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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2,4-dimethyl-6-oxo-1-propyl-1,6-dihydro-pyridine-3-carboxylic acid 1247803-01-5 C11H15NO3
2,4-dimethyl-6-oxo-1-propyl-1,6-dihydro-pyridine-3-carboxylic acid
—— 6-(imidazo[1,2-a]pyrazin-3-yl)-N-[(2R,3R)-2-methylpiperidin-3-yl]pyrazin-2-amine 1207851-04-4 C16H19N7
6-(imidazo[1,2-a]pyrazin-3-yl)-N-[(2R,3R)-2-methylpiperidin-3-yl]pyrazin-2-amine
—— N-[4-(2-Bromo-ethyl)-phenyl]-2,2,2-trifluoro-acetamide 1813-85-0 C10H9BrF3NO
N-[4-(2-Bromo-ethyl)-phenyl]-2,2,2-trifluoro-acetamide
—— (S)-[3-(3-t-butoxycarbonylaminopropyl)-4-[(4-guanidinobenzoylamino)acetyl]-2-oxopiperazin-1-yl]acetic acid t-butyl ester 184576-58-7 C28H43N7O7
(S)-[3-(3-t-butoxycarbonylaminopropyl)-4-[(4-guanidinobenzoylamino)acetyl]-2-oxopiperazin-1-yl]acetic acid t-butyl ester
—— 4-[4-Amino-5-(3-hydroxy-phenyl)-pyrrolo[2,3-d]pyrimidin-7-yl]-piperidine-1-carboxylic acid tert-butyl ester 197525-89-6 C22H27N5O3
4-[4-Amino-5-(3-hydroxy-phenyl)-pyrrolo[2,3-d]pyrimidin-7-yl]-piperidine-1-carboxylic acid tert-butyl ester
—— <i>N</i>-(2-chloro-1-methyl-2-phenyl-ethyl)-benzamide 131591-52-1 C16H16ClNO
<i>N</i>-(2-chloro-1-methyl-2-phenyl-ethyl)-benzamide
—— 4-[N-(3-Carboxypropyl)-N-Methylamino]-6,7,8-Trimethoxyquinazoline 165953-60-6 C16H21N3O5
4-[N-(3-Carboxypropyl)-N-Methylamino]-6,7,8-Trimethoxyquinazoline
—— methyl 3-methyl-8-phenyl-4-(trifluoromethyl)-3-azabicyclo[4.2.0]octa-1(8),5-diene-4-carboxylate 1351377-95-1 C17H16F3NO2
methyl 3-methyl-8-phenyl-4-(trifluoromethyl)-3-azabicyclo[4.2.0]octa-1(8),5-diene-4-carboxylate
—— 3-Bromo-8-(2,6-dichlorobenzoylamino)-4-(4-methylpiperazin-1-yl)quinoline 190129-31-8 C21H19BrCl2N4O
3-Bromo-8-(2,6-dichlorobenzoylamino)-4-(4-methylpiperazin-1-yl)quinoline
—— methyl N-[(1S)-2-[(2S)-2-[5-[4-[2-[4-[(2S)-1-[(2S)-2-(methoxycarbonylamino)-3-methylbutanoyl]pyrrolidin-2-yl]-3,5-diazatricyclo[8.4.0.02,6]tetradeca-1(10),2(6),3,11,13-pentaen-12-yl]ethynyl]phenyl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-1-(oxan-4-yl)-2-oxoethyl]carbamate 1228968-20-4 C47H56N8O7
methyl N-[(1S)-2-[(2S)-2-[5-[4-[2-[4-[(2S)-1-[(2S)-2-(methoxycarbonylamino)-3-methylbutanoyl]pyrrolidin-2-yl]-3,5-diazatricyclo[8.4.0.02,6]tetradeca-1(10),2(6),3,11,13-pentaen-12-yl]ethynyl]phenyl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-1-(oxan-4-yl)-2-oxoethyl]carbamate
—— (S)-4-((1-(2-chloro-3-fluorophenyl)-2-(methylamino)ethyl)amino)-2-methylquinazoline-8-carboxamide 1357079-81-2 C19H19ClFN5O
(S)-4-((1-(2-chloro-3-fluorophenyl)-2-(methylamino)ethyl)amino)-2-methylquinazoline-8-carboxamide
—— 6-bromo-N-[6,7-dimethoxy-5-(4-phenylphenyl)naphthalen-1-yl]-2,3-dimethoxy-N-methylbenzamide 1235871-50-7 C34H30BrNO5
