| 中文名称 | 英文名称 | CAS号 | 化学式 |
|---|---|---|---|
| —— | 5-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-([1,2,4]triazolo[4,3-b]pyridazin-6-yl)-1H-pyrazol-3-one | —— | C20H23N9O |
| —— | 5-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl)-1H-pyrazol-3-one | —— | C21H25N9O |
| —— | 5-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-4-methylpyrimidin-5-yl]-2-(3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl)-1H-pyrazol-3-one | —— | C21H25N9O |
| —— | 4-(6-methoxy-[1,2,4]triazolo[4,3-b]pyridazin-3-yl)-N-[[(2R)-oxolan-2-yl]methyl]butanamide | —— | C15H21N5O3 |
| —— | N-[(3S)-1,1-dioxothiolan-3-yl]-3-(6-propan-2-yloxy-[1,2,4]triazolo[4,3-b]pyridazin-3-yl)propanamide | —— | C15H21N5O4S |
| —— | N-[(3R)-1,1-dioxothiolan-3-yl]-3-(6-propan-2-yloxy-[1,2,4]triazolo[4,3-b]pyridazin-3-yl)propanamide | —— | C15H21N5O4S |
| —— | 3-(6-methoxy-[1,2,4]triazolo[4,3-b]pyridazin-3-yl)-N-[(2S)-4-phenylbutan-2-yl]propanamide | —— | C19H23N5O2 |
| —— | N-[(4S)-2,2-dimethyloxan-4-yl]-4-(6-methoxy-[1,2,4]triazolo[4,3-b]pyridazin-3-yl)butanamide | —— | C17H25N5O3 |
| —— | N-[(3R)-1,1-dioxothiolan-3-yl]-3-(6-methoxy-[1,2,4]triazolo[4,3-b]pyridazin-3-yl)propanamide | —— | C13H17N5O4S |
| —— | 4-(6-methoxy-[1,2,4]triazolo[4,3-b]pyridazin-3-yl)-N-[[(2S)-oxolan-2-yl]methyl]butanamide | —— | C15H21N5O3 |
| —— | N-[(4R)-2,2-dimethyloxan-4-yl]-4-(6-methoxy-[1,2,4]triazolo[4,3-b]pyridazin-3-yl)butanamide | —— | C17H25N5O3 |
| —— | N-[(3S)-1,1-dioxothiolan-3-yl]-3-(6-methoxy-[1,2,4]triazolo[4,3-b]pyridazin-3-yl)propanamide | —— | C13H17N5O4S |
| —— | N-[(1R)-1-(5-methyl-1,2,4-oxadiazol-3-yl)propyl]-1-[3-(trifluoromethyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidine-4-carboxamide | —— | C18H21F3N8O2 |
| —— | N-[(1S)-1-(5-methyl-1,2,4-oxadiazol-3-yl)propyl]-1-[3-(trifluoromethyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidine-4-carboxamide | —— | C18H21F3N8O2 |
| —— | (2S)-2-methyl-3-[[3-(trifluoromethyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]amino]propanenitrile | —— | C10H9F3N6 |
| —— | (2R)-2-methyl-3-[[3-(trifluoromethyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]amino]propanenitrile | —— | C10H9F3N6 |
| —— | N-[(1S)-1-(2-ethoxyphenyl)-3-methylbutyl]-3-(trifluoromethyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-amine | —— | C19H22F3N5O |
| —— | N-[(1R)-1-(2-ethoxyphenyl)-3-methylbutyl]-3-(trifluoromethyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-amine | —— | C19H22F3N5O |
| —— | N-[(2R)-2-[(2,5-difluorophenyl)methyl]-3-hydroxypropyl]-1-([1,2,4]triazolo[4,3-b]pyridazin-6-yl)piperidine-4-carboxamide | —— | C21H24F2N6O2 |
| —— | N-[(2S)-2-[(2,5-difluorophenyl)methyl]-3-hydroxypropyl]-1-([1,2,4]triazolo[4,3-b]pyridazin-6-yl)piperidine-4-carboxamide | —— | C21H24F2N6O2 |
| —— | N-(4-methylcyclohexyl)-N-[[(2R)-oxolan-2-yl]methyl]-3-(trifluoromethyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-amine | —— | C18H24F3N5O |
| —— | 3-methyl-N-[(2R)-2-morpholin-4-yl-2-thiophen-2-ylethyl]-[1,2,4]triazolo[4,3-b]pyridazin-6-amine | —— | C16H20N6OS |
| —— | 3-methyl-N-[(2S)-2-morpholin-4-yl-2-thiophen-2-ylethyl]-[1,2,4]triazolo[4,3-b]pyridazin-6-amine | —— | C16H20N6OS |
| —— | (5R)-3-methyl-7-[2-([1,2,4]triazolo[4,3-b]pyridazin-6-yloxy)acetyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one | —— | C14H16N6O4 |
| —— | (5S)-3-methyl-7-[2-([1,2,4]triazolo[4,3-b]pyridazin-6-yloxy)acetyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one | —— | C14H16N6O4 |
