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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-cyclopropyl-2-methyl-4-{6-phenoxy-8-[(3,3,3-trifluoropropyl)amino]imidazo[1,2-a]pyrazin-3-yl}benzamide 1383120-08-8 C26H24F3N5O2
N-cyclopropyl-2-methyl-4-{6-phenoxy-8-[(3,3,3-trifluoropropyl)amino]imidazo[1,2-a]pyrazin-3-yl}benzamide
—— N-((1R,3S)-3-((2-(5-chloro-1H-pyrazolo[3,4-b]pyridin-3-yl)-5-fluoropyrimidin-4-yl)amino)cyclohexyl)pyrrolidine-1-carboxamide 1383446-97-6 C21H24ClFN8O
N-((1R,3S)-3-((2-(5-chloro-1H-pyrazolo[3,4-b]pyridin-3-yl)-5-fluoropyrimidin-4-yl)amino)cyclohexyl)pyrrolidine-1-carboxamide
—— 4-chloro-3-[3,3,3-trifluoro-2-hydroxy-1-methyl-2-(6-methyl-pyrazin-2-yl)-propyl]-benzoic acid methyl ester 1134914-86-5 C17H16ClF3N2O3
4-chloro-3-[3,3,3-trifluoro-2-hydroxy-1-methyl-2-(6-methyl-pyrazin-2-yl)-propyl]-benzoic acid methyl ester
—— N-(4-(2-fluoropyridin-4-yl)benzyl)-7-phenylquinazolin-4-amine 1384181-57-0 C26H19FN4
N-(4-(2-fluoropyridin-4-yl)benzyl)-7-phenylquinazolin-4-amine
—— ((1R,6S)-8-(6-fluoroquinoxalin-2-yl)-3,8-diazabicyclo[4.2.0]octan-3-yl)(5-methyl-2-(1H-pyrazol-1-yl)phenyl)methanone 1384065-96-6 C25H23FN6O
((1R,6S)-8-(6-fluoroquinoxalin-2-yl)-3,8-diazabicyclo[4.2.0]octan-3-yl)(5-methyl-2-(1H-pyrazol-1-yl)phenyl)methanone
—— —— 1169704-21-5 C12H25NO3S
—— —— 1033701-64-2 C33H34F2N4O7S
—— N-(5-(4-bromo-benzoyl)-4-dimethylamino-thiazol-2-yl)-2-chlorobenzamide 1264379-18-1 C19H15BrClN3O2S
N-(5-(4-bromo-benzoyl)-4-dimethylamino-thiazol-2-yl)-2-chlorobenzamide
—— (4-chlorophenyl)(cyclopentenylmethyl)sulfane 1384172-78-4 C12H13ClS
(4-chlorophenyl)(cyclopentenylmethyl)sulfane
—— CpTaCl2(ArCCAr) 103148-33-0 C21H19Cl2O2Ta
CpTaCl2(ArCCAr)
—— (2R,3R,5R)-dimethyl 5-(benzamido-9H-purin-9-yl)-1,4-dioxane-2,3-dicarboxylate 1094674-83-5 C20H19N5O7
(2R,3R,5R)-dimethyl 5-(benzamido-9H-purin-9-yl)-1,4-dioxane-2,3-dicarboxylate
—— 4-Chloro-5-methyl-3-(3-quinuclidinyloxy)isoxazole hydrochloride 138731-21-2 C11H15ClN2O2*ClH
4-Chloro-5-methyl-3-(3-quinuclidinyloxy)isoxazole hydrochloride
—— 2'-Nitro-1-(2-(pyridin-2-yl)ethyl)-spiro(piperidine-4,6'-(6'H)thieno[2,3-b]thiopyran)-4'(5'H)-one 136074-37-8 C18H19N3O3S2
2'-Nitro-1-(2-(pyridin-2-yl)ethyl)-spiro(piperidine-4,6'-(6'H)thieno[2,3-b]thiopyran)-4'(5'H)-one
—— 5-(3-chloro-4-((6-((1-(3-isopropyl-1,2,4-oxadiazol-5-yl)piperidin-4-yl)oxy)-5-methylpyrimidin-4-yl)oxy)benzyl)-1,3,2-dioxathiane 2,2-dioxide 1258604-01-1 C25H30ClN5O7S
