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苯并硫平类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 9-fluoro-N-(2-phenoxyethyl)-3-propan-2-yl-5,6-dihydrobenzo[b][1]benzothiepine-2-sulfonamide —— C25H26FNO3S2
9-fluoro-N-(2-phenoxyethyl)-3-propan-2-yl-5,6-dihydrobenzo[b][1]benzothiepine-2-sulfonamide
—— N-(1-hydroxy-1-phenylpropan-2-yl)-3-methyl-5,6-dihydrobenzo[b][1]benzothiepine-2-sulfonamide —— C24H25NO3S2
N-(1-hydroxy-1-phenylpropan-2-yl)-3-methyl-5,6-dihydrobenzo[b][1]benzothiepine-2-sulfonamide
—— (4R)-5-[4-[[4-(4-aza-1-azoniabicyclo[2.2.2]octan-1-ylmethyl)phenyl]methoxy]phenyl]-3,3-dibutyl-7-(dimethylamino)-1,1-dioxo-4,5-dihydro-2H-1lambda6-benzothiepin-4-ol —— C40H56N3O4S+
(4R)-5-[4-[[4-(4-aza-1-azoniabicyclo[2.2.2]octan-1-ylmethyl)phenyl]methoxy]phenyl]-3,3-dibutyl-7-(dimethylamino)-1,1-dioxo-4,5-dihydro-2H-1lambda6-benzothiepin-4-ol
—— (5R)-7-(dimethylamino)-3,3-dimethyl-1,1-dioxo-5-phenyl-4,5-dihydro-2H-1lambda6-benzothiepin-4-ol;N-methylhexanamide —— C27H40N2O4S
(5R)-7-(dimethylamino)-3,3-dimethyl-1,1-dioxo-5-phenyl-4,5-dihydro-2H-1lambda6-benzothiepin-4-ol;N-methylhexanamide
—— (4R,5R)-5-[3-[2-[2-(4,4-dimethylpiperazin-4-ium-1-yl)ethoxy]ethoxy]phenyl]-3,3,7-trimethyl-1,1-dioxo-4,5-dihydro-2H-1lambda6-benzothiepin-4-ol;(4R,5R)-5-[4-[2-[2-(4,4-dimethylpiperazin-4-ium-1-yl)ethoxy]ethoxy]phenyl]-3,3,8-trimethyl-1,1-dioxo-4,5-dihydro-2H-1lambda6-benzothiepin-4-ol;2-[2-[3-[(4R,5R)-4-hydroxy-3,3,8-trimethyl-1,1-dioxo-4,5-dihydro-2H-1lambda6-benzothiepin-5-yl]phenoxy]ethoxy]ethyl-trimethylazanium;iodide —— C84H124IN5O15S3+2
(4R,5R)-5-[3-[2-[2-(4,4-dimethylpiperazin-4-ium-1-yl)ethoxy]ethoxy]phenyl]-3,3,7-trimethyl-1,1-dioxo-4,5-dihydro-2H-1lambda6-benzothiepin-4-ol;(4R,5R)-5-[4-[2-[2-(4,4-dimethylpiperazin-4-ium-1-yl)ethoxy]ethoxy]phenyl]-3,3,8-trimethyl-1,1-dioxo-4,5-dihydro-2H-1lambda6-benzothiepin-4-ol;2-[2-[3-[(4R,5R)-4-hydroxy-3,3,8-trimethyl-1,1-dioxo-4,5-dihydro-2H-1lambda6-benzothiepin-5-yl]phenoxy]ethoxy]ethyl-trimethylazanium;iodide
—— 8-bromo-N-[2-chloro-6-[difluoro-(4-fluorophenyl)methyl]pyrimidin-4-yl]-5-methyl-4,5-dihydro-3H-1-benzothiepin-2-imine —— C22H16BrClF3N3S
8-bromo-N-[2-chloro-6-[difluoro-(4-fluorophenyl)methyl]pyrimidin-4-yl]-5-methyl-4,5-dihydro-3H-1-benzothiepin-2-imine
