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噻吩并嘧啶酮衍生物

中文名称 英文名称 CAS号 化学式 结构式图片
—— (2R)-N-[(2R)-2-cyano-3-methylbutan-2-yl]-2-[(12-oxo-11-pentyl-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9-trien-10-yl)sulfanyl]propanamide —— C23H32N4O2S2
(2R)-N-[(2R)-2-cyano-3-methylbutan-2-yl]-2-[(12-oxo-11-pentyl-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9-trien-10-yl)sulfanyl]propanamide
—— (2R)-N-[(2S)-2-cyano-3-methylbutan-2-yl]-2-[(12-oxo-11-pentyl-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9-trien-10-yl)sulfanyl]propanamide —— C23H32N4O2S2
(2R)-N-[(2S)-2-cyano-3-methylbutan-2-yl]-2-[(12-oxo-11-pentyl-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9-trien-10-yl)sulfanyl]propanamide
—— (2S)-N-[(2S)-2-cyano-3-methylbutan-2-yl]-2-[(12-oxo-11-pentyl-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9-trien-10-yl)sulfanyl]propanamide —— C23H32N4O2S2
(2S)-N-[(2S)-2-cyano-3-methylbutan-2-yl]-2-[(12-oxo-11-pentyl-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9-trien-10-yl)sulfanyl]propanamide
—— N-[(2S)-3-methylbutan-2-yl]-2-[[11-(4-methylphenyl)-12-oxo-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9-trien-10-yl]sulfanyl]acetamide —— C23H27N3O2S2
N-[(2S)-3-methylbutan-2-yl]-2-[[11-(4-methylphenyl)-12-oxo-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9-trien-10-yl]sulfanyl]acetamide
—— N-[(2R)-3-methylbutan-2-yl]-2-[[11-(4-methylphenyl)-12-oxo-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9-trien-10-yl]sulfanyl]acetamide —— C23H27N3O2S2
N-[(2R)-3-methylbutan-2-yl]-2-[[11-(4-methylphenyl)-12-oxo-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9-trien-10-yl]sulfanyl]acetamide
—— 4-[(Z)-(6-methyl-4-oxo-5-phenylthieno[2,3-d]pyrimidin-3-yl)iminomethyl]benzoate —— C21H14N3O3S-
4-[(Z)-(6-methyl-4-oxo-5-phenylthieno[2,3-d]pyrimidin-3-yl)iminomethyl]benzoate
—— 5-methyl-4-(3-morpholin-4-ylpropylamino)-N-[[(1R,2R,4S)-spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-yl]methyl]thieno[2,3-d]pyrimidine-6-carboxamide —— C25H33N5O2S
5-methyl-4-(3-morpholin-4-ylpropylamino)-N-[[(1R,2R,4S)-spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-yl]methyl]thieno[2,3-d]pyrimidine-6-carboxamide
—— 5-methyl-4-(3-morpholin-4-ylpropylamino)-N-[[(1R,2S,4S)-spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-yl]methyl]thieno[2,3-d]pyrimidine-6-carboxamide —— C25H33N5O2S
5-methyl-4-(3-morpholin-4-ylpropylamino)-N-[[(1R,2S,4S)-spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-yl]methyl]thieno[2,3-d]pyrimidine-6-carboxamide
—— Ethyl 4-[2-hydroxyethyl(methyl)amino]-5-methyl-2-(morpholin-4-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxylate —— C18H26N4O4S
Ethyl 4-[2-hydroxyethyl(methyl)amino]-5-methyl-2-(morpholin-4-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxylate
—— 6-methyl-5-phenyl-3-[(Z)-(4-propoxyphenyl)methylideneamino]thieno[2,3-d]pyrimidin-4-one —— C23H21N3O2S
6-methyl-5-phenyl-3-[(Z)-(4-propoxyphenyl)methylideneamino]thieno[2,3-d]pyrimidin-4-one
—— 2-[[(7S)-7-methyl-2-(morpholin-4-ylmethyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl]sulfanyl]ethanol —— C18H25N3O2S2
2-[[(7S)-7-methyl-2-(morpholin-4-ylmethyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl]sulfanyl]ethanol
—— 5-methyl-4-(3-morpholin-4-ylpropylamino)-N-[[(1R,2R,4R)-spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-yl]methyl]thieno[2,3-d]pyrimidine-6-carboxamide —— C25H33N5O2S
