H-pyran-4-yl)methyl)-1H-indazol-4-yl)imidazo[1,2-a]pyridine-3-carboxamide 1383472-57-8 C24H27N5O4
7-(2-methoxyethoxy)-N-(1-((tetrahydro-2H-pyran-4-yl)methyl)-1H-indazol-4-yl)imidazo[1,2-a]pyridine-3-carboxamide
—— 4-[5-chloro-4-(2,5-difluoro-phenyl)-thiophene-2-sulfonylamino]-2-hydroxy-benzoic acid 1353434-82-8 C17H10ClF2NO5S2
4-[5-chloro-4-(2,5-difluoro-phenyl)-thiophene-2-sulfonylamino]-2-hydroxy-benzoic acid
—— 4-(3-chloro-2-methyl-benzenesulfonylamino)-2-hydroxy-benzoic acid 1353434-97-5 C14H12ClNO5S
4-(3-chloro-2-methyl-benzenesulfonylamino)-2-hydroxy-benzoic acid
—— 2-[(3-fluoro-4-piperidino)phenylamino]-6-(isobutylamino)-3-nitropyridine 1229015-70-6 C20H26FN5O2
2-[(3-fluoro-4-piperidino)phenylamino]-6-(isobutylamino)-3-nitropyridine
—— N-(2-chloro-3-(2-cyclopropyl-5-(2-(methylthio)pyrimidin-4-yl)thiazol-4-yl)phenyl)pivalamide 1353576-13-2 C22H23ClN4OS2
N-(2-chloro-3-(2-cyclopropyl-5-(2-(methylthio)pyrimidin-4-yl)thiazol-4-yl)phenyl)pivalamide
—— N-cyclopropyl-4-{8-[(3-hydroxypropyl)amino]-6-(pyridin-4-yl)imidazo[1,2-a]pyrazin-3-yl}benzamide 1383118-91-9 C24H24N6O2
N-cyclopropyl-4-{8-[(3-hydroxypropyl)amino]-6-(pyridin-4-yl)imidazo[1,2-a]pyrazin-3-yl}benzamide
—— 2-hydroxy-4-{[3-(2,3,6-trifluorophenyl)benzene]sulfonamido}benzoic acid 1353434-25-9 C19H12F3NO5S
2-hydroxy-4-{[3-(2,3,6-trifluorophenyl)benzene]sulfonamido}benzoic acid
—— 2-{[3-fluoro-4-(3-hydroxymethylpiperidino)]phenylamino}-6-(t-butylamino)-3-nitropyridine 1229016-23-2 C21H28FN5O3
2-{[3-fluoro-4-(3-hydroxymethylpiperidino)]phenylamino}-6-(t-butylamino)-3-nitropyridine
—— 4-[4-(2-aminopyrimidin-5-yl)phenyl]-N-[3-(trifluoromethoxy)phenyl]tetrahydro-2H-pyran-4-carboxamide 1382482-43-0 C23H21F3N4O3
4-[4-(2-aminopyrimidin-5-yl)phenyl]-N-[3-(trifluoromethoxy)phenyl]tetrahydro-2H-pyran-4-carboxamide
—— 2-((1H-indol-3-yl)methyl)-7-(4-methoxypyridin-2-yl)-2,7-diazaspiro[4,4]nonan-1-one 1383574-52-4 C22H24N4O2
2-((1H-indol-3-yl)methyl)-7-(4-methoxypyridin-2-yl)-2,7-diazaspiro[4,4]nonan-1-one
—— —— 1055895-25-4 C56H44N2O4
—— quinolin-6-yl-carbamic acid dydrogesterone-11-yl ester 1059179-64-4 C31H34N2O4
quinolin-6-yl-carbamic acid dydrogesterone-11-yl ester
—— —— 1053184-24-9 C53H64N10O13S2
—— 3-(4-bromophenyl)-1-dimethylamino-3-phenylthio-2-propene (E) hydrochloride 102360-65-6 C17H18BrNS*ClH
3-(4-bromophenyl)-1-dimethylamino-3-phenylthio-2-propene (E) hydrochloride
