激动剂抑制剂-摩熵化学

中文名称	英文名称	CAS号	化学式
N-[双(4-甲氧基苯基)甲基]-4-羟基-2-哒嗪-3-基嘧啶-5-甲酰胺	N-(bis(4-methoxyphenyl)methyl)-6-oxo-2-(pyridazin-3-yl)-1,6-dihydropyrimidine-5-carboxamide	1187990-87-9	C₂₄H₂₁N₅O₄
N-[[3-[5-(1-羟基-1-甲基乙基)-1,2,4-恶二唑-3-基]苯基]甲基]-2-(2-吡啶基)-5-嘧啶甲酰胺	2-(pyridin-2-yl)pyrimidine-5-carboxylic acid 3-[5-(1-hydroxy-1-methylethyl)-1,2,4]oxadiazol-3-yl-benzylamide	1234708-04-3	C₂₂H₂₀N₆O₃
N-[[(5S)-3-[3-氟-4-[4-(2-羟基乙酰基)-1-哌嗪基]苯基]-2-氧代-5-噁唑烷基]甲基]-乙酰胺	eperezolid	165800-04-4	C₁₈H₂₃FN₄O₅
N-[[(4-氨基苯基)氨基]硫代甲酰基]-4-(叔丁基)苯甲酰胺	4-(tert-butyl)-N-((4-aminophenyl)thiocarbamyl)benzamide	1011301-27-1	C₁₈H₂₁N₃OS
N-[7-氯-1-[(3R)-1-[(2E)-4-(二甲基氨基)-1-氧代-2-丁烯-1-基]六氢-1H-氮杂革-3-基]-1H-苯并咪唑-2-基]-2-甲基-4-吡啶羧酰胺	(R,E)-N-(7-chloro-1-(1-(4-(dimethylamino)but-2-enoyl)azepan-3-yl)-1H-benzo[d]imidazol-2-yl)-2-methylisonicotinamide	1508250-71-2	C₂₆H₃₁ClN₆O₂
N-[6-甲氧基-5-(2-甲氧基苯氧基)-2-(4-吡啶基)-4-嘧啶基]-5-甲基吡啶-2-磺酰胺	Avosentan	290815-26-8	C₂₃H₂₁N₅O₅S
N-[5-[[[5-(1,1-二甲基乙基)-2-恶唑基]甲基]硫基]-2-噻唑基]-4-哌啶甲酰胺L-酒石酸盐(2:1)	N-[5-[[[5-(1,1-Dimethylethyl)-2-oxazolyl]methyl]thio]-2-thiazolyl]-4-piperidinecarboxamide L-tartaric acid salt (2:1)	345627-92-1	C38H54N8O10S4
N-[5-[[6-[3-(1,3-二氧代异吲哚-2-基)苯基]嘧啶-4-基]氨基]-2-甲基苯基]甲烷磺酰胺	Cdk9-IN-1	1415559-43-1	C₂₆H₂₁N₅O₄S
N-[5-[3-(3-羟基-1-哌啶基)-1,2,4-恶二唑-5-基]-4-甲基-2-噻唑基]乙酰胺	N-{5-[3-(3-hydroxypiperidin-1-yl)-1,2,4-oxadiazol-5-yl]-4-methyl-1,3-thiazol-2-yl}acetamide	1292300-75-4	C₁₃H₁₇N₅O₃S
N-[5-[(1-甲基乙基)氨基]-7-(三氟甲基)[1,2,4]三唑并[1,5-a]吡啶-2-基]-3-吡啶甲酰胺	N-[5-(isopropylamino)-7-(trifluoromethyl)[1,2,4]triazolo[1,5-a]pyridin-2-yl]nicotinamide	1124381-69-6	C₁₆H₁₅F₃N₆O
N-[5-(氨基磺酰基)-4-甲基-1,3-噻唑-2-基]-N-甲基-2-(4-吡啶-2-基苯基)乙酰胺	N-[5-(aminosulfonyl)-4-methyl-1,3-thiazol-2-yl]-N-methyl-2-[4-(2-pyridinyl)-phenyl]acetamide	348086-71-5	C₁₈H₁₈N₄O₃S₂