5-methyl-4-(3-morpholin-4-ylpropylamino)-N-[[(1R,2R,4R)-spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-yl]methyl]thieno[2,3-d]pyrimidine-6-carboxamide
—— 5-methyl-4-(3-morpholin-4-ylpropylamino)-N-[[(1R,2S,4R)-spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-yl]methyl]thieno[2,3-d]pyrimidine-6-carboxamide —— C25H33N5O2S
5-methyl-4-(3-morpholin-4-ylpropylamino)-N-[[(1R,2S,4R)-spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-yl]methyl]thieno[2,3-d]pyrimidine-6-carboxamide
—— 2-[[5,6-Dimethyl-2-(phenylsulfanylmethyl)thieno[2,3-d]pyrimidin-4-yl]-methylamino]ethanol —— C18H21N3OS2
2-[[5,6-Dimethyl-2-(phenylsulfanylmethyl)thieno[2,3-d]pyrimidin-4-yl]-methylamino]ethanol
—— 4-[[12-(Benzotriazol-1-yl)-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(12),2(6),8,10-tetraen-10-yl]methyl]morpholine —— C20H20N6OS
4-[[12-(Benzotriazol-1-yl)-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(12),2(6),8,10-tetraen-10-yl]methyl]morpholine
—— 4-[[(7R)-4-(benzotriazol-1-yl)-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl]methyl]morpholine —— C22H24N6OS
4-[[(7R)-4-(benzotriazol-1-yl)-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl]methyl]morpholine
—— 2-[Methyl-[10-[(4-methylpiperidin-1-ium-1-yl)methyl]-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(12),2(6),8,10-tetraen-12-yl]amino]ethanol —— C19H29N4OS+
2-[Methyl-[10-[(4-methylpiperidin-1-ium-1-yl)methyl]-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(12),2(6),8,10-tetraen-12-yl]amino]ethanol
—— 2-[methyl-[(7S)-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl]amino]ethanol —— C14H19N3OS
2-[methyl-[(7S)-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl]amino]ethanol
—— (7R)-2-[(1S)-1-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylsulfanyl)ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H24N2O3S2
(7R)-2-[(1S)-1-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylsulfanyl)ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-2-[(1S)-1-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylsulfanyl)ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H24N2O3S2
(7S)-2-[(1S)-1-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylsulfanyl)ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (2R,6R)-2,6-dimethyl-4-[10-(morpholin-4-ium-4-ylmethyl)-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(12),2(6),8,10-tetraen-12-yl]morpholine —— C20H29N4O2S+
(2R,6R)-2,6-dimethyl-4-[10-(morpholin-4-ium-4-ylmethyl)-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(12),2(6),8,10-tetraen-12-yl]morpholine
—— 4-[(5,6-Dimethyl-4-pyrrolidin-1-ylthieno[2,3-d]pyrimidin-2-yl)methyl]morpholin-4-ium —— C17H25N4OS+
4-[(5,6-Dimethyl-4-pyrrolidin-1-ylthieno[2,3-d]pyrimidin-2-yl)methyl]morpholin-4-ium
—— 10-(morpholin-4-ium-4-ylmethyl)-N-[(1S)-1-phenylethyl]-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(12),2(6),8,10-tetraen-12-amine —— C22H27N4OS+
10-(morpholin-4-ium-4-ylmethyl)-N-[(1S)-1-phenylethyl]-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(12),2(6),8,10-tetraen-12-amine
—— (7R)-2-[(1R)-1-[[5-[(4-methoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C23H24N4O3S2