—— (8RS)-8-methoxy-6-methyl-5,6,7,8-tetrahydro-4H-thieno[2,3-d]azepine-2-carboxylic acid [(1R)-1-(5-chloro-1H-benzimidazol-2-yl)-2-methoxy-ethyl]-amide trifluoroacetate 1080026-74-9 C2HF3O2*C21H25ClN4O3S
(8RS)-8-methoxy-6-methyl-5,6,7,8-tetrahydro-4H-thieno[2,3-d]azepine-2-carboxylic acid [(1R)-1-(5-chloro-1H-benzimidazol-2-yl)-2-methoxy-ethyl]-amide trifluoroacetate
—— 2-(4'-Methoxystilben-4-yl)-naphtho<1,2-d>triazol 16184-17-1 C25H19N3O
2-(4'-Methoxystilben-4-yl)-naphtho<1,2-d>triazol
—— 2-(5-Acetoxymethyl-3-hydroxy-2-methyl-pyridin-4-yl)-[1,3]thiazinane-4-carboxylic acid 19708-19-1 C14H18N2O5S
2-(5-Acetoxymethyl-3-hydroxy-2-methyl-pyridin-4-yl)-[1,3]thiazinane-4-carboxylic acid
—— —— 1079170-06-1 C22H26N4O2
—— —— 1079176-37-6 C26H34N4O
—— N-(Carboxymethyl)-N-(3-mercapto-2(S)-methyl-1-oxopropyl)-β-alanine 1-cyclohexyl ester adamantanamine salt 133273-50-4 C10H17N*C15H25NO5S
N-(Carboxymethyl)-N-(3-mercapto-2(S)-methyl-1-oxopropyl)-β-alanine 1-cyclohexyl ester adamantanamine salt
—— (6R,7R)-7-[(R)-2-(4-Ethyl-2,3-dioxopiperazin-1-yl)carbonylamino-2-phenylacetamido]-7-formamido-3-(5-hydroxy-4-oxo-1,4-dihydropyridin-2-yl)carbonyloxymethylceph-3-em-4-carboxylic acid 118680-33-4 C30H29N7O12S
(6R,7R)-7-[(R)-2-(4-Ethyl-2,3-dioxopiperazin-1-yl)carbonylamino-2-phenylacetamido]-7-formamido-3-(5-hydroxy-4-oxo-1,4-dihydropyridin-2-yl)carbonyloxymethylceph-3-em-4-carboxylic acid
—— Sodium (6R,7R)-7-[(R)-2-(4-Ethyl-2,3-dioxopiperazin-1-yl)carbonylamino-2-phenylacetamido]-7-formamido-3-(3,4, 5-trihydroxybenzoyloxy)methylceph-3-em-4-carboxylate 118708-53-5 C31H29N6O13S*Na
Sodium (6R,7R)-7-[(R)-2-(4-Ethyl-2,3-dioxopiperazin-1-yl)carbonylamino-2-phenylacetamido]-7-formamido-3-(3,4, 5-trihydroxybenzoyloxy)methylceph-3-em-4-carboxylate
—— 5-(2-((dimethylamino)methyl)pyridin-4-yloxy)-4-fluoro-2-methyl-N-(3-(trifluoromethyl)phenyl)-1H-indole-1-carboxamide 1229449-51-7 C25H22F4N4O2
5-(2-((dimethylamino)methyl)pyridin-4-yloxy)-4-fluoro-2-methyl-N-(3-(trifluoromethyl)phenyl)-1H-indole-1-carboxamide
—— N-(4-(4-(3-chlorobenzyloxy)-3-fluorophenylamino)-7-methoxyquinazolin-6-yl)-2-(piperidin-4-ylidene)acetamide 1005195-69-6 C29H27ClFN5O3
N-(4-(4-(3-chlorobenzyloxy)-3-fluorophenylamino)-7-methoxyquinazolin-6-yl)-2-(piperidin-4-ylidene)acetamide
—— (S)-4-(4-fluoro-phenyl)-1-methyl-6-oxo-1,4,5,6-tetrahydro-pyridine-3-carboxylic acid [4-chloro-5-(2-hydroxy-ethoxy)-2-methyl-phenyl]-amide 1232505-48-4 C22H22ClFN2O4