N-[5-(4-氰基苯基)-1H-吡咯并[2,3-B]吡啶-3-基]-3-吡啶甲酰胺	N-[5-(4-cyanophenyl)-1H-pyrrolo[2,3-b]pyridin-3-yl]pyridine-3-carboxamide	1093222-27-5	C₂₀H₁₃N₅O
N-[4-氯-3-[5-(二甲基氨基)-1H-苯并咪唑-2-基]苯基]-3,5-二甲氧基苯甲酰胺	HhAntag	496794-70-8	C₂₄H₂₃ClN₄O₃
N-[4-氯-2-[(1,3-二氢-1,3-二氧代-2H-异吲哚-2-基)甲基]苯基]-2-羟基苯甲酰胺	CPPHA	693288-97-0	C₂₂H₁₅ClN₂O₄
N-[4-氟-3-(三氟甲基)苯基]-N'-[5-(4-吡啶基)-1,3,4-噻二唑-2-基]脲	ML216	1430213-30-1	C₁₅H₉F₄N₅OS
N-[4-乙酰基-2-(2,4-二氟苯氧基)苯基]-甲烷磺酰胺	N-[4-acetyl-2-(2,4-difluorophenoxy)phenyl]methanesulfonamide	116686-15-8	C₁₅H₁₃F₂NO₄S
N-[4-[[[[四氢-4-(4-甲氧基苯基)-2H-吡喃-4-基]甲基]氨基]羰基]苯基]-2-呋喃甲酰胺	JW55	664993-53-7	C₂₅H₂₆N₂O₅
N-[4-[[[[5-(叔丁基)-3-异恶唑基]氨基]羰基]氨基]苯基]-5-[(1-乙基-2,2,6,6-四甲基-4-哌啶基)氧基]-2-吡啶甲酰胺	N-(4-(3-(5-tert-butylisoxazol-3-yl)ureido)phenyl)-5-(1-ethyl-2,2,6,6-tetramethylpiperidin-4-yloxy)picolinamide	1351522-04-7	C₃₁H₄₂N₆O₄
N-[4-[[6-[4-(三氟甲基)苯基]-4-嘧啶基]氧基]-2-苯并噻唑基]乙酰胺	N-[4-[[6-[4-(trifluoromethyl)phenyl]-4-pyrimidinyl]oxy]-2-benzothiazolyl]acetamide	659730-32-2	C₂₀H₁₃F₃N₄O₂S
N-[4-[[3-氯-4-[(3-氟苯基)甲氧基]苯基]氨基]-6-喹唑啉]-2-丙酰胺	N-(4-(4-(3-fluorobenzyloxy)-3-chlorophenylamino)quinazolin-6-yl)acrylamide	897383-62-9	C₂₄H₁₈ClFN₄O₂
N-[4-[4-氨基-6-(甲氧基甲基)-7-(4-吗啉基甲基)吡咯并[2,1-f][1,2,4]三嗪-5-基]-2-氟苯基]-N'-[2-氟-5-(三氟甲基)苯基]脲	N-{4-[4-amino-6-(methoxymethyl)-7-(morpholin-4-ylmethyl)pyrrolo[2,1-f][1,2,4]triazin-5-yl]-2-fluorophenyl}-N'-[2-fluoro-5-(trifluoromethyl)phenyl]urea	939805-30-8	C₂₇H₂₆F₅N₇O₃
N-[4-[2,2,2-三氟-1-羟基-1-(三氟甲基)乙基]苯基]-2-噻吩磺酰胺	SR3335	293753-05-6	C₁₃H₉F₆NO₃S₂
N-[4-[1-[反式-4-(4-乙酰基-1-哌嗪基)环己基]-4-氨基-1H-吡唑并[3,4-D]嘧啶-3-基]-2-甲氧基苯基]-1-甲基-1H-吲哚-2-甲酰胺	1H-Indole-2-carboxamide, N-(4-(1-(trans-4-(4-acetyl-1-piperazinyl)cyclohexyl)-4-amino-1H-pyrazolo(3,4-d)pyrimidin-3-yl)-2-methoxyphenyl)-1-methyl-	869748-10-7	C₃₄H₃₉N₉O₃
