激动剂抑制剂-摩熵化学

中文名称	英文名称	CAS号	化学式
(6R)-6-[[[(4-氯苯基)磺酰基]氨基]-5,6,7,8-四氢-2-甲基-1-萘丙酸	Terutroban	165538-40-9	C₂₀H₂₂ClNO₄S
(5Z,8Z,11Z,14Z)-N-环丙基-5,8,11,14-二十碳四烯酰胺	arachidonylcyclopropylamide	229021-64-1	C₂₃H₃₇NO
(5R)-5-[(7-氯-1H-吲哚-3-基)甲基]-3-甲基-2,4-咪唑烷二酮	(R)-5-((7-chloro-1H-indol-3-yl)methyl)-3-methylimidazolidine-2,4-dione	852391-19-6	C₁₃H₁₂ClN₃O₂
(5-甲氧基-1H-吲哚-2-基)苯基甲酮	(5-methoxy-1H-indol-2-yl)(phenyl)methanone	74588-78-6	C₁₆H₁₃NO₂
(4S,4aS,5aR,12aS)-4-(二甲基氨基)-1,4,4a,5,5a,6,11,12a-八氢-3,10,12,12a-四羟基-7-[(甲氧基甲基氨基)甲基]-1,11-二氧代-2-并四苯甲酰胺盐酸盐	Sarecycline Hydrochloride	1035979-44-2	C24H30ClN3O8
(4S)-8-氯-6-(4-氯苯基)-1-甲基-4H-异恶唑并[5,4-d][2]苯并氮杂卓-4-乙酰胺	2-[(4S)-8-chloro-6-(4-chlorophenyl)-1-methyl-4H-[1,2]oxazolo[5,4-d][2]benzazepin-4-yl]acetamide	1380087-86-4	C₂₀H₁₅Cl₂N₃O₂
(4R)-甘氨酰基-4-(苯甲酰基氨基)-L-脯氨酸盐酸盐	Danegaptide hydrochloride	943133-81-1	C₁₄H₁₇N₃O₄*ClH
(4-环丙基哌嗪-1-基)-[4-(吗啉-4-基甲基)苯基]甲酮	Bavisant	929622-08-2	C₁₉H₂₇N₃O₂
(4-溴苯基)[2-氟-4-[[6-(甲基-2-丙烯基氨基)己基]氧基]苯基]甲酮	[4-[6-(allyl-methyl-amino)-hexyloxy]-2-fluoro-phenyl]-(4-bromo-phenyl)-methanone	161582-11-2	C₂₃H₂₇BrFNO₂
(3aR,4S,7aR)-八氢-4-羟基-4-[2-(3-甲基苯基)乙炔基]-1H-吲哚-1-羧酸甲酯	mavoglurant	543906-09-8	C₁₉H₂₃NO₃
(3S-反式)-1,4-二氢-7-[3-甲氧基-4-(甲基氨基)-1-吡咯烷基]-4-氧代-1-(2-噻唑基)-1,8-萘啶-3-羧酸单盐酸盐	AG-7352 hydrochloride	175519-16-1	C₁₈H₁₉N₅O₄S*ClH
(3S,5R,8R,9S,10S,13R,14S,17R)-17-(3-呋喃基)-10,13-二甲基-2,3,4,5,6,7,8,9,11,12,15,16-十二氢-1H-环戊二烯并[a]菲-3,14,17-三酚	17-β-(3-furyl)-5-β-androstane-3-β, 14-β, 17-α-triol	156722-18-8	C₂₃H₃₄O₄
(3S)-N-[2-[2-(二甲基氨基)乙氧基]-4-(1H-吡唑-4-基)苯基]-3,4-二氢-6-甲氧基-2H-1-苯并吡喃-3-甲酰胺	Chroman 1	1273579-40-0	C₂₄H₂₈N₄O₄