(S)-4-(4-fluoro-phenyl)-1-methyl-6-oxo-1,4,5,6-tetrahydro-pyridine-3-carboxylic acid [4-chloro-5-(2-hydroxy-ethoxy)-2-methyl-phenyl]-amide
—— methyl 4-(2-chloro-5-methylphenoxy)-6-(2,3-difluorophenyl)nicotinate 1013914-24-3 C20H14ClF2NO3
methyl 4-(2-chloro-5-methylphenoxy)-6-(2,3-difluorophenyl)nicotinate
—— 6-(4-(3-(tetrahydro-2H-pyran-4-yl)pyridin-2-yloxy)phenylamino)nicotinonitrile 1231923-41-3 C22H20N4O2
6-(4-(3-(tetrahydro-2H-pyran-4-yl)pyridin-2-yloxy)phenylamino)nicotinonitrile
—— methyl 3-{(S)-(3-chlorophenyl)[(2-{[(methyloxy)carbonyl]amino}ethyl)oxy]methyl}-4-methylbenzoate 1093865-24-7 C20H22ClNO5
methyl 3-{(S)-(3-chlorophenyl)[(2-{[(methyloxy)carbonyl]amino}ethyl)oxy]methyl}-4-methylbenzoate
—— 6-(2-ethyl-8-methoxyquinolin-5-yl)-5-methyl-2-[4-[4-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)phenoxy]butyl]-4,5-dihydro-2H-pyridazin-3-one 1094102-24-5 C31H35N5O4
6-(2-ethyl-8-methoxyquinolin-5-yl)-5-methyl-2-[4-[4-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)phenoxy]butyl]-4,5-dihydro-2H-pyridazin-3-one
—— N-cyclopropyl-4-[5-fluoro-4-[[2-methyl-1-oxo-1-(2,2,2-trifluoroethylamino)propan-2-yl]amino]pyrimidin-2-yl]-1H-pyrrole-2-carboxamide 1062564-48-0 C18H20F4N6O2
N-cyclopropyl-4-[5-fluoro-4-[[2-methyl-1-oxo-1-(2,2,2-trifluoroethylamino)propan-2-yl]amino]pyrimidin-2-yl]-1H-pyrrole-2-carboxamide
—— N-[((1R,2S,5S)-3-{[2-methyl-5-(3-methylphenyl)-1,3-thiazol-4-yl]carbonyl}-3-azabicyclo[3.1.0]hex-2-yl)methyl]-1,3-benzoxazol-2-amine 1092505-44-6 C25H24N4O2S
N-[((1R,2S,5S)-3-{[2-methyl-5-(3-methylphenyl)-1,3-thiazol-4-yl]carbonyl}-3-azabicyclo[3.1.0]hex-2-yl)methyl]-1,3-benzoxazol-2-amine
—— sodium;3-[4-[[1-(benzenesulfonyl)-3,4-dihydro-2H-quinolin-8-yl]methoxy]-2-fluorophenyl]propanoate 1030841-57-6 C25H23FNO5S*Na
sodium;3-[4-[[1-(benzenesulfonyl)-3,4-dihydro-2H-quinolin-8-yl]methoxy]-2-fluorophenyl]propanoate
—— (S)-2-(1-(2-methoxyethyl)piperidin-4-ylidene)-N-(4-(1-phenylethylamino)quinazolin-6-yl)acetamide 1005195-50-5 C26H31N5O2
(S)-2-(1-(2-methoxyethyl)piperidin-4-ylidene)-N-(4-(1-phenylethylamino)quinazolin-6-yl)acetamide
—— N-(cyclopropylmethyl)-12-oxo-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9-triene-10-carboxamide 1029685-62-8 C14H15N3O2S
N-(cyclopropylmethyl)-12-oxo-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9-triene-10-carboxamide
