| 中文名称 | 英文名称 | CAS号 | 化学式 |
|---|---|---|---|
| —— | 5-[5-[(1R,2R)-2-methylcyclopropyl]-1,3,4-oxadiazol-2-yl]-3-phenyl-[1,2]oxazolo[5,4-b]pyridine | —— | C18H14N4O2 |
| —— | 5-[5-[(1R,2S)-2-methylcyclopropyl]-1,3,4-oxadiazol-2-yl]-3-phenyl-[1,2]oxazolo[5,4-b]pyridine | —— | C18H14N4O2 |
| —— | 5-[5-[(1S,2S)-2-methylcyclopropyl]-1,3,4-oxadiazol-2-yl]-3-phenyl-[1,2]oxazolo[5,4-b]pyridine | —— | C18H14N4O2 |
| —— | 5-[5-[(1S,2R)-2-methylcyclopropyl]-1,3,4-oxadiazol-2-yl]-3-phenyl-[1,2]oxazolo[5,4-b]pyridine | —— | C18H14N4O2 |
| —— | (3-methyl-[1,2]oxazolo[5,4-b]pyridin-5-yl)-[(2R)-2-(1,3,5-trimethylpyrazol-4-yl)pyrrolidin-1-yl]methanone | —— | C18H21N5O2 |
| —— | (3-methyl-[1,2]oxazolo[5,4-b]pyridin-5-yl)-[(2S)-2-(1,3,5-trimethylpyrazol-4-yl)pyrrolidin-1-yl]methanone | —— | C18H21N5O2 |
| —— | (3R)-N-(3-methyl-[1,2]oxazolo[5,4-b]pyridin-5-yl)-1-methylsulfonylpiperidine-3-carboxamide | —— | C14H18N4O4S |
| —— | (3S)-N-(3-methyl-[1,2]oxazolo[5,4-b]pyridin-5-yl)-1-methylsulfonylpiperidine-3-carboxamide | —— | C14H18N4O4S |
| —— | [(1S,2R)-2-methylcyclopropyl]-[(3S)-3-[6-propan-2-yl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]methanone | —— | C20H24F3N3O2 |
| —— | (2S)-2-methyl-1-[(3S)-3-[6-propan-2-yl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-3-pyrazol-1-ylpropan-1-one | —— | C22H26F3N5O2 |
| —— | [(2R)-oxolan-2-yl]-[(3S)-3-[6-propan-2-yl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]methanone | —— | C20H24F3N3O3 |
| —— | (2S)-1-[(3S)-3-[6-propan-2-yl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-2-(1,2,4-triazol-1-yl)propan-1-one | —— | C20H23F3N6O2 |
| —— | (2S)-2-(5-methylpyrazol-1-yl)-1-[(3S)-3-[6-propan-2-yl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]propan-1-one | —— | C22H26F3N5O2 |
| —— | (2S)-1-[(3S)-3-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-2-methyl-3-pyrazol-1-ylpropan-1-one | —— | C21H24F3N5O2 |
| —— | (3R)-1-[(3R)-3-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-3-imidazol-1-ylbutan-1-one | —— | C21H24F3N5O2 |
| —— | [(1S,2S)-2-methylcyclopropyl]-[(3R)-3-[6-methyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]methanone | —— | C18H20F3N3O2 |
| —— | (3S)-3-imidazol-1-yl-1-[(3S)-3-[6-propan-2-yl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]butan-1-one | —— | C22H26F3N5O2 |
| —— | 4-(difluoromethyl)-3-methyl-6-[(3R)-1-(pyridin-4-ylmethyl)piperidin-3-yl]-[1,2]oxazolo[5,4-b]pyridine | —— | C19H20F2N4O |
| —— | (2R)-1-[(3R)-3-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-2-(5-methylpyrazol-1-yl)propan-1-one | —— | C21H24F3N5O2 |
| —— | (3R)-3-imidazol-1-yl-1-[(3R)-3-[6-propan-2-yl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]butan-1-one | —— | C22H26F3N5O2 |
| —— | [(1S,3S)-3-methoxycyclohexyl]-[4-[6-methyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]methanone | —— | C21H26F3N3O3 |
| —— | 1-[(3R)-3-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-3-(4-methylpyrazol-1-yl)propan-1-one | —— | C21H24F3N5O2 |
| —— | (2R)-1-[(3R)-3-[6-propan-2-yl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-2-(1,2,4-triazol-1-yl)propan-1-one | —— | C20H23F3N6O2 |
| —— | (3S)-1-[(3R)-3-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-3-imidazol-1-ylbutan-1-one | —— | C21H24F3N5O2 |
| —— | (3S)-1-[(3R)-3-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-3-pyrazol-1-ylbutan-1-one | —— | C21H24F3N5O2 |