(3S)-2-(2,2-二苯基乙酰基)-1,2,3,4-四氢-6-甲氧基-5-苄氧基-3-异喹啉羧酸	EMA401	1316755-16-4	C₃₂H₂₉NO₅
(3R,4R)-4-氨基-1-[[4-[(3-甲氧基苯基)氨基]吡咯并[2,1-f][1,2,4]三嗪-5-基]甲基]哌啶-3-醇	BMS-690514	859853-30-8	C₁₉H₂₄N₆O₂
(3R)-N-[5-氯-4-(5-氟-2-甲氧基苯基)-2-吡啶基]-3-哌啶甲酰胺	(3R)-N-[5-chloro-4-(5-fluoro-2-methoxyphenyl)pyridin-2-yl]piperidine-3-carboxamide	1269815-17-9	C₁₈H₁₉ClFN₃O₂
(3R)-1,2,3,4-四氢-7-羟基-N-[(1S)-1-[[(3R,4R)-4-(3-羟基苯基)-3,4-二甲基-1-哌啶基]甲基]-2-甲基丙基]-3-异喹啉甲酰胺盐酸盐	JDTic dihydrochloride	785835-79-2	C28H41Cl2N3O3
(3E)-5-氯-3-[[5-[3-[(六氢-4-甲基-1H-14-二氮杂革-1-基)羰基]苯基]-2-呋喃]亚甲基]-1,3-二氢-2H-吲哚-2-酮	CX-6258	1202916-90-2	C₂₆H₂₄ClN₃O₃
(3-氯苯基)[3,4-二氢-6,7-二甲氧基-1-[[(4-甲氧基苯氧基)甲基]-2(1H)-异喹啉基]甲酮	(3-chlorophenyl)(6,7-dimethoxy-1-((4-methoxyphenoxy)methyl)-3,4-dihydroisoquinolin-2(1H)-yl)methanone	486427-17-2	C₂₆H₂₆ClNO₅
(2Z)-2-氰基-N-(2,5-二溴苯基)-3-羟基-2-丁烯酰胺	α-Cyano-β-hydroxy-β-methyl-N-(2,5-dibromophenyl)-propenamide	62004-35-7	C₁₁H₈Br₂N₂O₂
(2S,5R)-5-(4-((2-氟苄基)氧基)苯基)吡咯烷-2-甲酰胺盐酸盐	(5R)-5-(4-{[(2-fluorophenyl)methyl]oxy}phenyl)-L-prolinamide hydrochloride	934240-31-0	C₁₈H₁₉FN₂O₂*ClH
(2S,4R)-1-(2-氨基乙酰基)-4-苯甲酰胺吡咯烷-2-甲酸	(2S,4R)-1-(2-aminoacetyl)-4-benzoylamino-pyrrolidine-2-carboxylic acid	943134-39-2	C₁₄H₁₇N₃O₄
(2S,3S,4R,5R)-2-(4-氨基-5H-吡咯并[3,2-D]嘧啶-7-基)-5-(羟基甲基)-3,4-吡咯烷二醇单盐酸盐	(2S,3S,4R,5R)-2-(4-amino-5H-pyrrolo[3,2-d]pyrimidin-7-yl)-5-(hydroxymethyl)pyrrolidine-3,4-diol dihydrochloride	222631-44-9	C₁₁H₁₅N₅O₃*2ClH
(2S,3S)-3-[[3-(异丙基)-7-[(苯基甲基)氨基]吡唑并[1,5-a]嘧啶-5-基]氨基]-1,2,4-丁三醇	BS-194	1092443-55-4	C₂₀H₂₇N₅O₃
(2S,3S)-2-(3-氯苯基)-3,5,5-三甲基吗啉-2-醇	radafaxine	192374-14-4	C₁₃H₁₈ClNO₂
