激动剂抑制剂-摩熵化学

中文名称	英文名称	CAS号	化学式
N-[2-氟-5-[[3-[(1E)-2-(2-吡啶基)乙烯基]-1H-吲唑-6-基]氨基]苯基]-1,3-二甲基-1H-吡唑-5-甲酰胺	AG-013958	319460-94-1	C₂₆H₂₂FN₇O
N-[2-[[2-(二甲基氨基)乙基]甲基氨基]-5-[[4-(1H-吲哚-3-基)-2-嘧啶基]氨基]-4-甲氧基苯基]-2-丙烯酰胺	AZ5104	1421373-98-9	C₂₇H₃₁N₇O₂
N-[2-[[(2,3-二氟苯基)甲基]硫基]-6-[[(1S,2R)-2,3-二羟基-1-甲基丙基]氨基]-4-嘧啶基]-1-氮杂环丁烷磺酰胺	N-(2-[(2,3-difluorobenzyl)thio]-6-{[(1S,2R)-2,3-dihydroxy-1-methylpropyl]amino}pyrimidin-4-yl)azetidine-1-sulfonamide	1204707-73-2	C₁₈H₂₃F₂N₅O₄S₂
N-[2-[[((3R)-1-][反式-4-羟基-4-(6-甲氧基-3-吡啶基)环己基]-3-吡咯烷基]氨基]-2-氧代乙基]-3-(三氟甲基)-苯甲酰胺二甲磺酸盐	INCB 3284 dimesylate	887401-93-6	C28H39F3N4O10S2
N-[2-[P-溴苯丙烯盐基氨基]乙基]-5-异喹啉磺酰胺	N-[2-(4-bromocinnamylamino)ethyl]isoquinoline-5-sulfonamide	127243-85-0	C₂₀H₂₀BrN₃O₂S
N-[2-[N-(4-氯肉桂)-N-甲基氨基]苯基]-N-(2-羟乙基)-4-甲氧苯磺酰胺磷酸酯盐	N-[2-({[(2E)-3-(4-chlorophenyl)prop-2-en-1-yl](methyl)amino}methyl)phenyl]-N-(2-hydroxyethyl)-4-methoxybenzenesulfonamide	139298-40-1	C₂₆H₂₉ClN₂O₄S
N-[2-[2-(二甲基氨基)乙基]-2,3-二氢-1,3-二氧代-1H-苯[de]异喹啉-5-基]脲R	UNBS-5126	956590-23-1	C₁₇H₁₈N₄O₃
N-[2-[2-(4-氯苯基)-4-噻唑基]乙基]丁酰胺	azoramide	932986-18-0	C₁₅H₁₇ClN₂OS
N-[2-[(R)-(3-氯苯基)[(3R)-1-[[[(2S)-2-(甲基氨基)-3-[(3R)-四氢-2H-吡喃-3-基]丙基]氨基]羰基]-3-哌啶基]甲氧基]乙基]氨基甲酸甲酯，2,2,2-三氟乙酸盐	VTP-27999 2,2,2-trifluoroacetate	1013937-63-7	C28H42ClF3N4O7
N-[2-[(R)-(3-氯苯基)[(3R)-1-[[[(2S)-2-(甲基氨基)-3-[(3R)-四氢-2H-吡喃-3-基]丙基]氨基]羰基]-3-哌啶基]甲氧基]乙基]氨基甲酸甲酯	VTP-27999	942142-51-0	C₂₆H₄₁ClN₄O₅
N-[2-[(3S)-3-[[4-羟基-4-[5-(嘧啶-2-基)吡啶-2-基]环己基]氨基]吡咯烷-1-基]-2-氧代乙基]-3-(三氟甲基)苯甲酰胺	PF-04136309	1341224-83-6	C₂₉H₃₁F₃N₆O₃
N-[2-(4'-氰基联苯-4-基)丙基]-2-丙烷磺酰胺	LY 404187	211311-95-4	C₁₉H₂₂N₂O₂S
N-[2-(3-溴苯基)乙基]-2,4,6-三甲基-N-[[3'-(甲基磺酰基)[1,1'-联苯]-4-基]甲基]苯磺酰胺	SR9243	1613028-81-1	C₃₁H₃₂BrNO₄S₂
