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噻烯杂卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (7R)-7-(3,5-difluorophenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene —— C20H18F2N2S
(7R)-7-(3,5-difluorophenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene
—— (7R)-7-(4-ethoxyphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene —— C22H24N2OS
(7R)-7-(4-ethoxyphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene
—— (7S)-7-(4-ethoxyphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene —— C22H24N2OS
(7S)-7-(4-ethoxyphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene
—— (7S)-7-(3-ethoxyphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene —— C22H24N2OS
(7S)-7-(3-ethoxyphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene
—— (7R)-7-(3-fluorophenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene —— C20H19FN2S
(7R)-7-(3-fluorophenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene
—— (7S)-N-cyclohexyl-9-oxo-8-[[(2S)-oxolan-2-yl]methyl]-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-7-carboxamide —— C26H33N3O3S
(7S)-N-cyclohexyl-9-oxo-8-[[(2S)-oxolan-2-yl]methyl]-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-7-carboxamide
—— (7R)-N-cyclohexyl-9-oxo-8-[[(2R)-oxolan-2-yl]methyl]-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-7-carboxamide —— C26H33N3O3S
(7R)-N-cyclohexyl-9-oxo-8-[[(2R)-oxolan-2-yl]methyl]-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-7-carboxamide
—— 2-[5-(2-chlorophenyl)-2-oxo-6,7,8,9-tetrahydro-3H-[1]benzothiolo[2,3-e][1,4]diazepin-1-yl]-N-(4-fluorophenyl)acetamide —— C25H21ClFN3O2S
2-[5-(2-chlorophenyl)-2-oxo-6,7,8,9-tetrahydro-3H-[1]benzothiolo[2,3-e][1,4]diazepin-1-yl]-N-(4-fluorophenyl)acetamide
—— 5-(3,4-dimethoxyphenyl)-1-[(4-fluorophenyl)methyl]-6,7-dimethyl-3H-thieno[2,3-e][1,4]diazepin-2-one —— C24H23FN2O3S
5-(3,4-dimethoxyphenyl)-1-[(4-fluorophenyl)methyl]-6,7-dimethyl-3H-thieno[2,3-e][1,4]diazepin-2-one
—— 6,7-dimethyl-5-(2-methylphenyl)-1-(2-morpholin-4-ylethyl)-3H-thieno[2,3-e][1,4]diazepin-2-one —— C22H27N3O2S
6,7-dimethyl-5-(2-methylphenyl)-1-(2-morpholin-4-ylethyl)-3H-thieno[2,3-e][1,4]diazepin-2-one
—— 1-[(4-fluorophenyl)methyl]-5-thiophen-2-yl-6,7,8,9-tetrahydro-3H-[1]benzothiolo[2,3-e][1,4]diazepin-2-one —— C22H19FN2OS2
1-[(4-fluorophenyl)methyl]-5-thiophen-2-yl-6,7,8,9-tetrahydro-3H-[1]benzothiolo[2,3-e][1,4]diazepin-2-one
—— 2-[5-(3,4-dimethoxyphenyl)-6,7-dimethyl-2-oxo-3H-thieno[2,3-e][1,4]diazepin-1-yl]-N-(furan-2-ylmethyl)acetamide —— C24H25N3O5S
2-[5-(3,4-dimethoxyphenyl)-6,7-dimethyl-2-oxo-3H-thieno[2,3-e][1,4]diazepin-1-yl]-N-(furan-2-ylmethyl)acetamide
—— 6,7-dimethyl-1-(2-morpholin-4-ylethyl)-5-thiophen-2-yl-3H-thieno[2,3-e][1,4]diazepin-2-one —— C19H23N3O2S2
6,7-dimethyl-1-(2-morpholin-4-ylethyl)-5-thiophen-2-yl-3H-thieno[2,3-e][1,4]diazepin-2-one
—— 1-[2-(azepan-1-yl)-2-oxoethyl]-5-thiophen-2-yl-6,7,8,9-tetrahydro-3H-[1]benzothiolo[2,3-e][1,4]diazepin-2-one —— C23H27N3O2S2
1-[2-(azepan-1-yl)-2-oxoethyl]-5-thiophen-2-yl-6,7,8,9-tetrahydro-3H-[1]benzothiolo[2,3-e][1,4]diazepin-2-one
—— 6,7-dimethyl-1-(2-morpholin-4-ylethyl)-5-phenyl-3H-thieno[2,3-e][1,4]diazepin-2-one —— C21H25N3O2S
6,7-dimethyl-1-(2-morpholin-4-ylethyl)-5-phenyl-3H-thieno[2,3-e][1,4]diazepin-2-one
—— 2-[6,7-dimethyl-5-(3-methylphenyl)-2-oxo-3H-thieno[2,3-e][1,4]diazepin-1-yl]-N-(thiophen-2-ylmethyl)acetamide —— C23H23N3O2S2
2-[6,7-dimethyl-5-(3-methylphenyl)-2-oxo-3H-thieno[2,3-e][1,4]diazepin-1-yl]-N-(thiophen-2-ylmethyl)acetamide
