| 中文名称 | 英文名称 | CAS号 | 化学式 |
|---|---|---|---|
| —— | (2R)-2-[5-[(3aS,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]-N-(3-pyrrolidin-1-ylphenyl)pentanamide | —— | C25H37N5O3S |
| —— | (2R)-5-[2-[5-[(3aS,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]ethylamino]-2-[[4-[(2,4-diaminopteridin-6-yl)methyl-methylamino]benzoyl]amino]-5-oxopentanoic acid | —— | C32H42N12O6S |
| —— | (2S)-6-[5-[(3aS,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]-2-[[5-(dimethylamino)naphthalen-1-yl]sulfonylamino]-N-(2-methoxysulfonothioylethyl)hexanamide | —— | C31H46N6O7S4 |
| —— | (2R)-6-[5-[(3aS,4R,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]-2-[[5-(dimethylamino)naphthalen-1-yl]sulfonylamino]-N-(2-methoxysulfonothioylethyl)hexanamide | —— | C31H46N6O7S4 |
| —— | [10-[5-[5-[(3aS,4R,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]pentylamino]-10-oxodecyl]-ethoxyphosphinic acid | —— | C27H51N4O6PS |
| —— | [10-[5-[5-[(3aS,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]pentylamino]-10-oxodecyl]-ethoxyphosphinic acid | —— | C27H51N4O6PS |
| —— | (2S)-6-[5-[(3aS,4R,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]-2-[[5-(dimethylamino)naphthalen-1-yl]sulfonylamino]-N-(2-methoxysulfonothioylethyl)hexanamide | —— | C31H46N6O7S4 |
| —— | (2R)-6-[6-[5-[(3aS,4R,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]hexanoylamino]-2-amino-N-(2-methoxysulfonothioylethyl)hexanamide | —— | C25H46N6O6S3 |
| —— | (2S)-5-[2-[5-[(3aS,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]ethylamino]-2-[[4-[(2,4-diaminopteridin-6-yl)methyl-methylamino]benzoyl]amino]-5-oxopentanoic acid | —— | C32H42N12O6S |
| —— | 5-[(3aS,4R,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[2-[2-[2-[2-[2-[2-[5-[(3aR,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethyl]pentanamide | —— | C32H56N6O9S2 |
| —— | 5-[(3aS,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[2-[2-[2-[2-[2-[2-[5-[(3aS,4R,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethyl]pentanamide | —— | C32H56N6O9S2 |
| —— | 6-[6-[5-[(3aR,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]hexanoylamino]-N-[6-(2-methylsulfonylsulfanylethylamino)-6-oxohexyl]hexanamide | —— | C31H56N6O7S3 |
| —— | (2R)-2-[6-[5-[(3aS,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]hexanoylamino]-3-methylsulfonylsulfanylpropanoic acid | —— | C20H34N4O7S3 |
| —— | (2S)-2-[6-[5-[(3aS,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]hexanoylamino]-3-methylsulfonylsulfanylpropanoic acid | —— | C20H34N4O7S3 |
| —— | prop-2-enyl N-[9-[2-[5-[(3aR,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]ethylamino]-6-(prop-2-enoxycarbonylamino)acridin-3-yl]carbamate | —— | C33H39N7O6S |
| —— | prop-2-enyl N-[9-[2-[5-[(3aR,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]ethylamino]-6-(prop-2-enoxycarbonylamino)acridin-3-yl]carbamate | —— | C33H39N7O6S |
| —— | prop-2-enyl N-[9-[2-[5-[(3aS,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]ethylamino]-6-(prop-2-enoxycarbonylamino)acridin-3-yl]carbamate | —— | C33H39N7O6S |
| —— | N-[5-[5-[(3aS,4R,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]pentyl]-10-[ethoxy(phenylmethoxy)phosphoryl]decanamide | —— | C34H57N4O6PS |
| —— | N-[5-[5-[(3aS,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]pentyl]-10-[ethoxy(phenylmethoxy)phosphoryl]decanamide | —— | C34H57N4O6PS |
| —— | (2S)-6-[6-[5-[(3aS,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]hexanoylamino]-2-(6-aminohexanoylamino)-N-(2-methylsulfonylsulfanylethyl)hexanamide | —— | C31H57N7O7S3 |
| —— | (2S)-6-[6-[5-[(3aR,4R,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]hexanoylamino]-2-(6-aminohexanoylamino)-N-(2-methylsulfonylsulfanylethyl)hexanamide | —— | C31H57N7O7S3 |
| —— | tert-butyl N-[(2S)-6-[5-[(3aS,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]-1-(2-methylsulfonylsulfanylethylamino)-1-oxohexan-2-yl]carbamate | —— | C24H43N5O7S3 |
| —— | (2S)-6-[6-[5-[(3aR,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]hexanoylamino]-2-(6-aminohexanoylamino)-N-(2-methylsulfonylsulfanylethyl)hexanamide | —— | C31H57N7O7S3 |
| —— | 5-[(3aS,4R,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[2-[2-[2-[2-[2-[2-[5-[(3aR,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethyl]pentanamide | —— | C32H56N6O9S2 |
| —— | N-[5-[5-[(3aS,4R,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]pentyl]-10-[ethoxy(phenylmethoxy)phosphoryl]decanamide | —— | C34H57N4O6PS |
| —— | prop-2-enyl N-[9-[2-[5-[(3aS,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]ethylamino]-6-(prop-2-enoxycarbonylamino)acridin-3-yl]carbamate | —— | C33H39N7O6S |
| —— | 6-[6-[5-[(3aS,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]hexanoylamino]-N-[6-(2-methylsulfonylsulfanylethylamino)-6-oxohexyl]hexanamide | —— | C31H56N6O7S3 |
| —— | (2S)-6-[6-[5-[(3aS,4R,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]hexanoylamino]-2-(6-aminohexanoylamino)-N-(2-methylsulfonylsulfanylethyl)hexanamide | —— | C31H57N7O7S3 |
| —— | N-[5-[5-[(3aS,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]pentyl]-10-[ethoxy(phenylmethoxy)phosphoryl]decanamide | —— | C34H57N4O6PS |
| —— | 5-[(3aS,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[(1R)-2,2-dimethyl-1-[3-(trifluoromethyl)phenyl]propyl]pentanamide | —— | C22H30F3N3O2S |
| —— | 5-[(3aS,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[(1S)-2,2-dimethyl-1-[3-(trifluoromethyl)phenyl]propyl]pentanamide | —— | C22H30F3N3O2S |
| —— | 5-[(3aS,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[(1R)-1-[3-(trifluoromethyl)phenyl]butyl]pentanamide | —— | C21H28F3N3O2S |
| —— | 5-[(3aS,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[(S)-cyclopropyl-[4-(2-methylpropyl)phenyl]methyl]pentanamide | —— | C24H35N3O2S |
| —— | 5-[(3aS,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[(R)-cyclopropyl-[4-(2-methylpropyl)phenyl]methyl]pentanamide | —— | C24H35N3O2S |
| —— | 5-[(3aS,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[(2R)-1-(2,4-dichlorophenyl)propan-2-yl]pentanamide | —— | C19H25Cl2N3O2S |
| —— | 5-[(3aS,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[(2S)-1-(2,4-dichlorophenyl)propan-2-yl]pentanamide | —— | C19H25Cl2N3O2S |
| —— | 5-[(3aS,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[(1S)-1-[3-(difluoromethoxy)phenyl]ethyl]pentanamide | —— | C19H25F2N3O3S |
| —— | 5-[(3aS,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[(1R)-1-[3-(difluoromethoxy)phenyl]ethyl]pentanamide | —— | C19H25F2N3O3S |
| —— | (3aS,4S,6aR)-4-[5-[(2R)-2-(2-methylphenyl)pyrrolidin-1-yl]-5-oxopentyl]-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-2-one | —— | C21H29N3O2S |
| —— | (3aS,4S,6aR)-4-[5-[(2S)-2-(2-methylphenyl)pyrrolidin-1-yl]-5-oxopentyl]-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-2-one | —— | C21H29N3O2S |
| —— | 5-[(3aS,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[4-[[(2S)-2-methylpiperidin-1-yl]methyl]phenyl]pentanamide | —— | C23H34N4O2S |
| —— | 5-[(3aS,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[4-[[(2R)-2-methylpiperidin-1-yl]methyl]phenyl]pentanamide | —— | C23H34N4O2S |
| —— | 5-[(3aS,4R,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[(Z)-(2,3,4,5,6-pentafluorophenyl)methylideneamino]pentanamide | —— | C17H17F5N4O2S |
| —— | (3S)-1-[5-[(3aR,4R,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoyl]-2,5-dioxopyrrolidine-3-sulfonic acid | —— | C14H19N3O7S2 |
| —— | 5-[(3aR,4R,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-(6-hydrazinyl-6-oxohexyl)pentanamide | —— | C16H29N5O3S |
| —— | (3S)-1-[5-[(3aS,4R,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoyl]-2,5-dioxopyrrolidine-3-sulfonic acid | —— | C14H19N3O7S2 |
| —— | 5-[(3aR,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-(5-methyl-1,3,4-thiadiazol-2-yl)pentanamide | —— | C13H19N5O2S2 |
| —— | 5-[(3aR,4R,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-(5-methyl-1,3,4-thiadiazol-2-yl)pentanamide | —— | C13H19N5O2S2 |
| —— | 5-[(3aS,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-(5-methyl-1,3,4-thiadiazol-2-yl)pentanamide | —— | C13H19N5O2S2 |
| —— | [4-[3-[3-[5-[(3aS,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]propyl-methylamino]propylamino]-3-nitrophenyl]imino-methylideneazanium | —— | C24H37N8O4S+ |