—— N-cyclopentyl-3-methyl-5,6-dihydrobenzo[b][1]benzothiepine-2-sulfonamide —— C20H23NO2S2
N-cyclopentyl-3-methyl-5,6-dihydrobenzo[b][1]benzothiepine-2-sulfonamide
—— (5R)-3,3-dibutyl-5-(3,4-difluorophenyl)-8-methoxy-1,1-dioxo-4,5-dihydro-2H-1lambda6-benzothiepin-4-ol;(5R)-3,3-dibutyl-5-(4-fluoro-3-methoxyphenyl)-7-methyl-1,1-dioxo-4,5-dihydro-2H-1lambda6-benzothiepin-4-ol;ethane —— C53H73F3O8S2
(5R)-3,3-dibutyl-5-(3,4-difluorophenyl)-8-methoxy-1,1-dioxo-4,5-dihydro-2H-1lambda6-benzothiepin-4-ol;(5R)-3,3-dibutyl-5-(4-fluoro-3-methoxyphenyl)-7-methyl-1,1-dioxo-4,5-dihydro-2H-1lambda6-benzothiepin-4-ol;ethane
—— ethane;(4R,5R)-3,3,5-trimethyl-1,1-dioxo-4,5-dihydro-2H-1lambda6-benzothiepin-4-ol —— C15H24O3S
ethane;(4R,5R)-3,3,5-trimethyl-1,1-dioxo-4,5-dihydro-2H-1lambda6-benzothiepin-4-ol
—— Ethane;2-methyl-5,5-dioxo-4-phenyl-1,4,6,7-tetrahydro-[3]benzothiepino[5,4-b]pyridine-3-carboxylic acid —— C23H25NO4S
Ethane;2-methyl-5,5-dioxo-4-phenyl-1,4,6,7-tetrahydro-[3]benzothiepino[5,4-b]pyridine-3-carboxylic acid
—— 6H-benzo[b][1]benzothiepin-5-one;ethane —— C18H22OS
6H-benzo[b][1]benzothiepin-5-one;ethane
—— 3-(16-chloro-3,13-dithiatetracyclo[12.4.0.02,6.07,12]octadeca-1(14),2(6),4,7,9,11,15,17-octaen-4-yl)-N-[3-[(2R,3S,4R,5R,8R,10R,11R,12S,13S,14R)-2-ethyl-3,4,10,11,13-pentahydroxy-3,5,8,10,12,14-hexamethyl-15-oxo-1-oxa-6-azacyclopentadec-6-yl]propyl]prop-2-enamide —— C43H57ClN2O8S2
3-(16-chloro-3,13-dithiatetracyclo[12.4.0.02,6.07,12]octadeca-1(14),2(6),4,7,9,11,15,17-octaen-4-yl)-N-[3-[(2R,3S,4R,5R,8R,10R,11R,12S,13S,14R)-2-ethyl-3,4,10,11,13-pentahydroxy-3,5,8,10,12,14-hexamethyl-15-oxo-1-oxa-6-azacyclopentadec-6-yl]propyl]prop-2-enamide
—— N-[3-[(2R,3S,4R,5R,8R,10R,11R,12S,13S,14R)-2-ethyl-3,4,10,11,13-pentahydroxy-3,5,8,10,12,14-hexamethyl-15-oxo-1-oxa-6-azacyclopentadec-6-yl]propyl]-3-(16-methyl-3,13-dithiatetracyclo[12.4.0.02,6.07,12]octadeca-1(14),2(6),4,7,9,11,15,17-octaen-4-yl)prop-2-enamide —— C44H60N2O8S2
N-[3-[(2R,3S,4R,5R,8R,10R,11R,12S,13S,14R)-2-ethyl-3,4,10,11,13-pentahydroxy-3,5,8,10,12,14-hexamethyl-15-oxo-1-oxa-6-azacyclopentadec-6-yl]propyl]-3-(16-methyl-3,13-dithiatetracyclo[12.4.0.02,6.07,12]octadeca-1(14),2(6),4,7,9,11,15,17-octaen-4-yl)prop-2-enamide