(2S,3R,4R,5S,6R)-2-(4-氯-3-(4-乙氧基苄基)苯基)-6-(甲基硫代)四氢-2H-吡喃-3,4,5-三醇	sotagliflozin	1018899-04-1	C₂₁H₂₅ClO₅S
(2S,3R)-3-羟基丁烷-1,2,3-三羧酸	(2S,3R)-3-hydroxybutane-1,2,3-tricarboxylic acid	71183-66-9	C₇H₁₀O₇
(2S)-N6,N6,2-三甲基-1,2-二氢-1,3,5-三嗪-4,6-二胺	Imeglimin	775351-65-0	C₆H₁₃N₅
(2S)-N-[(1R)-1-(1,3-苯并二氧戊环-5-基)丁基]-3,3-二乙基-2-[4-[(4-甲基-1-哌嗪基)羰基]苯氧基]-4-氧代-1-氮杂环丁烷甲酰胺	L-694,458	157341-41-8	C₃₁H₄₀N₄O₆
(2S)-2-氨基-2-[(1S,2S)-2-羧基环丙-1-基]-3-(吨-9-基)丙酸	2-[(1S,2S)-2-carboxycyclopropyl]-3-(9H-xanthen-9-yl)-D-alanine	201943-63-7	C₂₀H₁₉NO₅
(2S)-2-[[((2S)-6,8-二氟-1,2,3,4-四氢-2-萘基]氨基]-N-[1-[2-[(2,2-二甲基丙基))氨基]-1,1-二甲基乙基]-1H-咪唑-4-基]戊酰胺二氢溴化物	Nirogacestat Hydrobromide	1962925-29-6	C27H43Br2F2N5O
(2S)-2-[4-(乙酰基氨基)苯基]-N-(5-异丙基噻唑-2-基)丙酰胺	(2S)-2-[4-(acetylamino)phenyl]-N-(5-isopropyl-1,3-thiazol-2-yl)propanamide	492445-28-0	C₁₇H₂₁N₃O₂S
(2S)-2-(4-氯苯基)-1-[4-[(5R,7R)-6,7-二氢-7-羟基-5-甲基-5H-环戊并嘧啶-4-基]-1-哌嗪基]-3-[(1-甲基乙基)氨基]-1-丙酮二盐酸盐	Ipatasertib dihydrochloride	1396257-94-5	C24H34Cl3N5O2
(2S)-2-(3-氨基丙基)-5-(2,5-二氟苯基)-N-甲氧基-N-甲基-2-苯基-1,3,4-噻二唑-3(2H)-甲酰胺	filanesib	885060-09-3	C₂₀H₂₂F₂N₄O₂S
(2S)-2-((4-(((2,7-二甲基-4-氧代-1,4-二氢喹唑啉-6-基)甲基)(丙-2-炔基)氨基)-2-氟苯甲酰)氨基)-4-(1H-四唑-5-基)丁酸	narlaprevir	865466-24-6	C₃₆H₆₁N₅O₇S
(2R，3S，4S)-5-[4-(3,5-二氯苯基)苯基]-2,3-二羟基-4-(2-甲氧基乙酰胺基)戊酸	4,5-Dideoxy-5-(3',5'-Dichlorobiphenyl-4-Yl)-4-[(Methoxyacetyl)amino]-L-Arabinonic Acid	1319207-44-7	C₂₀H₂₁Cl₂NO₆
(2R,4S)-N-[1-[3,5-双(三氟甲基)苯甲酰]-2-(4-氯苄基)哌啶-4-基]喹啉-4-甲酰胺	(2R,4S)-N-[1-(3,5-bis(trifluoromethyl)benzoyl)-2-(4-chlorobenzyl)-4-piperidinyl]quinoline-4-carboxamide	177707-12-9	C₃₁H₂₄ClF₆N₃O₂
(2R,4'R,8'aR)-1-[2-[4-[[2-(2,4-二氯苯氧基)乙酰基]氨基]苯基]乙酰基]四氢-6'-氧代螺[吡咯烷-2,7'(6'H)-[2H]吡咯并[2,1-b][1,3]噻嗪]-4'-甲酰胺	ST2825	894787-30-5	C₂₇H₂₈Cl₂N₄O₅S