6-bromo-N-[6,7-dimethoxy-5-(4-phenylphenyl)naphthalen-1-yl]-2,3-dimethoxy-N-methylbenzamide
—— (R)-7-(4-chloro-2-fluorophenyl)-10-(2-(4-methylpiperazin-1-yl)-2-oxyethyl)-2-((S)-1-piperidin-4-ylpyrrolidine-2-carbonyl)-1,3,4,11a-tetrahydro-2H,10H-2,4a,10-triazadibenzo[a,d]cycloheptene-5,11-dione 1262131-13-4 C35H43ClFN7O4
(R)-7-(4-chloro-2-fluorophenyl)-10-(2-(4-methylpiperazin-1-yl)-2-oxyethyl)-2-((S)-1-piperidin-4-ylpyrrolidine-2-carbonyl)-1,3,4,11a-tetrahydro-2H,10H-2,4a,10-triazadibenzo[a,d]cycloheptene-5,11-dione
—— (-)-(3R)-1-(2,3-dimethylbenzyl)-N-(9-chloro-2,3,4,5-tetrahydro-1-benzoxepin-7-ylmethyl)-N-isobutylpiperidine-3-carboxamide 1233926-67-4 C30H41ClN2O2
(-)-(3R)-1-(2,3-dimethylbenzyl)-N-(9-chloro-2,3,4,5-tetrahydro-1-benzoxepin-7-ylmethyl)-N-isobutylpiperidine-3-carboxamide
—— O-Benzoyl-O'-(3-chlor-benzoyl-dihydroxy-phenylmethan 1460-60-2 C21H15ClO4
O-Benzoyl-O'-(3-chlor-benzoyl-dihydroxy-phenylmethan
—— 3-(3-Indolyl)methyl-6-methoxy-4-chromanone 124049-47-4 C19H17NO3
3-(3-Indolyl)methyl-6-methoxy-4-chromanone
—— (S)-(1-benzylpyrrolidin-2-yl)bis(4-chlorophenyl)methanol 1609954-52-0 C24H23Cl2NO
(S)-(1-benzylpyrrolidin-2-yl)bis(4-chlorophenyl)methanol
—— 2-(4-Carboxypiperidino)-4-Diethylamino-6,7,8-Trimethoxyquinazoline 165953-86-6 C21H30N4O5
2-(4-Carboxypiperidino)-4-Diethylamino-6,7,8-Trimethoxyquinazoline
—— 2-((E)-3-(2-bromo-4,5-dimethoxyphenyl)-3-hydroxyprop-1-enyl)benzaldehyde 1370701-17-9 C18H17BrO4
2-((E)-3-(2-bromo-4,5-dimethoxyphenyl)-3-hydroxyprop-1-enyl)benzaldehyde
—— methyl (2R)-2-amino-2-[(2R,3R,4R,5S,6R)-2-(5-methyl-2,4-dioxopyrimidin-1-yl)-4,5-bis(phenylmethoxy)-6-(phenylmethoxymethyl)oxan-3-yl]acetate 1151746-94-9 C35H39N3O8
methyl (2R)-2-amino-2-[(2R,3R,4R,5S,6R)-2-(5-methyl-2,4-dioxopyrimidin-1-yl)-4,5-bis(phenylmethoxy)-6-(phenylmethoxymethyl)oxan-3-yl]acetate
—— 5,5-Bis((2-chloro-4-pyridinyl)methyl)-5H-indeno-[1,2-b]pyridine 160588-67-0 C24H17Cl2N3
5,5-Bis((2-chloro-4-pyridinyl)methyl)-5H-indeno-[1,2-b]pyridine
—— 2-O-ethyl 3-O,4-O-dimethyl (2R,3R,4R,5S)-5-(4-cyanophenyl)pyrrolidine-2,3,4-tricarboxylate 1179815-76-9 C18H20N2O6
2-O-ethyl 3-O,4-O-dimethyl (2R,3R,4R,5S)-5-(4-cyanophenyl)pyrrolidine-2,3,4-tricarboxylate
—— 10-methoxy-2-methyl-benzo[c]phenanthrene 1243027-66-8 C20H16O
10-methoxy-2-methyl-benzo[c]phenanthrene
—— N-[6-(4-Chlorophenyl)hexyl]-4-(4-methoxyphenylsulfonyl)-2-oxoazetidin-1-ylacetamide 180203-68-3 C24H29ClN2O5S
N-[6-(4-Chlorophenyl)hexyl]-4-(4-methoxyphenylsulfonyl)-2-oxoazetidin-1-ylacetamide
—— dimethyl 1-benzyl-4-methyl-4H-pyridine-2,3-dicarboxylate 1314023-00-1 C17H19NO4
dimethyl 1-benzyl-4-methyl-4H-pyridine-2,3-dicarboxylate
—— tert-butyl [(2R)-1-[(3-amino-2-oxo-1,2-dihydropyridin-4-yl)sulfanyl]-3-{[tert-butyl(diphenyl)silyl]oxy}propan-2-yl]carbamate 1374041-23-2 C29H39N3O4SSi
tert-butyl [(2R)-1-[(3-amino-2-oxo-1,2-dihydropyridin-4-yl)sulfanyl]-3-{[tert-butyl(diphenyl)silyl]oxy}propan-2-yl]carbamate
—— 2-[4-[3-[2-(4-Bromophenyl)-3-methylbutan-2-yl]-1,2,4-oxadiazol-5-yl]piperazin-1-yl]ethanol 1360552-91-5 C19H27BrN4O2
2-[4-[3-[2-(4-Bromophenyl)-3-methylbutan-2-yl]-1,2,4-oxadiazol-5-yl]piperazin-1-yl]ethanol
—— 5-(1,4-Dioxan-2-ylmethylamino)-6-ethyl-3-(3-methylsulfonylanilino)pyrazine-2-carboxamide 1254050-14-0 C19H25N5O5S
5-(1,4-Dioxan-2-ylmethylamino)-6-ethyl-3-(3-methylsulfonylanilino)pyrazine-2-carboxamide
—— 2-amino-2-((5-(4-(3-(1-adamantyl)-3-methoxyphenyl)-1,2,4-oxadiazol-3-yl)indolin-1-yl)methyl)propane-1,3-diol 1221258-41-8 C31H38N4O4
2-amino-2-((5-(4-(3-(1-adamantyl)-3-methoxyphenyl)-1,2,4-oxadiazol-3-yl)indolin-1-yl)methyl)propane-1,3-diol
—— 6-bromo-N-(6,7-dimethoxy-5-phenylnaphthalen-1-yl)-3-methoxy-N-methyl-2-propan-2-yloxybenzamide 1235871-55-2 C30H30BrNO5
6-bromo-N-(6,7-dimethoxy-5-phenylnaphthalen-1-yl)-3-methoxy-N-methyl-2-propan-2-yloxybenzamide
—— N-[4-chloro-2-methyl-6-(propan-2-ylcarbamoyl)phenyl]-2-(3-chloropyridin-2-yl)-5-[[[3-(trifluoromethyl)phenyl]sulfonylamino]methyl]pyrazole-3-carboxamide 1352400-35-1 C28H25Cl2F3N6O4S
N-[4-chloro-2-methyl-6-(propan-2-ylcarbamoyl)phenyl]-2-(3-chloropyridin-2-yl)-5-[[[3-(trifluoromethyl)phenyl]sulfonylamino]methyl]pyrazole-3-carboxamide
—— US8653087, III-403 1213246-90-2 C28H28F4N8O2
US8653087, III-403
—— N-[(1R)-1-[3-[(2S)-but-3-yn-2-yl]oxyphenyl]ethyl]-3-(methoxymethoxy)propane-1-sulfonamide 1198224-70-2 C17H25NO5S
N-[(1R)-1-[3-[(2S)-but-3-yn-2-yl]oxyphenyl]ethyl]-3-(methoxymethoxy)propane-1-sulfonamide
—— 8-(2,6-dichlorobenzoylamino)-4-ethoxy-3-ethoxycarbonylquinoline 190128-46-2 C21H18Cl2N2O4
8-(2,6-dichlorobenzoylamino)-4-ethoxy-3-ethoxycarbonylquinoline
—— 2-(Furan-2-ylmethyl)-3,3-bis(prop-2-enyl)pyrrolo[3,4-b]quinolin-1-one 1207374-34-2 C22H20N2O2
2-(Furan-2-ylmethyl)-3,3-bis(prop-2-enyl)pyrrolo[3,4-b]quinolin-1-one
—— (2R,3S,3aR,5aS,8aR,8bS)-methyl-3-propyl-1,2,3,3a,5a,6,7,8,8a,8b-decahydro-as-indacene-2-carboxylate 1021177-73-0 C17H26O2
(2R,3S,3aR,5aS,8aR,8bS)-methyl-3-propyl-1,2,3,3a,5a,6,7,8,8a,8b-decahydro-as-indacene-2-carboxylate
—— ((3-fluoro-2-methylpropoxy)methanetriyl)-tribenzene 1082738-96-2 C23H23FO
((3-fluoro-2-methylpropoxy)methanetriyl)-tribenzene
—— methyl (2R,3aS,4S,5S,6S)-4,5-bis(phenylmethoxy)-6-(phenylmethoxymethyl)-2,3,3a,4,5,6-hexahydropyrrolo[1,2-b][1,2]oxazole-2-carboxylate 1333128-42-9 C30H33NO6
methyl (2R,3aS,4S,5S,6S)-4,5-bis(phenylmethoxy)-6-(phenylmethoxymethyl)-2,3,3a,4,5,6-hexahydropyrrolo[1,2-b][1,2]oxazole-2-carboxylate
—— Methyl 2-[4-[4-(3-methoxy-3-oxoprop-1-ynyl)phenyl]phenyl]-3,4,5,6-tetramethylbenzoate 1303613-42-4 C28H26O4