—— (1S,1aR,7bR)-1,1a,2,7b-tetrahydrocyclopropa[c]thiochromene-1-carboxylic acid —— C11H10O2S
(1S,1aR,7bR)-1,1a,2,7b-tetrahydrocyclopropa[c]thiochromene-1-carboxylic acid
—— (4R,5R)-3,3-dibutyl-7-(dimethylamino)-5-[4-[4-(3-hydroxyphenyl)butoxy]phenyl]-1,1-dioxo-4,5-dihydro-2H-1lambda6-benzothiepin-4-ol;methylsulfonylmethane —— C38H55NO7S2
(4R,5R)-3,3-dibutyl-7-(dimethylamino)-5-[4-[4-(3-hydroxyphenyl)butoxy]phenyl]-1,1-dioxo-4,5-dihydro-2H-1lambda6-benzothiepin-4-ol;methylsulfonylmethane
—— 1-(8-Methoxy-2,3-dihydro-1-benzothiepin-5-yl)-2-(4-methoxyphenyl)hydrazine —— C18H20N2O2S
1-(8-Methoxy-2,3-dihydro-1-benzothiepin-5-yl)-2-(4-methoxyphenyl)hydrazine
—— (4S,5S)-7-(dimethylamino)-5-(4-hydroxyphenyl)-3,3-dimethyl-1,1-dioxo-4,5-dihydro-2H-1lambda6-benzothiepin-4-ol;7-(dimethylamino)-5-(4-methoxyphenyl)-3,3-dimethyl-1,1-dioxo-4,5-dihydro-2H-1lambda6-benzothiepin-4-ol —— C41H52N2O8S2
(4S,5S)-7-(dimethylamino)-5-(4-hydroxyphenyl)-3,3-dimethyl-1,1-dioxo-4,5-dihydro-2H-1lambda6-benzothiepin-4-ol;7-(dimethylamino)-5-(4-methoxyphenyl)-3,3-dimethyl-1,1-dioxo-4,5-dihydro-2H-1lambda6-benzothiepin-4-ol
—— 1-[3-[3-(Trifluoromethyl)-1,2,5,6-tetrahydrobenzo[b][1]benzothiepin-5-yl]propyl]piperidine —— C23H28F3NS
1-[3-[3-(Trifluoromethyl)-1,2,5,6-tetrahydrobenzo[b][1]benzothiepin-5-yl]propyl]piperidine
—— 4-[[6-benzyl-4-[(5,8-dimethyl-4,5-dihydro-3H-1-benzothiepin-2-ylidene)amino]-4,5-dihydropyrimidin-2-yl]amino]-3-methylbenzenesulfonamide —— C30H33N5O2S2
4-[[6-benzyl-4-[(5,8-dimethyl-4,5-dihydro-3H-1-benzothiepin-2-ylidene)amino]-4,5-dihydropyrimidin-2-yl]amino]-3-methylbenzenesulfonamide
—— N-[4-[(4-hydroxy-2-oxo-3H-1,3-oxazol-5-yl)methyl]phenyl]-8-methyl-9-oxo-5,6-dihydrothiepino[4,5-f][1,3]benzodioxole-6-carboxamide —— C23H20N2O7S
N-[4-[(4-hydroxy-2-oxo-3H-1,3-oxazol-5-yl)methyl]phenyl]-8-methyl-9-oxo-5,6-dihydrothiepino[4,5-f][1,3]benzodioxole-6-carboxamide
—— ethane;(4S,5S)-5-[4-[[4-(hydroxymethyl)phenyl]methoxy]phenyl]-3,3-dimethyl-1,1-dioxo-4,5-dihydro-2H-1lambda6-benzothiepin-4-ol —— C28H34O5S
ethane;(4S,5S)-5-[4-[[4-(hydroxymethyl)phenyl]methoxy]phenyl]-3,3-dimethyl-1,1-dioxo-4,5-dihydro-2H-1lambda6-benzothiepin-4-ol