N-[4-[(6,7-二甲氧基-4-喹啉基)氧基]-2-甲氧基苯基]-N’-[1-(2-噻唑基)乙基]脲	Ki20227	623142-96-1	C₂₄H₂₄N₄O₅S
N-[4-[(2-氨基-4-嘧啶基)氧基]苯基]-N'-[4-[(4-甲基-1-哌嗪基)甲基]-3-(三氟甲基)苯基]脲	K03861	853299-07-7	C₂₄H₂₆F₃N₇O₂
N-[4-[(1S)-1-[3,5-二甲基-4-[4-(三氟甲基)-1H-吡唑-1-基]苯氧基]丁基]苯甲酰基]-beta-丙氨酸	(S)-3-(4-(1-(3,5-dimethyl-4-(4-(trifluoromethyl)-1H-pyrazol-1-yl)phenoxy)butyl)benzamido)propanoic acid	1393124-08-7	C₂₆H₂₈F₃N₃O₄
N-[4-[(1R)-2-乙基-1-(1H-1,2,4-三唑-1-基)丁基]苯基]-2-苯并噻唑胺	(R)-Talarozole	870093-23-5	C₂₁H₂₃N₅S
N-[4-[(1R)-1-甲基-2-[[异丙基磺酰基]氨基]乙基]苯基]-3,5-二氟苯基甲酰胺	LY 450108	376594-67-1	C₁₉H₂₂F₂N₂O₃S
N-[4,6-二氨基-2-[1-[(2-氟苯基)甲基]-1H-吡唑并[3,4-b]吡啶-3-基]-5-嘧啶]-氨基甲酸甲酯	methyl 4,6-diamino-2-(1-(2-fluorobenzyl)-1H-pyrazolo[3,4-b] pyridin-3-yl)pyrimidin-5-ylcarbamate	625115-52-8	C₁₉H₁₇FN₈O₂
N-[3-氟-4-[[1-甲基-6-(1H-吡唑-4-基)-1H-吲唑-5-基]氧基]苯基]-1-(4-氟苯基)-1,2-二氢-6-甲基-2-氧代-3-吡啶甲酰胺二盐酸盐	Merestinib dihydrochloride	1206801-37-7	C30H24Cl2F2N6O3
N-[3-氟-4-[[1-甲基-6-(1H-吡唑-4-基)-1H-吲唑-5-基]氧基]苯基]-1-(4-氟苯基)-1,2-二氢-6-甲基-2-氧代-3-吡啶甲酰胺	merestinib	1206799-15-6	C₃₀H₂₂F₂N₆O₃
N-[3-[[5-环丙基-2-[[3-(4-吗啉基甲基)苯基]氨基]-4-嘧啶基]氨基]丙基]环丁烷甲酰胺	N-{3-[(5-Cyclopropyl-2-{[3-(Morpholin-4-Ylmethyl)phenyl]amino}pyrimidin-4-Yl)amino]propyl}cyclobutanecarboxamide	1190378-57-4	C₂₆H₃₆N₆O₂
N-[3-[6-[[4-(1,4-二甲基-3-氧代-2-哌嗪基)苯基]氨基]-4,5-二氢-4-甲基-5-氧代-2-吡嗪基]-2-甲基苯基]-4,5,6,7-四氢苯并[b]噻吩-2-甲酰胺	GDC-0834	1133432-46-8	C₃₃H₃₆N₆O₃S
N-[3-[1,4-二氢-1-甲基-7-[(6-甲基-3-吡啶基)氨基]-2-氧代嘧啶并[4,5-D]嘧啶-3(2H)-基]-4-甲基苯基]-3-(三氟甲基)苯甲酰胺	GNF-7	839706-07-9	C₂₈H₂₄F₃N₇O₂
N-[3-(2,4-二氯苯氧基)丙基]-N-甲基-2-丙炔胺盐酸盐	3-(2,4-dichlorophenoxy)-N-methyl-N-prop-2-ynylpropan-1-amine;hydron;chloride	17780-75-5	C13H16Cl3NO
N-[2-（苯甲酰氨基）-6-苯并噻唑基]三环[3.3.1.13,7]癸烷-1-甲酰胺	NVP-231	362003-83-6	C₂₅H₂₅N₃O₂S