N-[2-(2-吡啶基)-6-(1,2,4,5-四氢-3H-3-苯并氮杂卓-3-基)-4-嘧啶基]-beta-丙氨酸	GSK-J1	1373422-53-7	C₂₂H₂₃N₅O₂
N-[2,4-二氟-3-[[5-(3-吡啶基)-1H-吡咯并[2,3-B]吡啶-3-基]羰基]苯基]-2-丙磺酰胺	propane-2-sulfonic acid [2,4-difluoro-3-(5-pyridin-3-yl-1H-pyrrolo[2,3-b]pyridine-3-carbonyl)-phenyl]-amide	918505-61-0	C₂₂H₁₈F₂N₄O₃S
N-[1-[[(氰基氨基)(5-喹啉亚氨基)甲基]氨基]-2,2-二甲基丙基]-3,4-二甲氧基苯乙酰胺	N-[1-({(cyanoimino)[(5-quinolinyl)amino]methyl}amino)-2,2-dimethylpropyl]-2-(3,4-dimethoxyphenyl)acetamide	861393-28-4	C₂₆H₃₀N₆O₃
N-[1-(1-氧丙基)-4-哌啶基]-N'-[4-(三氟甲氧基)苯基]脲	TPPU	1222780-33-7	C₁₆H₂₀F₃N₃O₃
N-[1,4-二氢-3-[4-[[4-(2-甲氧基乙基)-1-哌嗪基]甲基]苯基]-4-氧代茚并[1,2-c]吡唑-5-基]-N'-4-吗啉基脲	RGB-286638	784210-88-4	C₂₉H₃₅N₇O₄
N-[(9H-氟代-9-甲氧基)羰基]-L-戊基-N5-(氨基羰基)-N-[4-[[[(4-硝基苯氧基)羰基]氧]甲基]苯基]-L-鸟氨酸酰胺	(9H-fluoren-9-yl)methyl (3-methyl-1-((1-((4-((((4-nitrophenoxy)carbonyl)oxy)methyl)phenyl)amino)-1-oxo-5-ureidopentan-2-yl)amino)-1-oxobutan-2-yl)carbamate	863971-53-3	C₄₀H₄₂N₆O₁₀
N-[(3R,4S)-3,4-二氢-3-[[(甲基氨基)羰基]氧基]-6-[4-(3-氧杂环丁基)-1-哌嗪基]-2H-1-苯并吡喃-4-基]-4-氟-苯甲酰胺	(3R,4S)-4-(4-fluorobenzamido)-6-(4-(oxetan-3-yl)piperazin-1-yl)chroman-3-yl methylcarbamate	1373215-15-6	C₂₅H₂₉FN₄O₅
N-[(3R,4R)-4-氟-1-[6-[（3-甲氧基-1-甲基-1H-吡唑-4-基）氨基]-9-甲基-9H-嘌呤-2-基]吡咯烷-3-基]丙烯酰胺	PF-06747775	1776112-90-3	C₁₈H₂₂FN₉O₂
N-[(3R)-3-(二甲基氨基)-2,3,4,9-四氢-1H-咔唑-6-基]-4-氟苯甲酰胺盐酸盐	N-[(6R)-6-(dimethylamino)-6,7,8,9-tetrahydro-5H-carbazol-3-yl]-4-fluorobenzamide	186544-26-3	C₂₁H₂₂FN₃O
N-[(1S)-2-[[(7S)-6,7-二氢-5-(2-羟基乙基)-6-氧代-5H-吡啶并[3,2-a][3]苯并氮杂卓-7-基]氨基]-1-甲基-2-氧代乙基]-4,4,4-三氟丁酰胺	LY3039478	1421438-81-4	C₂₂H₂₃F₃N₄O₄
N-[(1R,2R)-1-(2,3-二氢苯并[b][1,4]二恶英-6-基)-1-羟基-3-(吡咯烷-1-基)丙-2-基]壬酰胺	genz-123346	491833-30-8	C₂₄H₃₈N₂O₄