—— N,N-dimethyl-2-(13-thia-3,4-diazatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),2(6),4,7,9,11,14,16-octaen-3-ylmethoxy)ethanamine —— C20H21N3OS
N,N-dimethyl-2-(13-thia-3,4-diazatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),2(6),4,7,9,11,14,16-octaen-3-ylmethoxy)ethanamine
—— 9-fluoro-3-propan-2-yl-N-(2-pyridin-2-ylethyl)-5,6-dihydrobenzo[b][1]benzothiepine-2-sulfonamide —— C24H25FN2O2S2
9-fluoro-3-propan-2-yl-N-(2-pyridin-2-ylethyl)-5,6-dihydrobenzo[b][1]benzothiepine-2-sulfonamide
—— 8-bromo-5-methyl-N-(2-methylsulfonylpyrimidin-4-yl)-4,5-dihydro-3H-1-benzothiepin-2-imine —— C16H16BrN3O2S2
8-bromo-5-methyl-N-(2-methylsulfonylpyrimidin-4-yl)-4,5-dihydro-3H-1-benzothiepin-2-imine
—— (4R,5R)-5-[4-[3-(4-aza-1-azoniabicyclo[2.2.2]octan-1-yl)propoxy]phenyl]-3,3-dibutyl-7-(dimethylamino)-1,1-dioxo-4,5-dihydro-2H-1lambda6-benzothiepin-4-ol;1,4-xylene —— C43H64N3O4S+
(4R,5R)-5-[4-[3-(4-aza-1-azoniabicyclo[2.2.2]octan-1-yl)propoxy]phenyl]-3,3-dibutyl-7-(dimethylamino)-1,1-dioxo-4,5-dihydro-2H-1lambda6-benzothiepin-4-ol;1,4-xylene
—— Methyl 3-[[4-[[7-(4-methylphenyl)-1,1-dioxo-2,3-dihydro-1lambda6-benzothiepine-4-carbonyl]amino]phenyl]methylamino]propanoate —— C29H30N2O5S
Methyl 3-[[4-[[7-(4-methylphenyl)-1,1-dioxo-2,3-dihydro-1lambda6-benzothiepine-4-carbonyl]amino]phenyl]methylamino]propanoate
—— (6R,8S)-N-[4-[(4-hydroxy-2-oxo-3H-1,3-oxazol-5-yl)methyl]phenyl]-8-methyl-9-oxo-5,6-dihydrothiepino[4,5-f][1,3]benzodioxole-6-carboxamide —— C23H20N2O7S
(6R,8S)-N-[4-[(4-hydroxy-2-oxo-3H-1,3-oxazol-5-yl)methyl]phenyl]-8-methyl-9-oxo-5,6-dihydrothiepino[4,5-f][1,3]benzodioxole-6-carboxamide
—— 9-fluoro-3-propan-2-yl-N-(2-pyridin-4-ylethyl)-5,6-dihydrobenzo[b][1]benzothiepine-2-sulfonamide —— C24H25FN2O2S2
9-fluoro-3-propan-2-yl-N-(2-pyridin-4-ylethyl)-5,6-dihydrobenzo[b][1]benzothiepine-2-sulfonamide
—— N-[4-[(4-hydroxy-2-oxo-3H-1,3-thiazol-5-yl)methyl]phenyl]-8-methyl-9-oxo-5,6-dihydrothiepino[4,5-f][1,3]benzodioxole-6-carboxamide —— C23H20N2O6S2
N-[4-[(4-hydroxy-2-oxo-3H-1,3-thiazol-5-yl)methyl]phenyl]-8-methyl-9-oxo-5,6-dihydrothiepino[4,5-f][1,3]benzodioxole-6-carboxamide
—— 5-Ethyl-2-(4-fluorophenyl)-4-thiophen-2-yl-2,3-dihydro-1-benzothiepine —— C22H19FS2