5-(3-chloro-4-((6-((1-(3-isopropyl-1,2,4-oxadiazol-5-yl)piperidin-4-yl)oxy)-5-methylpyrimidin-4-yl)oxy)benzyl)-1,3,2-dioxathiane 2,2-dioxide
—— 7-chloro-2-[4-(2-hydroxyethoxy)-3,5-dimethylphenyl]quinazolin-4(3H)-one 1253732-63-6 C18H17ClN2O3
7-chloro-2-[4-(2-hydroxyethoxy)-3,5-dimethylphenyl]quinazolin-4(3H)-one
—— N-(1-(7-(9-((2,4-difluoro-phenyl)sulfonyl)-3,9-diazaspiro[5.5]undecane-3-carbonyl)-1H-benzoimidazol-2-yl)-ethyl)-4-methoxy-N,2,6-trimethyl-benzenesulfonic acid amide 1258069-99-6 C35H41F2N5O6S2
N-(1-(7-(9-((2,4-difluoro-phenyl)sulfonyl)-3,9-diazaspiro[5.5]undecane-3-carbonyl)-1H-benzoimidazol-2-yl)-ethyl)-4-methoxy-N,2,6-trimethyl-benzenesulfonic acid amide
—— Example 47 in WO2010147792 1259019-92-5 C18H32N4O5S
Example 47 in WO2010147792
—— N-(2-(5-fluoro-2-(1-methyl-1H-pyrazol-3-ylamino)pyrimidin-4-ylamino)-5-methoxyphenyl)methanesulfonamide 1258943-78-0 C16H18FN7O3S
N-(2-(5-fluoro-2-(1-methyl-1H-pyrazol-3-ylamino)pyrimidin-4-ylamino)-5-methoxyphenyl)methanesulfonamide
—— 2-[3-({1-[2-(dimethylamino)ethyl]-4-methyl-1H-indol-3-yl}methyl)imidazo[1,2-a]pyridin-2-yl]-1-naphthoic acid 1258872-81-9 C32H30N4O2
2-[3-({1-[2-(dimethylamino)ethyl]-4-methyl-1H-indol-3-yl}methyl)imidazo[1,2-a]pyridin-2-yl]-1-naphthoic acid
—— 6-(4-methoxycarbonylpiperidin-1-ylsulfonyl)isoquinoline 1258833-73-6 C16H18N2O4S
6-(4-methoxycarbonylpiperidin-1-ylsulfonyl)isoquinoline
—— N-methyl-1-{4-[4-(5-methyl-1H-indazol-3-yl)-1H-1,2,3-triazol-1-yl]phenyl}methanamine 1383702-23-5 C18H18N6
N-methyl-1-{4-[4-(5-methyl-1H-indazol-3-yl)-1H-1,2,3-triazol-1-yl]phenyl}methanamine
—— 2-amino-N-cyclopropylmethyl-N'-m-hydroxybenzylmorphinan 1372134-50-3 C27H34N2O
2-amino-N-cyclopropylmethyl-N'-m-hydroxybenzylmorphinan
—— (1-((2,4-dichlorophenyl)amino)-5-methylisoquinolin-4-yl)(piperidin-1-yl)methanone 1384249-20-0 C22H21Cl2N3O
(1-((2,4-dichlorophenyl)amino)-5-methylisoquinolin-4-yl)(piperidin-1-yl)methanone
—— 4-chloro-2',4'-dihydroxy-3'-methylchalcone 1355027-37-0 C16H13ClO3
4-chloro-2',4'-dihydroxy-3'-methylchalcone
—— {3-[2-(4-chloro-benzylamino)-pyrimidin-4-yl]-1H-pyrazolo[3,4-d]pyrimidin-6-yl}-(2-morpholin-4-yl-ethyl)-amine hydrochloride 1386398-43-1 C22H24ClN9O*ClH
{3-[2-(4-chloro-benzylamino)-pyrimidin-4-yl]-1H-pyrazolo[3,4-d]pyrimidin-6-yl}-(2-morpholin-4-yl-ethyl)-amine hydrochloride
—— ingenol 3-(N-ethyl-carbamate) 1383549-11-8 C23H33NO6
ingenol 3-(N-ethyl-carbamate)
—— 2-(2-aminomethyl-5-chloro-phenylamino)-ethanol 1067658-48-3 C9H13ClN2O