N-[(1-丁基-4-哌啶基)甲基]-3,4-二氢-2H-[1,3]噁嗪并[3,2-a]吲哚-10-羧胺	piboserod	152811-62-6	C₂₂H₃₁N₃O₂
N-[(1,3-二环己基六氢-2,4,6-三氧代-5-嘧啶基)羰基]甘氨酸	daprodustat	960539-70-2	C₁₉H₂₇N₃O₆
N-2-联苯基-7-硝基-2,1,3-苯并恶二唑-4-胺	N-([1,1'-biphenyl]-2-yl)-7-nitrobenzo[c][1,2,5]oxadiazol-4-amine	413611-93-5	C₁₈H₁₂N₄O₃
N-(氰基甲基)-4-[2-[[4-(4-吗啉基)苯基]氨基]-4-嘧啶基]苯甲酰胺硫酸盐(1:2)	Momelotinib sulfate	1056636-06-6	C23H26N6O10S2
N-(6-甲基-2-苯并噻唑基)-2-[(3,4,6,7-四氢-3-(2-甲氧基苯基)-4-氧噻吩并[3,2-d]嘧啶-2-基)硫代]-乙酰胺	2-((3-(2-methoxyphenyl)-4-oxo-3,4,6,7-tetrahydrothieno[3,2-d]pyrimidin-2-yl)thio)-N-(6-methylbenzo[d]thiazol-2-yl)acetamide	686772-17-8	C₂₃H₂₀N₄O₃S₃
N-(6-氯-9H-beta-咔啉-8-基)烟酰胺	N-(6-chloro-9H-β-carbolin-8-yl)nicotinamide	431898-65-6	C₁₇H₁₁ClN₄O
N-(6-氯-7-甲氧基-9h-吡啶并[3,4-b]吲哚-8-基)-2-甲基-3-吡啶羧酰胺	MLN120B	783348-36-7	C₁₉H₁₅ClN₄O₂
N-(5-氨基戊基)乙酰胺	N-acetylcadaverine	32343-73-0	C₇H₁₆N₂O
N-(5-乙基-2,4-二甲基苯基)-4-[3-氟-4-(4-甲基-1H-咪唑-1-基)苯基]-2-噻唑胺	N-(5-ethyl-2,4-dimethylphenyl)-4-(3-fluoro-4-(4-methyl-1H-imidazol-1-yl)phenyl)thiazol-2-amine	1304630-27-0	C₂₃H₂₃FN₄S
N-(5-((5-(4-乙酰基哌嗪-1-甲酰基)-4-甲氧基-2-甲基苯基)硫基)噻唑-2-基)-4-(((3-甲基丁烷-2-基)氨基)甲基)	HY-11066	439574-61-5	C₃₁H₃₉N₅O₄S₂
N-(5-((5-(4-乙酰基哌嗪-1-甲酰基)-4-甲氧基-2-甲基苯基)硫基)噻唑-2-基)-4-(((3,3-二甲基丁烷-2-基)氨基)甲基)苯甲酰胺	BMS-509744	439575-02-7	C₃₂H₄₁N₅O₄S₂
N-(4-溴苯基)-N'-(2,2,6,6-四甲基哌啶-4-基)草酰胺	N-(4-Bromophenyl)-N'-(2,2,6,6-Tetramethylpiperidin-4-Yl)ethanediamide	333352-59-3	C₁₇H₂₄BrN₃O₂
N-(4-氯苯基)-2-(3,5-二甲基-1H-吡唑-1-基)-9-甲基-9H-嘌呤-6-胺	(4-chloro-phenyl)-[2-(3,5-dimethyl-pyrazol-1-yl)-9-methyl-9H-purin-6-yl]-amine	1063331-94-1	C₁₇H₁₆ClN₇
N-(4-氯-3-吡啶基)-4-[(2,2-二氟-1,3-苯并二恶茂-5-基)甲基]-1-哌嗪甲酰胺	N-(4-chloropyridin-3-yl)-4-((2,2-difluorobenzo[d][1,3]dioxol-5-yl)methyl)piperazine-1-carboxamide	1346528-50-4	C₁₈H₁₇ClF₂N₄O₃