5-Ethyl-2-(4-fluorophenyl)-4-thiophen-2-yl-2,3-dihydro-1-benzothiepine
—— 3,3-dimethyl-5-phenyl-2H-1lambda4-benzothiepine 1-oxide;ethane;prop-1-yne —— C23H28OS
3,3-dimethyl-5-phenyl-2H-1lambda4-benzothiepine 1-oxide;ethane;prop-1-yne
—— 9-fluoro-N-[2-(oxan-4-yl)ethyl]-3-propan-2-yl-5,6-dihydrobenzo[b][1]benzothiepine-2-sulfonamide —— C24H30FNO3S2
9-fluoro-N-[2-(oxan-4-yl)ethyl]-3-propan-2-yl-5,6-dihydrobenzo[b][1]benzothiepine-2-sulfonamide
—— N-[3-(7H-benzo[c][1]benzothiepin-11-ylidenemethyl)phenyl]methanesulfonamide —— C22H19NO2S2
N-[3-(7H-benzo[c][1]benzothiepin-11-ylidenemethyl)phenyl]methanesulfonamide
—— N-[2-(2-fluorophenyl)ethyl]-3-methyl-5,6-dihydrobenzo[b][1]benzothiepine-2-sulfonamide —— C23H22FNO2S2
N-[2-(2-fluorophenyl)ethyl]-3-methyl-5,6-dihydrobenzo[b][1]benzothiepine-2-sulfonamide
—— Ethane;methyl 2-methyl-5,5-dioxo-4-phenyl-1,4,6,7-tetrahydro-[3]benzothiepino[5,4-b]pyridine-3-carboxylate —— C24H27NO4S
Ethane;methyl 2-methyl-5,5-dioxo-4-phenyl-1,4,6,7-tetrahydro-[3]benzothiepino[5,4-b]pyridine-3-carboxylate
—— 3-(3,13-dithiatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),2(6),4,7,9,11,14,16-octaen-4-yl)-N-[3-[(2R,3S,4R,5R,8R,10R,11R,12S,13S,14R)-2-ethyl-3,4,10,11,13-pentahydroxy-3,5,8,10,12,14-hexamethyl-15-oxo-1-oxa-6-azacyclopentadec-6-yl]propyl]prop-2-enamide —— C43H58N2O8S2
3-(3,13-dithiatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),2(6),4,7,9,11,14,16-octaen-4-yl)-N-[3-[(2R,3S,4R,5R,8R,10R,11R,12S,13S,14R)-2-ethyl-3,4,10,11,13-pentahydroxy-3,5,8,10,12,14-hexamethyl-15-oxo-1-oxa-6-azacyclopentadec-6-yl]propyl]prop-2-enamide
—— 3-fluoro-4H-benzo[b][1]benzothiepin-6-one —— C14H9FOS
3-fluoro-4H-benzo[b][1]benzothiepin-6-one
—— Ethane;2,2,3,3,5-pentamethyl-1-benzothiepine —— C17H26S
Ethane;2,2,3,3,5-pentamethyl-1-benzothiepine
—— 3-methyl-N-(3-morpholin-4-ylpropyl)-5,6-dihydrobenzo[b][1]benzothiepine-2-sulfonamide —— C22H28N2O3S2
3-methyl-N-(3-morpholin-4-ylpropyl)-5,6-dihydrobenzo[b][1]benzothiepine-2-sulfonamide
—— 3-methyl-N-(2-morpholin-4-ylethyl)-5,6-dihydrobenzo[b][1]benzothiepine-2-sulfonamide —— C21H26N2O3S2
3-methyl-N-(2-morpholin-4-ylethyl)-5,6-dihydrobenzo[b][1]benzothiepine-2-sulfonamide