—— 6,7-dimethyl-1-(2-oxo-2-pyrrolidin-1-ylethyl)-5-thiophen-2-yl-3H-thieno[2,3-e][1,4]diazepin-2-one —— C19H21N3O2S2
6,7-dimethyl-1-(2-oxo-2-pyrrolidin-1-ylethyl)-5-thiophen-2-yl-3H-thieno[2,3-e][1,4]diazepin-2-one
—— 2-[6,7-dimethyl-2-oxo-5-(3,4,5-trimethoxyphenyl)-3H-thieno[2,3-e][1,4]diazepin-1-yl]-N-(4-methylphenyl)acetamide —— C27H29N3O5S
2-[6,7-dimethyl-2-oxo-5-(3,4,5-trimethoxyphenyl)-3H-thieno[2,3-e][1,4]diazepin-1-yl]-N-(4-methylphenyl)acetamide
—— 2-[5-(3-chlorophenyl)-6,7-dimethyl-2-oxo-3H-thieno[2,3-e][1,4]diazepin-1-yl]-N-cyclohexylacetamide —— C23H26ClN3O2S
2-[5-(3-chlorophenyl)-6,7-dimethyl-2-oxo-3H-thieno[2,3-e][1,4]diazepin-1-yl]-N-cyclohexylacetamide
—— (7S)-N-(2,3-dimethylphenyl)-7-(3-fluorophenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C29H28FN3OS
(7S)-N-(2,3-dimethylphenyl)-7-(3-fluorophenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7R)-N-(3,4-dimethylphenyl)-7-(3-fluorophenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C29H28FN3OS
(7R)-N-(3,4-dimethylphenyl)-7-(3-fluorophenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7S)-N-(2,4-dimethylphenyl)-7-(4-ethoxyphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C31H33N3O2S
(7S)-N-(2,4-dimethylphenyl)-7-(4-ethoxyphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7R)-N-(3,5-dimethylphenyl)-7-(3-fluorophenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C29H28FN3OS
(7R)-N-(3,5-dimethylphenyl)-7-(3-fluorophenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7R)-N-(2,3-dimethylphenyl)-7-(3-fluorophenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C29H28FN3OS
(7R)-N-(2,3-dimethylphenyl)-7-(3-fluorophenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7S)-N-cyclopentyl-7-(4-ethylphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C28H33N3OS
(7S)-N-cyclopentyl-7-(4-ethylphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7S)-N-(2,3-dimethylphenyl)-7-(3-ethoxyphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C31H33N3O2S
(7S)-N-(2,3-dimethylphenyl)-7-(3-ethoxyphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7R)-7-(4-methylphenyl)-N-(2-phenylethyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C30H31N3OS
(7R)-7-(4-methylphenyl)-N-(2-phenylethyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7R)-N-(3,4-dimethylphenyl)-7-(4-methylphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C30H31N3OS
(7R)-N-(3,4-dimethylphenyl)-7-(4-methylphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7R)-N-(2,5-dimethylphenyl)-7-(3-fluorophenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C29H28FN3OS
(7R)-N-(2,5-dimethylphenyl)-7-(3-fluorophenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7R)-N-benzyl-7-(4-ethylphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C30H31N3OS
(7R)-N-benzyl-7-(4-ethylphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7R)-N-(2,3-dimethylphenyl)-7-(3-ethoxyphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C31H33N3O2S
(7R)-N-(2,3-dimethylphenyl)-7-(3-ethoxyphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7S)-7-(4-methylphenyl)-N-(2-phenylethyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C30H31N3OS
(7S)-7-(4-methylphenyl)-N-(2-phenylethyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7R)-7-(4-ethoxyphenyl)-N-[(4-methylphenyl)methyl]-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C31H33N3O2S
(7R)-7-(4-ethoxyphenyl)-N-[(4-methylphenyl)methyl]-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7S)-7-(4-methylphenyl)-N-[(4-methylphenyl)methyl]-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C30H31N3OS