2-(2-aminomethyl-5-chloro-phenylamino)-ethanol
—— (1R,4R,6R)-3-{[6-methyl-3-(2-pyrimidinyl)-2-pyridinyl]carbonyl}-4-{2-[6-methyl-4-(trifluoromethyl)-3-pyridazinyl]ethyl}-3-azabicyclo[4.1.0]heptane 1384261-56-6 C25H25F3N6O
(1R,4R,6R)-3-{[6-methyl-3-(2-pyrimidinyl)-2-pyridinyl]carbonyl}-4-{2-[6-methyl-4-(trifluoromethyl)-3-pyridazinyl]ethyl}-3-azabicyclo[4.1.0]heptane
—— methyl (3S)-3-(1,3-benzodioxol-5-yl)-3-[({(2R)-1-[bis(thiophen-2-ylmethyl)amino]-1-oxohexan-2-yl}carbamoyl)amino]propanoate 1378535-48-8 C28H33N3O6S2
methyl (3S)-3-(1,3-benzodioxol-5-yl)-3-[({(2R)-1-[bis(thiophen-2-ylmethyl)amino]-1-oxohexan-2-yl}carbamoyl)amino]propanoate
—— 3-isopropyl-5-(1-(7-(4-methanesulfonylphenyl)thieno[3,2-d]pyrimidin-4-yl)piperidin-4-yl)-1,2,4-oxadiazole 1384950-48-4 C23H25N5O3S2
3-isopropyl-5-(1-(7-(4-methanesulfonylphenyl)thieno[3,2-d]pyrimidin-4-yl)piperidin-4-yl)-1,2,4-oxadiazole
—— 2-(2,4-diaminophenyl)ethyl (2E)-3-(4-{difluoro[4-(3-fluoropropoxy)phenyl]-methoxy}phenyl)prop-2-enoate 1345472-67-4 C27H27F3N2O4
2-(2,4-diaminophenyl)ethyl (2E)-3-(4-{difluoro[4-(3-fluoropropoxy)phenyl]-methoxy}phenyl)prop-2-enoate
—— 4-methoxy-N-[4-(trifluoromethoxy)phenyl]quinolin-7-amine 1258454-45-3 C17H13F3N2O2
4-methoxy-N-[4-(trifluoromethoxy)phenyl]quinolin-7-amine
—— 5-(3-chloro-phenyl)-oxazole-4-carboxylic acid {2-[4-(1,1-difluoro-ethyl)-thiazol-2-ylmethyl]-2H-[1,2,3]triazol-4-yl}-amide 1258417-17-2 C18H13ClF2N6O2S
5-(3-chloro-phenyl)-oxazole-4-carboxylic acid {2-[4-(1,1-difluoro-ethyl)-thiazol-2-ylmethyl]-2H-[1,2,3]triazol-4-yl}-amide
—— 1-{(4-benzyl-4H-1,2,4-triazol-3-yl)[4-(1H-pyrazol-1-yl)phenyl]methyl}-4-cyclobutylpiperazine 1256487-66-7 C27H31N7
1-{(4-benzyl-4H-1,2,4-triazol-3-yl)[4-(1H-pyrazol-1-yl)phenyl]methyl}-4-cyclobutylpiperazine
—— N-(5-methyl-pyrazin-2-ylmethyl)-3-(5-methyl-pyridin-2-yl)-5-(5-oxo-6-oxa-4-aza-spiro[2.4]hept-4-yl)-benzamide 1258950-34-3 C24H23N5O3
N-(5-methyl-pyrazin-2-ylmethyl)-3-(5-methyl-pyridin-2-yl)-5-(5-oxo-6-oxa-4-aza-spiro[2.4]hept-4-yl)-benzamide
—— 6-methyl-2'-(4-(4-methylbenzamido)phenyl)-[2,6'-bibenzo[d]thiazole]-7-sullfonic acid ammonium salt 1403245-68-0 C29H21N3O4S3*H3N
6-methyl-2'-(4-(4-methylbenzamido)phenyl)-[2,6'-bibenzo[d]thiazole]-7-sullfonic acid ammonium salt
—— (2S,3S,5S,6S)-3-(tert-butyldiphenylsilanyloxymethyl)-5,6-dihydroxy-2-hydroxymethylcyclohexanone 1256355-93-7 C24H32O5Si
(2S,3S,5S,6S)-3-(tert-butyldiphenylsilanyloxymethyl)-5,6-dihydroxy-2-hydroxymethylcyclohexanone