(7R)-2-[(1R)-1-[[5-[(4-methoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (2R,6S)-2,6-dimethyl-4-[(7R)-7-methyl-2-(morpholin-4-ium-4-ylmethyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl]morpholine —— C22H33N4O2S+
(2R,6S)-2,6-dimethyl-4-[(7R)-7-methyl-2-(morpholin-4-ium-4-ylmethyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl]morpholine
—— (2R,6R)-2,6-dimethyl-4-[(7R)-7-methyl-2-(morpholin-4-ylmethyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl]morpholine —— C22H32N4O2S
(2R,6R)-2,6-dimethyl-4-[(7R)-7-methyl-2-(morpholin-4-ylmethyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl]morpholine
—— 10-(morpholin-4-ium-4-ylmethyl)-N-[(1R)-1-phenylethyl]-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(12),2(6),8,10-tetraen-12-amine —— C22H27N4OS+
10-(morpholin-4-ium-4-ylmethyl)-N-[(1R)-1-phenylethyl]-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(12),2(6),8,10-tetraen-12-amine
—— 10-(morpholin-4-ylmethyl)-N-[[(2S)-oxolan-2-yl]methyl]-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(12),2(6),8,10-tetraen-12-amine —— C19H26N4O2S
10-(morpholin-4-ylmethyl)-N-[[(2S)-oxolan-2-yl]methyl]-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(12),2(6),8,10-tetraen-12-amine
—— (7S)-2-[(1R)-1-[[5-[(4-methoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C23H24N4O3S2
(7S)-2-[(1R)-1-[[5-[(4-methoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 4-[[12-[(2R)-2-ethylpiperidin-1-yl]-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(12),2(6),8,10-tetraen-10-yl]methyl]morpholine —— C21H30N4OS
4-[[12-[(2R)-2-ethylpiperidin-1-yl]-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(12),2(6),8,10-tetraen-10-yl]methyl]morpholine
—— 5,6-Dimethyl-2-[(4-methylpiperidin-1-yl)methyl]-4-pyrrolidin-1-ylthieno[2,3-d]pyrimidine —— C19H28N4S
5,6-Dimethyl-2-[(4-methylpiperidin-1-yl)methyl]-4-pyrrolidin-1-ylthieno[2,3-d]pyrimidine
—— (7S)-2-[(1S)-1-[[5-[(4-methoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C23H24N4O3S2
(7S)-2-[(1S)-1-[[5-[(4-methoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-[(1S)-1-[[5-[(4-methoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C23H24N4O3S2
(7R)-2-[(1S)-1-[[5-[(4-methoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (6S)-6-(2-methylbutan-2-yl)-N-[(E)-(3-nitrophenyl)methylideneamino]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine —— C22H25N5O2S
(6S)-6-(2-methylbutan-2-yl)-N-[(E)-(3-nitrophenyl)methylideneamino]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine
—— N-(1-adamantylmethyl)-2-[[(7S)-3-(3-chloro-4-methylphenyl)-7-methyl-4-oxo-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl]sulfanyl]acetamide —— C31H36ClN3O2S2
N-(1-adamantylmethyl)-2-[[(7S)-3-(3-chloro-4-methylphenyl)-7-methyl-4-oxo-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl]sulfanyl]acetamide
—— (6R)-6-(2-methylbutan-2-yl)-N-[(E)-(3-nitrophenyl)methylideneamino]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine —— C22H25N5O2S
(6R)-6-(2-methylbutan-2-yl)-N-[(E)-(3-nitrophenyl)methylideneamino]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine
—— N-(1-adamantylmethyl)-2-[[(7R)-3-(3-chloro-4-methylphenyl)-7-methyl-4-oxo-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl]sulfanyl]acetamide —— C31H36ClN3O2S2
N-(1-adamantylmethyl)-2-[[(7R)-3-(3-chloro-4-methylphenyl)-7-methyl-4-oxo-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl]sulfanyl]acetamide