(7S)-7-(4-methylphenyl)-N-[(4-methylphenyl)methyl]-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7S)-N-(2,5-dimethylphenyl)-7-(4-methylphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C30H31N3OS
(7S)-N-(2,5-dimethylphenyl)-7-(4-methylphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7R)-7-(4-methylsulfanylphenyl)-N-(2-phenylethyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C30H31N3OS2
(7R)-7-(4-methylsulfanylphenyl)-N-(2-phenylethyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7R)-7-(4-methylphenyl)-N-[(4-methylphenyl)methyl]-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C30H31N3OS
(7R)-7-(4-methylphenyl)-N-[(4-methylphenyl)methyl]-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7S)-N-[(4-fluorophenyl)methyl]-7-(4-methylsulfanylphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C29H28FN3OS2
(7S)-N-[(4-fluorophenyl)methyl]-7-(4-methylsulfanylphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7S)-7-(4-methylsulfanylphenyl)-N-(2-phenylethyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C30H31N3OS2
(7S)-7-(4-methylsulfanylphenyl)-N-(2-phenylethyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7S)-7-(4-ethoxyphenyl)-N-[(4-methylphenyl)methyl]-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C31H33N3O2S
(7S)-7-(4-ethoxyphenyl)-N-[(4-methylphenyl)methyl]-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7R)-N-(2,4-dimethylphenyl)-7-(3-fluorophenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C29H28FN3OS
(7R)-N-(2,4-dimethylphenyl)-7-(3-fluorophenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7R)-N-[(4-fluorophenyl)methyl]-7-(4-methylsulfanylphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C29H28FN3OS2
(7R)-N-[(4-fluorophenyl)methyl]-7-(4-methylsulfanylphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7R)-N-(2,4-dimethylphenyl)-7-(4-ethoxyphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C31H33N3O2S
(7R)-N-(2,4-dimethylphenyl)-7-(4-ethoxyphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7R)-N-(2,3-dimethylphenyl)-7-(4-methylphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C30H31N3OS
(7R)-N-(2,3-dimethylphenyl)-7-(4-methylphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7S)-N-benzyl-7-(4-ethylphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C30H31N3OS
(7S)-N-benzyl-7-(4-ethylphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7R)-N-(2,5-dimethylphenyl)-7-(4-ethoxyphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C31H33N3O2S
(7R)-N-(2,5-dimethylphenyl)-7-(4-ethoxyphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7S)-N-(2,3-dimethylphenyl)-7-(4-methylphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C30H31N3OS
(7S)-N-(2,3-dimethylphenyl)-7-(4-methylphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7R)-N-(3-fluoro-4-methylphenyl)-7-(4-methylphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C29H28FN3OS
(7R)-N-(3-fluoro-4-methylphenyl)-7-(4-methylphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7S)-N-(3,4-dimethylphenyl)-7-(4-ethoxyphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C31H33N3O2S
(7S)-N-(3,4-dimethylphenyl)-7-(4-ethoxyphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7S)-N-(3,5-dimethylphenyl)-7-(4-fluorophenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C29H28FN3OS
(7S)-N-(3,5-dimethylphenyl)-7-(4-fluorophenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide