| 中文名称 | 英文名称 | CAS号 | 化学式 |
|---|---|---|---|
| —— | N-methyl-5-[[(1S,9S)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-diene-11-carbonyl]amino]thiadiazole-4-carboxamide | —— | C16H18N6O3S |
| —— | N-methyl-5-[[(1R,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-diene-11-carbonyl]amino]thiadiazole-4-carboxamide | —— | C16H18N6O3S |
| —— | (1S,9R)-11-[2-[3-tert-butyl-5-(trifluoromethyl)pyrazol-1-yl]-1,3-thiazole-4-carbonyl]-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one | —— | C23H24F3N5O2S |
| —— | 6-[(1R,9S)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-diene-11-carbonyl]-1H-pyrimidine-2,4-dione | —— | C16H16N4O4 |
| —— | (1S,9S)-6-oxo-N-[4-(piperidine-1-carbonyl)thiadiazol-5-yl]-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-diene-11-carboxamide | —— | C20H24N6O3S |
| —— | N-[(4-methoxyphenyl)methyl]-5-[[(1R,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-diene-11-carbonyl]amino]thiadiazole-4-carboxamide | —— | C23H24N6O4S |
| —— | N-[(4-methoxyphenyl)methyl]-5-[[(1S,9S)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-diene-11-carbonyl]amino]thiadiazole-4-carboxamide | —— | C23H24N6O4S |
| —— | N-[2-(1H-indol-3-yl)ethyl]-5-[[(1S,9S)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-diene-11-carbonyl]amino]thiadiazole-4-carboxamide | —— | C25H25N7O3S |
| —— | N-cyclohexyl-5-[[(1S,9S)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-diene-11-carbonyl]amino]thiadiazole-4-carboxamide | —— | C21H26N6O3S |
| —— | 4-chloro-N-[2-oxo-2-[(1R,9S)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]ethyl]benzenesulfonamide | —— | C19H20ClN3O4S |
| —— | 2-[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]-N-[4-(trifluoromethyl)phenyl]acetamide | —— | C20H20F3N3O2 |
| —— | (1R,9R)-N-[4-(4-benzylpiperidine-1-carbonyl)thiadiazol-5-yl]-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-diene-11-carboxamide | —— | C27H30N6O3S |
| —— | (1S,9R)-11-(2-oxopropyl)-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one | —— | C14H18N2O2 |
| —— | (1R,9R)-N-[4-(morpholine-4-carbonyl)thiadiazol-5-yl]-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-diene-11-carboxamide | —— | C19H22N6O4S |
| —— | (1S,9S)-N-[4-(morpholine-4-carbonyl)thiadiazol-5-yl]-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-diene-11-carboxamide | —— | C19H22N6O4S |
| —— | (1R,9S)-11-[2-[3-methyl-5-(trifluoromethyl)pyrazol-1-yl]-1,3-thiazole-4-carbonyl]-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one | —— | C20H18F3N5O2S |
| —— | 4-chloro-N-[2-oxo-2-[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]ethyl]benzenesulfonamide | —— | C19H20ClN3O4S |
| —— | 2,2,2-trifluoro-N-[5-[(1S,9S)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]-1,3,4-thiadiazol-2-yl]acetamide | —— | C15H14F3N5O2S |
| —— | N-[(4-fluorophenyl)methyl]-2-[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]acetamide | —— | C20H22FN3O2 |
| —— | N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]-2-[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]acetamide | —— | C23H24N4O3S |
| —— | N-[5-[(1S,9S)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]-1,3,4-thiadiazol-2-yl]formamide | —— | C14H15N5O2S |
| —— | (1R,9S)-11-[1-(2,1,3-benzothiadiazol-4-ylsulfonyl)piperidine-4-carbonyl]-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one | —— | C23H25N5O4S2 |
| —— | (1S,9R)-11-[1-(2,1,3-benzothiadiazol-4-ylsulfonyl)piperidine-4-carbonyl]-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one | —— | C23H25N5O4S2 |
| —— | N-[1-(2,3,4,6,7,8,9,9a-octahydro-1H-quinolizin-1-ylmethoxy)-2,2,2-trichloroethyl]-4-nitrobenzamide | —— | C19H24Cl3N3O4 |
| —— | 4-(6-Oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl)-1-pyrrolidin-1-ylbutane-1,3-dione | —— | C19H25N3O3 |
| —— | 11-(2,2-Diphenylethyl)-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one | —— | C25H26N2O |
| —— | 4-chloro-N-[(E)-1-(5-methylfuran-2-yl)-3-oxo-3-[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]prop-1-en-2-yl]benzamide | —— | C26H24ClN3O4 |
| —— | 3-[[2-(2-chloro-6-fluorophenyl)acetyl]amino]-N-(furan-2-ylmethyl)-4-[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]benzamide | —— | C31H28ClFN4O4 |
| —— | 2-(2-chloro-6-fluorophenyl)-N-[2-[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]-5-(pyrrolidine-1-carbonyl)phenyl]acetamide | —— | C30H30ClFN4O3 |
| —— | N-(2-benzylsulfanylethyl)-3-[(4-bromophenyl)sulfonylamino]-4-[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]benzamide | —— | C33H33BrN4O4S2 |
| —— | N-(2-benzylsulfanylethyl)-3-[[2-(2-chloro-6-fluorophenyl)acetyl]amino]-4-[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]benzamide | —— | C35H34ClFN4O3S |
| —— | N-[(E)-1-(furan-2-yl)-3-oxo-3-[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]prop-1-en-2-yl]-4-methylbenzamide | —— | C26H25N3O4 |
| —— | 4-fluoro-N-[(E)-3-oxo-3-[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]-1-(4-phenylmethoxyphenyl)prop-1-en-2-yl]benzamide | —— | C34H30FN3O4 |
| —— | 4-bromo-N-[5-[4-(3-chlorophenyl)piperazine-1-carbonyl]-2-[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]phenyl]benzenesulfonamide | —— | C34H33BrClN5O4S |
| —— | N-[(E)-1-(4-bromothiophen-2-yl)-3-oxo-3-[(1R,9S)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]prop-1-en-2-yl]-4-chloro-3-nitrobenzamide | —— | C25H20BrClN4O5S |
| —— | 3-[(2,4-dichlorophenyl)carbamothioylamino]-N-(furan-2-ylmethyl)-4-[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]benzamide | —— | C30H27Cl2N5O3S |
| —— | 3-[[2-(2-chloro-6-fluorophenyl)acetyl]amino]-N-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]benzamide | —— | C34H30ClFN4O5 |
| —— | N-[5-[4-(2-chlorophenyl)piperazine-1-carbonyl]-2-[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]phenyl]-3-morpholin-4-ylpropanamide | —— | C35H41ClN6O4 |
| —— | 4-tert-butyl-N-[(E)-1-(3-chlorophenyl)-3-oxo-3-[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]prop-1-en-2-yl]benzamide | —— | C31H32ClN3O3 |
| —— | 2-(2-chloro-6-fluorophenyl)-N-[5-[4-(2-chlorophenyl)piperazine-1-carbonyl]-2-[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]phenyl]acetamide | —— | C36H34Cl2FN5O3 |
| —— | N-[(Z)-1-(2-fluorophenyl)-3-oxo-3-[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]prop-1-en-2-yl]-4-methoxy-3-nitrobenzamide | —— | C28H25FN4O6 |
| —— | 4-methoxy-N-[(Z)-1-(5-methylfuran-2-yl)-3-oxo-3-[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]prop-1-en-2-yl]-3-nitrobenzamide | —— | C27H26N4O7 |
| —— | N-[(E)-1-(4-bromothiophen-2-yl)-3-oxo-3-[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]prop-1-en-2-yl]-4-methoxybenzamide | —— | C26H24BrN3O4S |
| —— | N-[(E)-1-(4-bromothiophen-2-yl)-3-oxo-3-[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]prop-1-en-2-yl]-4-chloro-3-nitrobenzamide | —— | C25H20BrClN4O5S |
| —— | N-[2-[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]-5-(4-pyridin-2-ylpiperazine-1-carbonyl)phenyl]-2,3-dihydro-1,4-benzodioxine-6-sulfonamide | —— | C35H36N6O6S |
| —— | N-[2-(cyclohexen-1-yl)ethyl]-3-[(2,4-dichlorophenyl)carbamothioylamino]-4-[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]benzamide | —— | C33H35Cl2N5O2S |
| —— | 3-[[(4-bromoanilino)-[(2-chlorophenyl)methylsulfanyl]methylidene]amino]-4-[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]benzoic acid | —— | C32H28BrClN4O3S |
| —— | 4-fluoro-N-[2-[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]-5-(4-pyridin-2-ylpiperazine-1-carbonyl)phenyl]benzenesulfonamide | —— | C33H33FN6O4S |
| —— | N-[1-(6-chloro-4-oxochromen-3-yl)-3-oxo-3-(6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl)prop-1-en-2-yl]-2-methylbenzamide | —— | C31H26ClN3O5 |
| —— | N-[2-(cyclohexen-1-yl)ethyl]-3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfonylamino)-4-[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]benzamide | —— | C34H38N4O6S |