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三唑并吡啶类

中文名称 英文名称 CAS号 化学式
—— 1-[5-(difluoromethyl)-1,3,4-thiadiazol-2-yl]-3-[(8S)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]urea —— C12H15F2N7OS
—— 1-[1-(3-cyanopropyl)pyrazol-3-yl]-3-[(8R)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]urea —— C16H22N8O
—— 1-[6-(dimethylamino)pyridin-3-yl]-3-[(8S)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]urea —— C16H23N7O
—— 1-[5-(difluoromethyl)-1,3,4-thiadiazol-2-yl]-3-[(8R)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]urea —— C12H15F2N7OS
—— 1-[(8S)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]-3-(5-propan-2-yl-1,2-oxazol-3-yl)urea —— C15H22N6O2
—— 1-[1-(cyclopropylmethyl)pyrazol-4-yl]-3-[(8R)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]urea —— C16H23N7O
—— 1-[(8R)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]-3-(5-propan-2-yl-1,2-oxazol-3-yl)urea —— C15H22N6O2
—— 1-(3,5-dimethyl-1,2-oxazol-4-yl)-3-[(8R)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]urea —— C14H20N6O2
—— 1-[(8R)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]-3-([1,2,4]triazolo[4,3-a]pyridin-3-yl)urea —— C15H18N8O
—— 1-[6-(dimethylamino)pyridin-3-yl]-3-[(8R)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]urea —— C16H23N7O
—— 1-[(8S)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]-3-(5-propyl-1,3,4-thiadiazol-2-yl)urea —— C14H21N7OS
—— 1-[(8S)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]-3-(2-methyl-1,3-benzoxazol-6-yl)urea —— C17H20N6O2
—— 1-[(8R)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]-3-(5-propyl-1,3,4-thiadiazol-2-yl)urea —— C14H21N7OS
—— N-(7-methyl-[1,2,4]triazolo[4,3-a]pyridin-3-yl)-3,4-dihydro-2H-pyran-6-carboxamide —— C13H14N4O2
—— 1-(2-tert-butylpyrimidin-5-yl)-3-[(8S)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]urea —— C17H25N7O
—— 1-(2-tert-butylpyrimidin-5-yl)-3-[(8R)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]urea —— C17H25N7O
—— 1-(3,5-dimethyl-1,2-oxazol-4-yl)-3-[(8S)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]urea —— C14H20N6O2
—— 1-[1-(3-cyanopropyl)pyrazol-3-yl]-3-[(8S)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]urea —— C16H22N8O
—— 1-[(8R)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]-3-(2-methyl-1,3-benzoxazol-6-yl)urea —— C17H20N6O2
—— 1-[1-(cyclopropylmethyl)pyrazol-4-yl]-3-[(8S)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]urea —— C16H23N7O
—— 3-methyl-N-[[(1'S,3S)-spiro[1,2-dihydroindene-3,2'-cyclopropane]-1'-yl]methyl]-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide —— C20H20N4O
—— 3-methyl-N-[[(1'R,3R)-spiro[1,2-dihydroindene-3,2'-cyclopropane]-1'-yl]methyl]-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide —— C20H20N4O
—— 3-methyl-N-[[(1'R,3S)-spiro[1,2-dihydroindene-3,2'-cyclopropane]-1'-yl]methyl]-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide —— C20H20N4O
—— 3-methyl-N-[[(1'S,3R)-spiro[1,2-dihydroindene-3,2'-cyclopropane]-1'-yl]methyl]-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide —— C20H20N4O
—— 1-[(1R,3S)-3-cyclopropylcyclohexyl]-3-[(8R)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]urea —— C18H29N5O
—— 2-[[8-chloro-6-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]pyridin-3-yl]sulfanyl]-N-[(3S)-1,1-dioxothiolan-3-yl]-N-(2-methylpropyl)acetamide —— C17H20ClF3N4O3S2
—— 1-[(1S,3S)-3-cyclopropylcyclohexyl]-3-[(8R)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]urea —— C18H29N5O
—— 1-[(8S)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]-3-[(1S)-1-(5-methyl-1,3-thiazol-2-yl)propyl]urea —— C16H24N6OS
—— 1-[(8S)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]-3-[3-(4-hydroxyphenyl)propyl]urea —— C18H25N5O2
—— 1-[(1R,3S)-3-cyclopropylcyclohexyl]-3-[(8S)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]urea —— C18H29N5O
—— N-[(8R)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]azocane-1-carboxamide —— C16H27N5O
—— 1-[(8R)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]-3-[(1R)-1-(5-methyl-1,3-thiazol-2-yl)propyl]urea —— C16H24N6OS
—— 1-[(8S)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]-3-[(1R)-1-(5-methyl-1,3-thiazol-2-yl)propyl]urea —— C16H24N6OS
—— 1-[(2R)-4-ethylsulfanylbutan-2-yl]-3-[(8S)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]urea —— C15H27N5OS
—— 1-[(8R)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]-3-[(1S)-1-(5-methyl-1,3-thiazol-2-yl)propyl]urea —— C16H24N6OS
—— 1-[(1S,3S)-3-cyclopropylcyclohexyl]-3-[(8S)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]urea —— C18H29N5O
—— 1-[(8R)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]-3-[(2R)-2-thiophen-3-ylpropyl]urea —— C16H23N5OS
—— N-[(8S)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]azocane-1-carboxamide —— C16H27N5O
—— 1-[(8R)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]-3-[3-(4-hydroxyphenyl)propyl]urea —— C18H25N5O2
—— 1-[(1S,2R)-2-cyclohexylcyclopropyl]-3-[(8R)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]urea —— C18H29N5O
—— 1-[(8S)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]-3-[(2R)-2-thiophen-3-ylpropyl]urea —— C16H23N5OS
—— 1-[(8S)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]-3-[2-(6-methylpyridin-3-yl)ethyl]urea —— C17H24N6O
—— 1-[(8S)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]-3-[(2S)-2-thiophen-3-ylpropyl]urea —— C16H23N5OS
—— 1-[(8R)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]-3-[(1R)-1-(1-propan-2-ylpyrazol-4-yl)ethyl]urea —— C17H27N7O
—— 1-[(8S)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]-3-(4-imidazol-1-ylbutyl)urea —— C16H25N7O
—— 1-[(8S)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]-3-[(1R)-1-(5-methyl-1,2,4-oxadiazol-3-yl)propyl]urea —— C15H23N7O2
—— 1-[(2R)-4-ethylsulfanylbutan-2-yl]-3-[(8R)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]urea —— C15H27N5OS
—— 1-[(8R)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]-3-[(2S)-2-thiophen-2-ylpropyl]urea —— C16H23N5OS
—— 1-[(2,4-dimethyl-1,3-thiazol-5-yl)methyl]-3-[(8R)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]urea —— C15H22N6OS
—— 1-[(2,4-dimethyl-1,3-thiazol-5-yl)methyl]-3-[(8S)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]urea —— C15H22N6OS