—— 2-[3-(Dimethylsulfamoylamino)propylamino]-4,5-dihydro-[1]benzothiepino[5,4-d][1,3]thiazole;ethane —— C18H28N4O2S3
2-[3-(Dimethylsulfamoylamino)propylamino]-4,5-dihydro-[1]benzothiepino[5,4-d][1,3]thiazole;ethane
—— 4-[[[4-benzyl-6-[[8-(2-hydroxyethyl)-5-methyl-4,5-dihydro-3H-1-benzothiepin-2-ylidene]amino]pyrimidin-2-yl]amino]methyl]cyclohexan-1-ol —— C31H38N4O2S
4-[[[4-benzyl-6-[[8-(2-hydroxyethyl)-5-methyl-4,5-dihydro-3H-1-benzothiepin-2-ylidene]amino]pyrimidin-2-yl]amino]methyl]cyclohexan-1-ol
—— Ethane;methanamine;1,2,3,4-tetrahydrocyclopenta[c][1]benzothiepin-10-one —— C16H23NOS
Ethane;methanamine;1,2,3,4-tetrahydrocyclopenta[c][1]benzothiepin-10-one
—— 6-(5-Ethyloctyl)-3-(trifluoromethyl)-5,6-dihydrobenzo[b][1]benzothiepine —— C25H31F3S
6-(5-Ethyloctyl)-3-(trifluoromethyl)-5,6-dihydrobenzo[b][1]benzothiepine
—— 9-fluoro-N-(2-morpholin-4-ylethyl)-3-propan-2-yl-5,6-dihydrobenzo[b][1]benzothiepine-2-sulfonamide —— C23H29FN2O3S2
9-fluoro-N-(2-morpholin-4-ylethyl)-3-propan-2-yl-5,6-dihydrobenzo[b][1]benzothiepine-2-sulfonamide
—— (8S)-6-[aminooxy-[4-(phosphorosomethyl)phenyl]methyl]-8-methyl-5,6-dihydrothiepino[4,5-f][1,3]benzodioxol-9-one;dimethoxymethane —— C23H28NO7PS
(8S)-6-[aminooxy-[4-(phosphorosomethyl)phenyl]methyl]-8-methyl-5,6-dihydrothiepino[4,5-f][1,3]benzodioxol-9-one;dimethoxymethane
—— 6-hydroxy-N-[4-[(4-hydroxy-2-oxo-3H-1,3-thiazol-5-yl)methyl]phenyl]-8-methoxy-5-oxo-1,2-dihydro-3-benzothiepine-2-carboxamide —— C22H20N2O6S2
6-hydroxy-N-[4-[(4-hydroxy-2-oxo-3H-1,3-thiazol-5-yl)methyl]phenyl]-8-methoxy-5-oxo-1,2-dihydro-3-benzothiepine-2-carboxamide
—— (1S,1aR)-1,1a,2,7b-tetrahydrocyclopropa[c]thiochromene-1-carboxylic acid —— C11H10O2S
(1S,1aR)-1,1a,2,7b-tetrahydrocyclopropa[c]thiochromene-1-carboxylic acid
—— (3S)-3-butyl-3-ethyl-4-methyl-5-phenylsulfanyl-4,5-dihydro-2H-1lambda6-benzothiepine 1,1-dioxide —— C23H30O2S2
(3S)-3-butyl-3-ethyl-4-methyl-5-phenylsulfanyl-4,5-dihydro-2H-1lambda6-benzothiepine 1,1-dioxide
—— tert-butyl 3-[2-(6,11-dihydro-3H-benzo[c][1]benzothiepin-4-ylidene)piperidin-1-yl]-3-oxopropanoate —— C26H31NO3S
tert-butyl 3-[2-(6,11-dihydro-3H-benzo[c][1]benzothiepin-4-ylidene)piperidin-1-yl]-3-oxopropanoate