| —— | (3R)-1-[(3R)-3-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-3-pyrazol-1-ylbutan-1-one | —— | C21H24F3N5O2 |
| —— | (2S)-1-[(3S)-3-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-2-methyl-3-(3-methylpyrazol-1-yl)propan-1-one | —— | C22H26F3N5O2 |
| —— | (2R)-2-imidazol-1-yl-1-[(3R)-3-[6-propan-2-yl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]propan-1-one | —— | C21H24F3N5O2 |
| —— | [4-[4-(difluoromethyl)-3-methyl-[1,2]oxazolo[5,4-b]pyridin-6-yl]piperidin-1-yl]-[(3S)-1,1-dioxothiolan-3-yl]methanone | —— | C18H21F2N3O4S |
| —— | (2R)-2-methyl-1-[(3R)-3-[6-propan-2-yl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-3-pyrazol-1-ylpropan-1-one | —— | C22H26F3N5O2 |
| —— | 3-[(2R)-oxolan-2-yl]-1-[(3S)-3-[6-propan-2-yl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]propan-1-one | —— | C22H28F3N3O3 |
| —— | (3R)-1-[(3S)-3-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-3-imidazol-1-ylbutan-1-one | —— | C21H24F3N5O2 |
| —— | (2R)-1-[(3S)-3-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-2-(5-methylpyrazol-1-yl)propan-1-one | —— | C21H24F3N5O2 |
| —— | (2S)-1-[(3R)-3-[6-propan-2-yl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-2-(1,2,4-triazol-1-yl)propan-1-one | —— | C20H23F3N6O2 |
| —— | (2R)-1-[(3S)-3-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-2-methyl-3-(3-methylpyrazol-1-yl)propan-1-one | —— | C22H26F3N5O2 |
| —— | (3R)-1-[(3R)-3-[6-propan-2-yl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-3-pyrazol-1-ylbutan-1-one | —— | C22H26F3N5O2 |
| —— | (2S)-3-(3,5-dimethylpyrazol-1-yl)-2-methyl-1-[(3S)-3-[6-methyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]propan-1-one | —— | C22H26F3N5O2 |
| —— | (2S)-2-(5-methylpyrazol-1-yl)-1-[(3R)-3-[6-propan-2-yl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]propan-1-one | —— | C22H26F3N5O2 |
| —— | (2R)-1-[4-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-2-(5-methylpyrazol-1-yl)propan-1-one | —— | C21H24F3N5O2 |
| —— | (2R)-1-[(3S)-3-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-2-methyl-3-pyrazol-1-ylpropan-1-one | —— | C21H24F3N5O2 |
| —— | (2R)-2-(5-methylpyrazol-1-yl)-1-[(3S)-3-[6-propan-2-yl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]propan-1-one | —— | C22H26F3N5O2 |
| —— | (2S)-2-imidazol-1-yl-1-[(3R)-3-[6-propan-2-yl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]propan-1-one | —— | C21H24F3N5O2 |
| —— | (3R)-1-[4-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-3-pyrazol-1-ylbutan-1-one | —— | C21H24F3N5O2 |
| —— | (2S)-1-[4-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-2-(5-methylpyrazol-1-yl)propan-1-one | —— | C21H24F3N5O2 |
| —— | (3S)-1-[(3S)-3-[6-propan-2-yl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-3-pyrazol-1-ylbutan-1-one | —— | C22H26F3N5O2 |
| —— | 2-methoxy-1-[(3S)-3-[6-propan-2-yl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]ethanone | —— | C18H22F3N3O3 |
| —— | (3S)-1-[(3S)-3-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-3-imidazol-1-ylbutan-1-one | —— | C21H24F3N5O2 |
| —— | (2R)-1-[(3R)-3-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-2-methyl-3-(3-methylpyrazol-1-yl)propan-1-one | —— | C22H26F3N5O2 |
| —— | (2S)-1-[(3S)-3-[6-ethyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]-2-(5-methylpyrazol-1-yl)propan-1-one | —— | C21H24F3N5O2 |
| —— | [(2S)-oxolan-2-yl]-[(3S)-3-[6-propan-2-yl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidin-1-yl]methanone | —— | C20H24F3N3O3 |