N-(4-异丙基-2-(3-氧代-3,4-二氢喹喔啉-2-基)苯基)噻吩-2-甲酰胺	N-(4-isopropyl-2-(3-oxo-3,4-dihydroquinoxalin-2-yl)phenyl)thiophene-2-carboxamide	1404437-62-2	C₂₂H₁₉N₃O₂S
N-(4-乙酰基-4,5-二氢-5-甲基-5-苯基-1,3,4-噻二唑-2-基)乙酰胺	(±)-N-(4-acetyl-5-methyl-5-phenyl-4,5-dihydro-1,3,4-thiadiazol-2-yl)acetamide	72926-24-0	C₁₃H₁₅N₃O₂S
N-(4-(3,4-二羟基苯基)-5-苯基噻唑-2-基)-3,4-二羟基苯甲酰胺	N-(4-(3,4-dihydroxyphenyl)-5-phenylthiazol-2-yl)-3 ,4-dihydroxybenzamide	1190932-38-7	C₂₂H₁₆N₂O₅S
N-(3-溴苯基)-6,7-二甲氧基-N-甲基-4-喹唑啉胺	EBE-A22	229476-53-3	C₁₇H₁₆BrN₃O₂
N-(3-溴-4-甲基苯基)-4-(4-吡啶甲基)-1-酞嗪胺	1-(3-Bromo-4-methyl-anilino)-4-(pyridin-4-yl-methyl)-phthalazine	300842-64-2	C₂₁H₁₇BrN₄
N-(3-氯-4-甲基苯基)-2-[2,6-二硝基-4-(三氟甲基)苯基]肼基硫代甲酰胺	N-(3-Chloro-4-methylphenyl)-2-[2,6-dinitro-4-(trifluoromethyl)phenyl]-hydrazinecarbothioamide	436133-68-5	C15H11ClF3N5O4S
N-(3-((2-((3-氟-4-(4-甲基哌嗪-1-基)苯基)氨基)-7H-吡咯并[2,3-D]嘧啶-4-基)氧基)苯基)丙烯酰胺酸盐	N-(3-(2-(3-fluoro-4-(4-methylpiperazin-1-yl)phenylamino)-7H-pyrrolo[2,3-d]pyrimidin-4-yloxy)phenyl)acrylamide maleate	1557268-88-8	C₄H₄O₄*C₂₆H₂₆FN₇O₂
N-(3,5-二氯-2-甲氧基苯基)-4-甲氧基-3-(1-哌嗪基)苯磺酰胺盐酸盐	SB 399885	402713-80-8	C₁₈H₂₁Cl₂N₃O₄S
N-(3,4-二氯苯基)-2-环己基-1H-咪唑并[4,5-c]喹啉-4-胺	LUF6000	890087-21-5	C₂₂H₂₀Cl₂N₄
N-(2-苯甲酰基苯基)-O-[2-(甲基-2-吡啶基氨基)乙基]-L-酪氨酸	(N-(2-benzoylphenyl)-O-[2-(methyl-2-pyridinylamino)ethyl]-L-tyrosine)	196808-24-9	C₃₀H₂₉N₃O₄
N-(2-氰基-3,12-二氧代-28-去甲齐墩果-1,9(11)-二烯-17-基)-2,2-二氟丙酰胺	omaveloxolone	1474034-05-3	C₃₃H₄₄F₂N₂O₃
N-(2-氯-5-甲氧基苯基)-6-甲氧基	N-(2-chloro-5-methoxyphenyl)-6-methoxy-7-((1-methylpiperidin-4-yl)methoxy)quinazolin-4-amine	476159-98-5	C₂₃H₂₇ClN₄O₃

1-25
26-29