—— (1R)-(2-(4-acetylaminomethyl-phenyl)-acetylamino)-(3-carboxy-2-hydroxy)benzyl-methylboronic acid 1256335-95-1 C20H23BN2O7
(1R)-(2-(4-acetylaminomethyl-phenyl)-acetylamino)-(3-carboxy-2-hydroxy)benzyl-methylboronic acid
—— 4-[(5-chloropyridin-2-yl)methoxy]-1-[6-[2-[[(2S)-oxolan-2-yl]methylamino]ethylamino]pyridin-3-yl]pyridin-2-one 1257515-59-5 C23H26ClN5O3
4-[(5-chloropyridin-2-yl)methoxy]-1-[6-[2-[[(2S)-oxolan-2-yl]methylamino]ethylamino]pyridin-3-yl]pyridin-2-one
—— 4-(4-cyanophenyl)(isoxazole-2,5-dicarbonyl)bispiperidine 1253696-75-1 C22H24N4O3
4-(4-cyanophenyl)(isoxazole-2,5-dicarbonyl)bispiperidine
—— 4-[5-Bromo-1-(4-bromobenzyl)-2-methyl-1H-indol-3-yl]-3,3-dimethylbutanoic acid 185737-39-7 C22H23Br2NO2
4-[5-Bromo-1-(4-bromobenzyl)-2-methyl-1H-indol-3-yl]-3,3-dimethylbutanoic acid
—— 3-(4-(1-((2-(trimethylsilyl)ethoxy)methyl)-1H-imidazol-2-yl)phenyl)pyrazolo[1,5-a]pyrimidin-5-ol 1269646-27-6 C21H25N5O2Si
3-(4-(1-((2-(trimethylsilyl)ethoxy)methyl)-1H-imidazol-2-yl)phenyl)pyrazolo[1,5-a]pyrimidin-5-ol
—— 2,4-dichloro-6-trifluoromethyl-trifluoromethoxybenzene 141872-89-1 C8H2Cl2F6O
2,4-dichloro-6-trifluoromethyl-trifluoromethoxybenzene
—— Ethyl 4-cyano-4-(p-chlorophenyl)-4-phenylbutyrate 173272-48-5 C19H18ClNO2
Ethyl 4-cyano-4-(p-chlorophenyl)-4-phenylbutyrate
—— (R)-5-(7-(1-(4-fluorophenyl)ethylcarbamoyl)-3-phenylquinolin-2-yl)pentanoic acid 1396317-09-1 C29H27FN2O3
(R)-5-(7-(1-(4-fluorophenyl)ethylcarbamoyl)-3-phenylquinolin-2-yl)pentanoic acid
—— (4-((3-chloro-4-methylphenyl)amino)-8-methylnaphthalen-1-yl)(morpholino)methanone 1384250-46-7 C23H23ClN2O2
(4-((3-chloro-4-methylphenyl)amino)-8-methylnaphthalen-1-yl)(morpholino)methanone
—— N-(5-(3-fluorobenzamido)bicyclo[3.2.1]octan-1-yl)nicotinamide 1383971-84-3 C21H22FN3O2
N-(5-(3-fluorobenzamido)bicyclo[3.2.1]octan-1-yl)nicotinamide
—— N-[(1S)-1-(2-fluoro-5-methylsulfonylphenyl)butyl]-1-(4-fluorophenyl)-5-(trifluoromethyl)-6,7-dihydro-5H-pyrazolo[4,3-b]pyridine-4-carboxamide 1383734-43-7 C25H25F5N4O3S
N-[(1S)-1-(2-fluoro-5-methylsulfonylphenyl)butyl]-1-(4-fluorophenyl)-5-(trifluoromethyl)-6,7-dihydro-5H-pyrazolo[4,3-b]pyridine-4-carboxamide
—— (2S,3R)-3-bromo-2-(4-fluorophenyl)-1-(4-nitrophenylsulfonyl)pyrrolidine 1374877-74-3 C16H14BrFN2O4S
(2S,3R)-3-bromo-2-(4-fluorophenyl)-1-(4-nitrophenylsulfonyl)pyrrolidine
—— N-(5-(3-chlorobenzamido)bicyclo[3.2.1]octan-1-yl)-5-methylpicolinamide 1383971-75-2 C22H24ClN3O2
N-(5-(3-chlorobenzamido)bicyclo[3.2.1]octan-1-yl)-5-methylpicolinamide