Methyl 2-[4-[4-(3-methoxy-3-oxoprop-1-ynyl)phenyl]phenyl]-3,4,5,6-tetramethylbenzoate
—— (2R)-3-ethoxycarbonylmethyl-4-oxo-pyrrolidine-1-carboxylic acid benzyl ester 1016976-64-9 C16H19NO5
(2R)-3-ethoxycarbonylmethyl-4-oxo-pyrrolidine-1-carboxylic acid benzyl ester
—— [(2R)-3-[2-(1,3-dioxoisoindol-2-yl)oxyethoxy-hydroxyphosphoryl]oxy-2-hexadecanoyloxypropyl] hexadecanoate 1214192-12-7 C45H76NO11P
[(2R)-3-[2-(1,3-dioxoisoindol-2-yl)oxyethoxy-hydroxyphosphoryl]oxy-2-hexadecanoyloxypropyl] hexadecanoate
—— 3-bromo-8-(2,6-dichlorobenzoylamino)-4-(ethoxycarbonylmethyl)quinoline 190128-56-4 C20H15BrCl2N2O3
3-bromo-8-(2,6-dichlorobenzoylamino)-4-(ethoxycarbonylmethyl)quinoline
—— N-[4-chloro-2-methyl-6-(propan-2-ylcarbamoyl)phenyl]-2-(3-chloropyridin-2-yl)-5-[[[2-(trifluoromethyl)phenyl]methylsulfonylamino]methyl]pyrazole-3-carboxamide 1352400-37-3 C29H27Cl2F3N6O4S
N-[4-chloro-2-methyl-6-(propan-2-ylcarbamoyl)phenyl]-2-(3-chloropyridin-2-yl)-5-[[[2-(trifluoromethyl)phenyl]methylsulfonylamino]methyl]pyrazole-3-carboxamide
—— 1-(4-chlorophenyl)-5-methyl-N-[(1S)-1-(2-methylsulfonylpyridin-4-yl)butyl]-6,7-dihydro-5H-pyrazolo[4,3-b]pyridine-4-carboxamide 1383734-58-4 C24H28ClN5O3S
1-(4-chlorophenyl)-5-methyl-N-[(1S)-1-(2-methylsulfonylpyridin-4-yl)butyl]-6,7-dihydro-5H-pyrazolo[4,3-b]pyridine-4-carboxamide
—— {(1R,5S)-5-[(pyrazine-2-carbonyl)-amino]-bicyclo[3.2.1]oct-1-yl}-carbamic acid tert-butyl ester 1383973-66-7 C18H26N4O3
{(1R,5S)-5-[(pyrazine-2-carbonyl)-amino]-bicyclo[3.2.1]oct-1-yl}-carbamic acid tert-butyl ester
—— N-[(1R)-2-[(2S)-2-[5-[4-[2-[4-[2-[(2S)-1-[(2R)-2-acetamido-2-phenylacetyl]pyrrolidin-2-yl]-1H-imidazol-5-yl]phenyl]ethynyl]phenyl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-2-oxo-1-phenylethyl]acetamide 1228964-87-1 C48H46N8O4
N-[(1R)-2-[(2S)-2-[5-[4-[2-[4-[2-[(2S)-1-[(2R)-2-acetamido-2-phenylacetyl]pyrrolidin-2-yl]-1H-imidazol-5-yl]phenyl]ethynyl]phenyl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-2-oxo-1-phenylethyl]acetamide
—— 1-(3-{1-[4-(2-amino-pyrimidin-5-yl)-phenyl]-1,2-dimethyl-propyl}-[1,2,4]oxadiazol-5-yl)-4-methyl-piperidin-4-ol 1360551-04-7 C23H30N6O2
1-(3-{1-[4-(2-amino-pyrimidin-5-yl)-phenyl]-1,2-dimethyl-propyl}-[1,2,4]oxadiazol-5-yl)-4-methyl-piperidin-4-ol
—— 6-(benzofuran-2-yl)-4-(4-methoxyphenyl)-3,4-dihydropyrimidin-2(1H)-one 1244782-02-2 C19H16N2O3
6-(benzofuran-2-yl)-4-(4-methoxyphenyl)-3,4-dihydropyrimidin-2(1H)-one
—— 2-phenylfuro[3,2-c]quinoline 5-oxide 1449680-37-8 C17H11NO2
2-phenylfuro[3,2-c]quinoline 5-oxide
—— 4-(((3-(2,4-dimethoxyphenyl)-isoxazol-5-yl))methylamino)quinazoline 1459184-37-2 C20H18N4O3
4-(((3-(2,4-dimethoxyphenyl)-isoxazol-5-yl))methylamino)quinazoline