—— (2S)-2-amino-3-[(5-chloro-2-fluoro-4-{5-[6-(trifluoromethyl)imidazo[1,2-a]pyridin-2-yl]-1,3,4-thiadiazol-2-yl}phenyl)oxy]propan-1-ol 1228374-85-3 C19H14ClF4N5O2S
(2S)-2-amino-3-[(5-chloro-2-fluoro-4-{5-[6-(trifluoromethyl)imidazo[1,2-a]pyridin-2-yl]-1,3,4-thiadiazol-2-yl}phenyl)oxy]propan-1-ol
—— N-(4-(3-chloro-4-fluorophenylamino)-3-cyano-7-ethoxyquinolin-6-yl)-2-(1-methylpiperidin-4-ylidene)acetamide 1005195-88-9 C26H25ClFN5O2
N-(4-(3-chloro-4-fluorophenylamino)-3-cyano-7-ethoxyquinolin-6-yl)-2-(1-methylpiperidin-4-ylidene)acetamide
—— (S)-2-(4-fluoro-phenyl)-4-oxo-3,4-dihydro-2H-pyridine-1-carboxylic acid (3-hydroxymethyl-2-methyl-phenyl)-amide 1232688-02-6 C20H19FN2O3
(S)-2-(4-fluoro-phenyl)-4-oxo-3,4-dihydro-2H-pyridine-1-carboxylic acid (3-hydroxymethyl-2-methyl-phenyl)-amide
—— 9-fluoro-6-{[(3R,4S)-3-fluoropiperidin-4-yl]amino}benzo[c]-1,6-naphthyridin-1(2H)-one 1058126-36-5 C17H16F2N4O
9-fluoro-6-{[(3R,4S)-3-fluoropiperidin-4-yl]amino}benzo[c]-1,6-naphthyridin-1(2H)-one
—— 2-methyl-3-(morpholine-4-carbonyl)-7-[1,2-dihydro-2-oxo-3H-indol-(Z)-3-ylidene]-4,5,6,7-tetrahydro-1H-indole 1032265-84-1 C22H23N3O3
2-methyl-3-(morpholine-4-carbonyl)-7-[1,2-dihydro-2-oxo-3H-indol-(Z)-3-ylidene]-4,5,6,7-tetrahydro-1H-indole
—— 7-((6-fluoro-3H-pyrazolo[3,4-c]quinolin-4-yl)amino)-3,4-dihydroquinolin-2(1H)-one 1604673-91-7 C19H14FN5O
7-((6-fluoro-3H-pyrazolo[3,4-c]quinolin-4-yl)amino)-3,4-dihydroquinolin-2(1H)-one
—— 6-chloro-N-[6-(propan-2-yloxy)-1H-indazol-5-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-amine 1589508-15-5 C16H15ClN6O
6-chloro-N-[6-(propan-2-yloxy)-1H-indazol-5-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-amine
—— 2-(1-Methyl-1-carboxy-ethyl)-1-isobutyryl-1,2,3,4-tetrahydro-chinolin 17211-19-7 C17H23NO3
2-(1-Methyl-1-carboxy-ethyl)-1-isobutyryl-1,2,3,4-tetrahydro-chinolin
—— 8-(1-Methylpyrazol-4-yl)-6-[4-(trifluoromethoxy)phenyl]-1,2,3,4-tetrahydro-1,6-naphthyridin-5-one 1590403-08-9 C19H17F3N4O2
8-(1-Methylpyrazol-4-yl)-6-[4-(trifluoromethoxy)phenyl]-1,2,3,4-tetrahydro-1,6-naphthyridin-5-one
—— 4-Pyridazinecarboxamide, 3-amino-5-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-methyl- 1540337-80-1 C14H14N4O3
4-Pyridazinecarboxamide, 3-amino-5-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-methyl-
—— 4-cyclohex-1-enylethynyl-benzaldehyde 1098336-48-1 C15H14O
4-cyclohex-1-enylethynyl-benzaldehyde