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异恶唑并吡啶类

中文名称 英文名称 CAS号 化学式
—— (2,4-dimethyl-1,3-thiazol-5-yl)-[(3R)-3-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]methanone —— C20H21F3N4O2S
—— 5-[[4-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]methyl]-N-methylpyrimidin-2-amine —— C20H23F3N6O
—— (5-ethyl-4-methyl-1H-pyrazol-3-yl)-[4-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]methanone —— C21H24F3N5O2
—— (5-Ethyl-1,2-oxazol-3-yl)-[4-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]methanone —— C20H21F3N4O3
—— 1-[(3R)-3-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-3-pyrazol-1-ylpropan-1-one —— C20H22F3N5O2
—— 1-[(3R)-3-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-2-(4-methylpyrazol-1-yl)ethanone —— C20H22F3N5O2
—— 1-[4-[6-Ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-4-pyridin-4-ylbutan-1-one —— C23H25F3N4O2
—— 2-(3,5-dimethyl-1,2,4-triazol-1-yl)-1-[(3S)-3-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]ethanone —— C20H23F3N6O2
—— (2,4-dimethyl-1,3-thiazol-5-yl)-[(3S)-3-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]methanone —— C20H21F3N4O2S
—— [4-[6-Ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-(2-methylpyrazol-3-yl)methanone —— C19H20F3N5O2
—— [4-[6-Ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-pyridin-2-ylmethanone —— C20H19F3N4O2
—— 3-[1-[(2R)-butan-2-yl]sulfonylpiperidin-4-yl]-6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridine —— C18H24F3N3O3S
—— 1-[(3S)-3-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-3-(1,2,4-triazol-1-yl)propan-1-one —— C19H21F3N6O2
—— 1-[4-[6-Ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-3-(3-methylpyrazol-1-yl)propan-1-one —— C21H24F3N5O2
—— 6-Ethyl-3-(1-propan-2-ylsulfonylpiperidin-4-yl)-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridine —— C17H22F3N3O3S
—— (5-Cyclopropyl-2-methylpyrazol-3-yl)-[4-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]methanone —— C22H24F3N5O2
—— [(3R)-3-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-(1H-pyrazol-5-yl)methanone —— C18H18F3N5O2
—— cyclopentyl-[(3S)-3-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]methanone —— C20H24F3N3O2
—— 1-[4-[6-Ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-4-(1,2,4-triazol-1-yl)butan-1-one —— C20H23F3N6O2
—— [(3S)-3-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-(1-methylpyrazol-4-yl)methanone —— C19H20F3N5O2
—— 6-Ethyl-3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridine —— C20H21F3N4O
—— 1-[4-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-3-[(2S)-oxolan-2-yl]propan-1-one —— C21H26F3N3O3
—— 1-[(3S)-3-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-2-(4-methylpyrazol-1-yl)ethanone —— C20H22F3N5O2
—— [(3S)-3-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-(1-propan-2-ylpyrazol-4-yl)methanone —— C21H24F3N5O2
—— 1-[4-[6-Ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-3-pyrazol-1-ylpropan-1-one —— C20H22F3N5O2
—— [4-[6-Ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-(2-methyl-5-propan-2-ylpyrazol-3-yl)methanone —— C22H26F3N5O2
—— 2-(3,5-dimethyl-1,2,4-triazol-1-yl)-1-[(3R)-3-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]ethanone —— C20H23F3N6O2
—— (2R)-1-[(3R)-3-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-2-methyl-3-(1,2,4-triazol-1-yl)propan-1-one —— C20H23F3N6O2
—— Cyclopropyl-[4-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]methanone —— C18H20F3N3O2
—— [4-[6-Ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-(1-propan-2-ylpyrazol-4-yl)methanone —— C21H24F3N5O2
—— [4-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-[(1S,3R)-3-methoxycyclohexyl]methanone —— C22H28F3N3O3
—— (2,4-Dimethyl-1,3-thiazol-5-yl)-[4-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]methanone —— C20H21F3N4O2S
—— [(3R)-3-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-(3-methyl-1,2-oxazol-5-yl)methanone —— C19H19F3N4O3
—— 2-(3,5-Dimethylpyrazol-1-yl)-1-[4-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]ethanone —— C21H24F3N5O2
—— 1-[(3R)-3-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-3-imidazol-1-ylpropan-1-one —— C20H22F3N5O2
—— [(3S)-3-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-(5-propan-2-yl-1,2-oxazol-3-yl)methanone —— C21H23F3N4O3
—— [4-[6-Ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-(3-methyl-1,2-oxazol-5-yl)methanone —— C19H19F3N4O3
—— 1-[4-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-2-[[(2S)-oxolan-2-yl]methoxy]ethanone —— C21H26F3N3O4
—— (2S)-1-[(3R)-3-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-2-(1,2,4-triazol-1-yl)propan-1-one —— C19H21F3N6O2
—— 1-[(3R)-3-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-3-methoxypropan-1-one —— C18H22F3N3O3
—— [(3S)-3-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-[(2S)-oxolan-2-yl]methanone —— C19H22F3N3O3
—— [4-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-[(2R)-oxolan-2-yl]methanone —— C19H22F3N3O3
—— 1-[(3S)-3-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-4-imidazol-1-ylbutan-1-one —— C21H24F3N5O2
—— 1-[(3S)-3-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-4-(1,2,4-triazol-1-yl)butan-1-one —— C20H23F3N6O2
—— [(3S)-3-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-(2-methylpyrazol-3-yl)methanone —— C19H20F3N5O2
—— [4-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-(1H-pyrazol-5-yl)methanone —— C18H18F3N5O2
—— 1-[(3R)-3-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-3-(1,2,4-triazol-1-yl)propan-1-one —— C19H21F3N6O2
—— [(3S)-3-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-pyridin-3-ylmethanone —— C20H19F3N4O2
—— Cyclopentyl-[4-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]methanone —— C20H24F3N3O2
—— (1,3-Dimethylpyrazol-4-yl)-[4-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]methanone —— C20H22F3N5O2