| —— | [(2S)-2-(6-methyl-1H-benzimidazol-2-yl)pyrrolidin-1-yl]-[1-[3-(trifluoromethyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidin-4-yl]methanone | —— | C24H25F3N8O |
| —— | [(2R)-2-(6-methyl-1H-benzimidazol-2-yl)pyrrolidin-1-yl]-[1-[3-(trifluoromethyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidin-4-yl]methanone | —— | C24H25F3N8O |
| —— | N-methyl-N-[(1R)-1-pyridin-3-ylethyl]-1-[3-(trifluoromethyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidine-4-carboxamide | —— | C20H22F3N7O |
| —— | N-[(1S)-1-(1-ethylbenzimidazol-2-yl)ethyl]-1-[3-(trifluoromethyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidine-4-carboxamide | —— | C23H25F3N8O |
| —— | N-[(1R)-1-(1-ethylbenzimidazol-2-yl)ethyl]-1-[3-(trifluoromethyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidine-4-carboxamide | —— | C23H25F3N8O |
| —— | N-methyl-N-[(1S)-1-pyridin-3-ylethyl]-1-[3-(trifluoromethyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidine-4-carboxamide | —— | C20H22F3N7O |
| —— | N-[(2S)-2-(4-methylpiperidin-1-yl)-2-phenylethyl]-1-([1,2,4]triazolo[4,3-b]pyridazin-6-yl)piperidine-4-carboxamide | —— | C25H33N7O |
| —— | N-[(2R)-2-(4-methylpiperidin-1-yl)-2-phenylethyl]-1-([1,2,4]triazolo[4,3-b]pyridazin-6-yl)piperidine-4-carboxamide | —— | C25H33N7O |
| —— | N-[(2S)-4-(4-propan-2-yloxyphenyl)butan-2-yl]-3-(trifluoromethyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-amine | —— | C19H22F3N5O |
| —— | N-[(2R)-4-(4-propan-2-yloxyphenyl)butan-2-yl]-3-(trifluoromethyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-amine | —— | C19H22F3N5O |
| —— | N-[(1R)-1-(4-chlorophenyl)-4-methylpentyl]-1-([1,2,4]triazolo[4,3-b]pyridazin-6-yl)piperidine-4-carboxamide | —— | C23H29ClN6O |
| —— | N-[(1S)-1-(4-chlorophenyl)-4-methylpentyl]-1-([1,2,4]triazolo[4,3-b]pyridazin-6-yl)piperidine-4-carboxamide | —— | C23H29ClN6O |
| —— | N-[(R)-cyclopentyl(phenyl)methyl]-1-([1,2,4]triazolo[4,3-b]pyridazin-6-yl)piperidine-4-carboxamide | —— | C23H28N6O |
| —— | N-[(S)-cyclopentyl(phenyl)methyl]-1-([1,2,4]triazolo[4,3-b]pyridazin-6-yl)piperidine-4-carboxamide | —— | C23H28N6O |
| —— | N-[(1S)-2-(2-fluorophenoxy)-1-phenylethyl]-1-([1,2,4]triazolo[4,3-b]pyridazin-6-yl)piperidine-4-carboxamide | —— | C25H25FN6O2 |
| —— | N-[(1R)-2-(2-fluorophenoxy)-1-phenylethyl]-1-([1,2,4]triazolo[4,3-b]pyridazin-6-yl)piperidine-4-carboxamide | —— | C25H25FN6O2 |
| —— | N-[[3-[[(2R)-2-methylbutanoyl]amino]phenyl]methyl]-1-([1,2,4]triazolo[4,3-b]pyridazin-6-yl)piperidine-4-carboxamide | —— | C23H29N7O2 |
| —— | N-[[3-[[(2S)-2-methylbutanoyl]amino]phenyl]methyl]-1-([1,2,4]triazolo[4,3-b]pyridazin-6-yl)piperidine-4-carboxamide | —— | C23H29N7O2 |
| —— | (1S,2R)-1-N,1-N-dimethyl-2-N-[3-(trifluoromethyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]cyclopentane-1,2-diamine | —— | C13H17F3N6 |
| —— | (1R,2S)-1-N,1-N-dimethyl-2-N-[3-(trifluoromethyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]cyclopentane-1,2-diamine | —— | C13H17F3N6 |
| —— | (1R,2R)-1-N,1-N-dimethyl-2-N-[3-(trifluoromethyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]cyclopentane-1,2-diamine | —— | C13H17F3N6 |
| —— | 6-[(2R,4R)-2,4-dimethylpiperidin-1-yl]-3-(trifluoromethyl)-[1,2,4]triazolo[4,3-b]pyridazine | —— | C13H16F3N5 |
| —— | 6-[(2R,4S)-2,4-dimethylpiperidin-1-yl]-3-(trifluoromethyl)-[1,2,4]triazolo[4,3-b]pyridazine | —— | C13H16F3N5 |
| —— | (7R)-7-methyl-1-[3-(trifluoromethyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]-1,4-diazepan-5-one | —— | C12H13F3N6O |
| —— | (7S)-7-methyl-1-[3-(trifluoromethyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]-1,4-diazepan-5-one | —— | C12H13F3N6O |