(2R,3R,4R,5S)-1-丁基-2-(羟基甲基)-3,4,5-哌啶三醇盐酸盐(1:1)	miglustat hydrochloride	210110-90-0	C₁₀H₂₁NO₄*ClH
(2R,2'R,3R,3'R,4S,4'S,5R,5'R,6S,6'S)-6,6'-硫代双(4-(4-(3-氟苯基)-1H-1,-1H-1,2,3-三唑-1-基)-2-(羟甲基)四氢-2H-吡喃-3,5-二醇)	TD139	1450824-22-2	C₂₈H₃₀F₂N₆O₈S
(2R)-2-[[6-[[(5-甲基噻吩-2-基)甲基]氨基]-9-丙基-9H-嘌呤-2-基]氨基]丁烷-1-醇	(2R)-2-[(6-{[(5-methylthiophen-2-yl)methyl]amino}-9-propyl-9H-purin-2-yl)amino]butan-1-ol	1402821-41-3	C₁₈H₂₆N₆OS
(2R)-2-[[6-[(3-氯-4-羧基苯基)氨基]-9-(1-甲基乙基)-9H-嘌呤-2-基]氨基]-3-甲基-1-丁醇(PURVALANOLB(NG95))	purvalanol B	212844-54-7	C₂₀H₂₅ClN₆O₃
(2R)-2-(3-氨基丙基)-5-(2,5-二氟苯基)-N-甲氧基-N-甲基-2-苯基-1,3,4-噻二唑-3(2H)-甲酰胺	(R)-Filanesib	885060-08-2	C₂₀H₂₂F₂N₄O₂S
(2R)-2,4-二甲基-1-哌嗪羧酸 4-[(3-氯-2-氟苯基)氨基]-7-甲氧基-6-喹唑啉基酯	AZD3759	1626387-80-1	C₂₂H₂₃ClFN₅O₃
(2R)-1-[[[4-氯-2-(脲基)苯氧基]甲基]羰基]-2-甲基-4-(4-氟苄基)哌嗪	1-(5-chloro-2-{2-[(2R)-4-(4-fluorobenzyl)-2-methylpiperazin-1-yl]-2-oxoethoxy}phenyl)urea	217645-70-0	C₂₁H₂₄ClFN₄O₃
(2E,5E)-2,5-二(2-噻吩基亚甲基)环戊酮	CCT007093	176957-55-4	C₁₅H₁₂OS₂
(2E,2'E)-1,1'-环己基亚基二[3-(3,4-二甲氧基苯基)-2-丙烯-1-酮]	FLLL32	1226895-15-3	C₂₈H₃₂O₆
(2E)-N-甲基-N-[(3-甲基-2-苯并呋喃基)甲基]-3-(5,6,7,8-四氢-7-氧代-1,8-萘啶-3-基)-2-丙烯酰胺	(2E)-N-methyl-N-[(3-methyl-1-benzofuran-2-yl)methyl]-3-(7-oxo-5,6,7,8-tetrahydro-1,8-naphthyridin-3-yl)prop-2-enamide	620175-39-5	C₂₂H₂₁N₃O₃
(2E)-3-苯基-N-[2,2,2-三氯-1-[[[(4-氯苯基)氨基]硫代甲酰基]氨基]乙基]-2-丙烯酰胺	(E)-3-phenyl-N-[2,2,2-trichloro-1-[(4-chlorophenyl)carbamothioylamino]ethyl]prop-2-enamide	301359-91-1	C₁₈H₁₅Cl₄N₃OS
(2E)-3-(4-溴苯基)-1-[4--4-甲氧基苯甲酰基)-1-哌嗪基]-2-丙烯-1-酮	NIBR189	1599432-08-2	C₂₁H₂₁BrN₂O₃

1-25
26-29