N-[2-氯-5-（三氟甲基）苯基]-2-[4-（2-呋喃基）-1-哌嗪基]乙酰胺	N-(2-chloro-5-(trifluoromethyl)phenyl)-2-(4-(furan-2-carbonyl)piperazin-1-yl)acetamide	899713-86-1	C₁₈H₁₇ClF₃N₃O₃
N-[2-氟-5-[[3-[(1E)-2-(2-吡啶基)乙烯基]-1H-吲唑-6-基]氨基]苯基]-1,3-二甲基-1H-吡唑-5-甲酰胺	AG-013958	319460-94-1	C₂₆H₂₂FN₇O
N-[2-[[2-(二甲基氨基)乙基]甲基氨基]-5-[[4-(1H-吲哚-3-基)-2-嘧啶基]氨基]-4-甲氧基苯基]-2-丙烯酰胺	AZ5104	1421373-98-9	C₂₇H₃₁N₇O₂
N-[2-[[(2,3-二氟苯基)甲基]硫基]-6-[[(1S,2R)-2,3-二羟基-1-甲基丙基]氨基]-4-嘧啶基]-1-氮杂环丁烷磺酰胺	N-(2-[(2,3-difluorobenzyl)thio]-6-{[(1S,2R)-2,3-dihydroxy-1-methylpropyl]amino}pyrimidin-4-yl)azetidine-1-sulfonamide	1204707-73-2	C₁₈H₂₃F₂N₅O₄S₂
N-[2-[[((3R)-1-][反式-4-羟基-4-(6-甲氧基-3-吡啶基)环己基]-3-吡咯烷基]氨基]-2-氧代乙基]-3-(三氟甲基)-苯甲酰胺二甲磺酸盐	INCB 3284 dimesylate	887401-93-6	C28H39F3N4O10S2
N-[2-[2-(二甲基氨基)乙基]-2,3-二氢-1,3-二氧代-1H-苯[de]异喹啉-5-基]脲R	UNBS-5126	956590-23-1	C₁₇H₁₈N₄O₃
N-[2-[2-(4-氯苯基)-4-噻唑基]乙基]丁酰胺	azoramide	932986-18-0	C₁₅H₁₇ClN₂OS
N-[2-[(R)-(3-氯苯基)[(3R)-1-[[[(2S)-2-(甲基氨基)-3-[(3R)-四氢-2H-吡喃-3-基]丙基]氨基]羰基]-3-哌啶基]甲氧基]乙基]氨基甲酸甲酯，2,2,2-三氟乙酸盐	VTP-27999 2,2,2-trifluoroacetate	1013937-63-7	C28H42ClF3N4O7
N-[2-[(R)-(3-氯苯基)[(3R)-1-[[[(2S)-2-(甲基氨基)-3-[(3R)-四氢-2H-吡喃-3-基]丙基]氨基]羰基]-3-哌啶基]甲氧基]乙基]氨基甲酸甲酯	VTP-27999	942142-51-0	C₂₆H₄₁ClN₄O₅
N-[2-(4'-氰基联苯-4-基)丙基]-2-丙烷磺酰胺	LY 404187	211311-95-4	C₁₉H₂₂N₂O₂S
N-[2-(3-溴苯基)乙基]-2,4,6-三甲基-N-[[3'-(甲基磺酰基)[1,1'-联苯]-4-基]甲基]苯磺酰胺	SR9243	1613028-81-1	C₃₁H₃₂BrNO₄S₂
N-[2-(2-吡啶基)-6-(1,2,4,5-四氢-3H-3-苯并氮杂卓-3-基)-4-嘧啶基]-beta-丙氨酸	GSK-J1	1373422-53-7	C₂₂H₂₃N₅O₂
N-[2,4-二氟-3-[[5-(3-吡啶基)-1H-吡咯并[2,3-B]吡啶-3-基]羰基]苯基]-2-丙磺酰胺	propane-2-sulfonic acid [2,4-difluoro-3-(5-pyridin-3-yl-1H-pyrrolo[2,3-b]pyridine-3-carbonyl)-phenyl]-amide	918505-61-0	C₂₂H₁₈F₂N₄O₃S
N-[1-(1-氧丙基)-4-哌啶基]-N'-[4-(三氟甲氧基)苯基]脲	TPPU	1222780-33-7	C₁₆H₂₀F₃N₃O₃

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