—— methyl 2-[[(2R)-2-[(5,6-dimethyl-4-oxo-3H-thieno[2,3-d]pyrimidin-2-yl)methylsulfanyl]propanoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C22H25N3O4S3
methyl 2-[[(2R)-2-[(5,6-dimethyl-4-oxo-3H-thieno[2,3-d]pyrimidin-2-yl)methylsulfanyl]propanoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— methyl 2-[[(2S)-2-[(5,6-dimethyl-4-oxo-3H-thieno[2,3-d]pyrimidin-2-yl)methylsulfanyl]propanoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C22H25N3O4S3
methyl 2-[[(2S)-2-[(5,6-dimethyl-4-oxo-3H-thieno[2,3-d]pyrimidin-2-yl)methylsulfanyl]propanoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— 3-[2-[(2R)-2-(4-methoxyphenyl)azepan-1-yl]-2-oxoethyl]thieno[2,3-d]pyrimidin-4-one —— C21H23N3O3S
3-[2-[(2R)-2-(4-methoxyphenyl)azepan-1-yl]-2-oxoethyl]thieno[2,3-d]pyrimidin-4-one
—— 2-[5-ethyl-6-methyl-4-oxo-3-[[(2S)-oxolan-2-yl]methyl]thieno[2,3-d]pyrimidin-2-yl]sulfanyl-N,N-bis(prop-2-enyl)acetamide —— C22H29N3O3S2
2-[5-ethyl-6-methyl-4-oxo-3-[[(2S)-oxolan-2-yl]methyl]thieno[2,3-d]pyrimidin-2-yl]sulfanyl-N,N-bis(prop-2-enyl)acetamide
—— N'-[5-(4-methoxyphenyl)thieno[2,3-d]pyrimidin-4-yl]-N,N,2,2-tetramethylpropane-1,3-diamine —— C20H26N4OS
N'-[5-(4-methoxyphenyl)thieno[2,3-d]pyrimidin-4-yl]-N,N,2,2-tetramethylpropane-1,3-diamine
—— [3-[[5-(4-Methoxyphenyl)thieno[2,3-d]pyrimidin-4-yl]amino]-2,2-dimethylpropyl]-dimethylazanium —— C20H27N4OS+
[3-[[5-(4-Methoxyphenyl)thieno[2,3-d]pyrimidin-4-yl]amino]-2,2-dimethylpropyl]-dimethylazanium
—— (6R)-N-[(E)-(2,4-dichlorophenyl)methylideneamino]-6-(2-methylbutan-2-yl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine —— C22H24Cl2N4S
(6R)-N-[(E)-(2,4-dichlorophenyl)methylideneamino]-6-(2-methylbutan-2-yl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine
—— (6S)-N-[(E)-(2,4-dichlorophenyl)methylideneamino]-6-(2-methylbutan-2-yl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine —— C22H24Cl2N4S
(6S)-N-[(E)-(2,4-dichlorophenyl)methylideneamino]-6-(2-methylbutan-2-yl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine
—— [(7R)-7-methyl-4-oxo-3-phenyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl] (1E)-N-anilino-2-oxopropanimidothioate —— C26H24N4O2S2
[(7R)-7-methyl-4-oxo-3-phenyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl] (1E)-N-anilino-2-oxopropanimidothioate
—— (6R)-N-[(E)-1-(4-ethoxyphenyl)ethylideneamino]-6-(2-methylbutan-2-yl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine —— C25H32N4OS
(6R)-N-[(E)-1-(4-ethoxyphenyl)ethylideneamino]-6-(2-methylbutan-2-yl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine
—— (6S)-N-[(E)-1-(4-ethoxyphenyl)ethylideneamino]-6-(2-methylbutan-2-yl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine —— C25H32N4OS
(6S)-N-[(E)-1-(4-ethoxyphenyl)ethylideneamino]-6-(2-methylbutan-2-yl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine
—— (6S)-N-[(E)-(4-ethylphenyl)methylideneamino]-6-(2-methylbutan-2-yl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine —— C24H30N4S
(6S)-N-[(E)-(4-ethylphenyl)methylideneamino]-6-(2-methylbutan-2-yl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine
—— (6R)-N-[(E)-(4-ethylphenyl)methylideneamino]-6-(2-methylbutan-2-yl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine —— C24H30N4S
(6R)-N-[(E)-(4-ethylphenyl)methylideneamino]-6-(2-methylbutan-2-yl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine